5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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SB 243213 dihydrochloride
CAS:1780372-25-9
SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H21Cl2F3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
501.33
Ref: TM-T12859L
| 1mg | 108.00 € | ||
| 5mg | 314.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Tipindole
CAS:7489-66-9
Tipindole is a serotonin antagonist utilized in research related to depression.
Formula:
C16H20N2O2S
Color and Shape:
Liquid
Molecular weight:
304.41
Ref: TM-T201819
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Etoperidone
CAS:52942-31-1
Etoperidone is an antidepressant that acts as an orally active reuptake inhibitor for serotonin (serotonin) …
Formula:
C19H28ClN5O
Color and Shape:
Liquid
Molecular weight:
377.91
Ref: TM-T201838
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
ASP-2205
CAS:1334440-09-3
ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), …
Formula:
C19H28N2O
Color and Shape:
Liquid
Molecular weight:
300.44
Ref: TM-T201450
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
YM-31636 free base
CAS:159081-22-8
YM-31636 (free base) is an orally active, potent, and selective agonist of the 5-HT3 receptor …
Formula:
C14H11N3S
Color and Shape:
Liquid
Molecular weight:
253.32
Ref: TM-T201587
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| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Tiprenolol hydrochloride
CAS:13379-87-8
Tiprenolol hydrochloride is a β-adrenoceptor (β-adrenoceptor) antagonist. This compound is effective in eliminating ventricular arrhythmias …
Formula:
C13H22ClNO2S
Color and Shape:
Liquid
Molecular weight:
291.84
Ref: TM-T201760
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| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
AAZ-A 154
CAS:2481740-94-5
AAZ-A 154 is a selective, competitive, and non-hallucinogenic antagonist of the 5-HT2AR. It promotes neuronal …
Formula:
C14H20N2O
Color and Shape:
Liquid
Molecular weight:
232.32
Ref: TM-T200737
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| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
AAZ-A 154 benzoate
CAS:2930845-92-2
AAZ-A 154 benzoate is a selective, competitive, and non-hallucinogenic 5-HT2AR antagonist. This compound facilitates neuronal …
Formula:
C21H26N2O3
Color and Shape:
Liquid
Molecular weight:
354.44
Ref: TM-T200491
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
SB-224289 hydrochloride
CAS:180084-26-8
SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
Formula:
C32H33ClN4O3
Purity:
97.82% - 98.09%
Color and Shape:
Solid
Molecular weight:
557.08
Ref: TM-T12841
| 5mg | 97.00 € | ||
| 10mg | 146.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
AAZ-A 154 mesylate
CAS:2930846-03-8
AAZ-A 154 mesylate mesylate is a selective, competitive, and non-hallucinogenic antagonist of 5-HT2AR. It enhances …
Formula:
C15H24N2O4S
Color and Shape:
Liquid
Molecular weight:
328.43
Ref: TM-T200486
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Elzasonan hydrochloride
CAS:220322-05-4
Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in …
Formula:
C22H24Cl3N3OS
Color and Shape:
Liquid
Molecular weight:
484.87
Ref: TM-T201763
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
F 14679
CAS:208109-38-0
F 14679 is a potent 5-HT1A agonist (pKi=10.23) with a maximum Ca2t response similar to …
Formula:
C21H25ClF2N4O
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
422.9
Ref: TM-T62269
| 25mg | 1,264.00 € | ||
| 50mg | 1,641.00 € | ||
| 100mg | 2,465.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
SB 243213 hydrochloride
CAS:200940-23-4
SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H20ClF3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
464.87
Ref: TM-T12859
| 25mg | 2,157.00 € | ||
| 50mg | 2,832.00 € | ||
| 100mg | 3,800.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Flucopride
CAS:1639925-34-0
Flucopride (Compound 4a) acts as an acetylcholinesterase inhibitor (AChE) with an IC50 value of 24 …
Formula:
C22H33FN2O2
Color and Shape:
Liquid
Molecular weight:
376.51
Ref: TM-T201815
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
R-137696
CAS:695185-73-0
R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal …
Formula:
C17H23N3O2
Color and Shape:
Liquid
Molecular weight:
301.38
Ref: TM-T201501
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Befiradol hydrochloride
CAS:2436760-81-3
Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 …
Formula:
C20H23Cl2F2N3O
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
430.32
Ref: TM-T62385
| 1mg | 149.00 € | ||
| 2mg | 213.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 525.00 € | ||
| 25mg | 847.00 € | ||
| 50mg | 1,169.00 € | ||
| 100mg | 1,568.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Sulamserod
CAS:219757-90-1
Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study …
Formula:
C19H28ClN3O5S
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
445.96
Ref: TM-T13021
| 25mg | 2,300.00 € | ||
| 50mg | 3,022.00 € | ||
| 100mg | 4,085.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
Remlifanserin
CAS:2289704-13-6
Remlifanserin is a potent inverse agonist of the serotonin receptor (5-HT2A).
Formula:
C24H29F2N3O2
Color and Shape:
Liquid
Molecular weight:
429.50
Ref: TM-T201055
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Jul 2025
5-HT2A/5-HT2C inverse agonist 1
CAS:2718990-76-0
5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A …
Formula:
C24H35N5O2
Color and Shape:
Liquid
Molecular weight:
425.57
Ref: TM-T200089
| 10mg | To inquire | ||
| 25mg | 2,372.00 € | ||
| 50mg | 3,117.00 € | ||
| 100mg | 4,215.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.
Formula:
C24H33BrN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.44
Ref: TM-T10294
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 15 Jul 2025
