5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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5-HT3 antagonist 3
CAS:120635-47-4
5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 …
Formula:
C20H21N3O
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
319.4
Ref: TM-T10162
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 22 Jan 2025
(±)-Fabesetron hydrochloride
CAS:129299-81-6
FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.
Formula:
C18H20ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.82
Ref: TM-T11293
| 25mg | 1,827.00 € | ||
| 50mg | 2,413.00 € | ||
| 100mg | 3,180.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2A receptor agonist-3
CAS:1391499-52-7
5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting …
Formula:
C21H26BrNO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
420.34
Ref: TM-T79155
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
WAY-607695
CAS:380469-52-3
WAY-607695 is a potential 5-HT1A receptor agonist.
Formula:
C13H12FNO2
Purity:
99.82%
Color and Shape:
Liquid
Molecular weight:
233.24
Ref: TM-T80805
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 214.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Wf-516
CAS:310392-94-0
Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor …
Formula:
C25H25Cl2N3O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
502.39
Ref: TM-T13339
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT3-In-1
CAS:186348-68-5
5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.
Formula:
C16H21ClN4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.82
Ref: TM-T10006
| 25mg | 1,827.00 € | ||
| 50mg | 2,404.00 € | ||
| 100mg | 3,168.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2A antagonist 1
CAS:204643-75-4
5-HT2A antagonist 1, from US5728835A & JP 1007727, may treat gastrointestinal and circulatory issues.
Formula:
C26H28N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
428.53
Ref: TM-T10498
| 25mg | 1,406.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
SB 216641 hydrochloride
CAS:193611-67-5
SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.
Formula:
C28H31ClN4O4
Purity:
98.40%
Color and Shape:
Solid
Molecular weight:
523.02
Ref: TM-T23315
| 1mg | 74.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 395.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 817.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Gepirone
CAS:83928-76-1
Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater …
Formula:
C19H29N5O2
Purity:
99.35% - 99.77%
Color and Shape:
Solid
Molecular weight:
359.47
Ref: TM-T19917
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 137.00 € | ||
| 50mg | 201.00 € | ||
| 100mg | 276.00 € | ||
| 500mg | 684.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Osemozotan HCl
CAS:137275-80-0
Osemozotan is a 5-HT1A receptor agonist potentially for the treatment of generalized anxiety disorder.
Formula:
C19H22ClNO5
Purity:
98.87% - 99.63%
Color and Shape:
Solid
Molecular weight:
379.84
Ref: TM-T28270
| 1mg | 350.00 € | ||
| 5mg | 837.00 € | ||
| 10mg | 1,144.00 € | ||
| 25mg | 1,688.00 € | ||
| 50mg | 2,287.00 € | ||
| 100mg | 3,061.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Brilaroxazine
CAS:1239729-06-6
Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.
Formula:
C22H25Cl2N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
450.36
Ref: TM-T14782
| 1mg | 104.00 € | ||
| 5mg | 247.00 € | ||
| 10mg | 402.00 € | ||
| 25mg | 692.00 € | ||
| 50mg | 994.00 € | ||
| 100mg | 1,360.00 € | ||
| 500mg | 2,678.00 € | ||
| 1mL*10mM (DMSO) | 363.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
YM348
CAS:372163-84-3
YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high …
Formula:
C14H17N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
243.3
Ref: TM-T17275
| 25mg | 1,299.00 € | ||
| 50mg | 1,723.00 € | ||
| 100mg | 2,670.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Flesinoxan
CAS:98206-10-1
Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor …
Formula:
C22H26FN3O4
Color and Shape:
Solid
Molecular weight:
415.46
Ref: TM-T16711
| 5mg | 349.00 € | ||
| 25mg | 1,113.00 € | ||
| 50mg | 1,470.00 € | ||
| 100mg | 2,209.00 € | ||
| 1mL*10mM (DMSO) | 431.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
4-Chloro-L-phenylalanine
CAS:14173-39-8
4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases …
Formula:
C9H10ClNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
199.63
Ref: TM-T78228
| 5g | 51.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Facinicline hydrochloride
CAS:677305-02-1
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = …
Formula:
C15H19ClN4O
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
306.79
Ref: TM-T28531
| 1mg | 52.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 404.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2C agonist-3 free base
CAS:2104810-17-3
5-HT2C agonist-3 ((+)-19) free base, a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), …
Formula:
C19H22FNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
315.38
Ref: TM-T79803
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
(S)-Bexicaserin
CAS:2035818-21-2
(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and …
Formula:
C15H19F2N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
295.33
Ref: TM-T79838
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2A&5-HT2C agonist-1
CAS:1640-02-4
5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with …
Formula:
C14H20N2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
232.32
Ref: TM-T79806
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Gentisein
CAS:529-49-7
Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency …
Formula:
C13H8O5
Purity:
96.74%
Color and Shape:
Solid
Molecular weight:
244.2
Ref: TM-T19931
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 254.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2 agonist-1
CAS:2708279-78-9
Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values …
Formula:
C19H23ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
346.85
Ref: TM-T79804
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
