Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Found 729 products of "Adrenergic Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ancarolol
CAS:Ancarolol is a blocking agent of beta-adrenergic.Formula:C18H24N2O4Purity:98%Color and Shape:SolidMolecular weight:332.39Rec 15/2615 dihydrochloride
CAS:Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.Formula:C26H35Cl2N5O5Purity:97.04% - 99.76%Color and Shape:SolidMolecular weight:568.49Arbutamine
CAS:<p>Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.</p>Formula:C18H23NO4Purity:95.06%Color and Shape:SolidMolecular weight:317.38(S)-(-)-Propranolol hydrochloride
CAS:(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。Formula:C16H22ClNO2Purity:99.02% - 99.91%Color and Shape:SolidMolecular weight:295.8(S)-Terazosin
CAS:(S)-Terazosin is an active S-enantiomer of Terazosin.Formula:C19H25N5O4Color and Shape:SolidMolecular weight:387.43T-0509
CAS:<p>T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-</p>Formula:C18H23NO5Purity:97.52% - 98.43%Color and Shape:SolidMolecular weight:333.38Cyclazosin HCl
CAS:Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formula:C23H28ClN5O4Purity:99.10%Color and Shape:SolidMolecular weight:473.95Levobunolol hydrochloride
CAS:Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。Formula:C17H26ClNO3Purity:98.49% - >99.99%Color and Shape:SolidMolecular weight:327.85L748337
CAS:L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formula:C26H31N3O5SPurity:99.67% - >99.99%Color and Shape:SolidMolecular weight:497.61ADRA1D receptor antagonist 1 HCl
CAS:ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activity.Formula:C15H14Cl2N4OPurity:98.13%Color and Shape:SolidMolecular weight:337.2Romifidine
CAS:Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Formula:C9H9BrFN3Color and Shape:SolidMolecular weight:258.09LY377604
CAS:LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.Formula:C31H32N4O4Purity:99.72% - >99.99%Color and Shape:SolidMolecular weight:524.61SM-2470
CAS:SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.Formula:C23H30ClN5O3Purity:98.91%Color and Shape:SolidMolecular weight:459.97Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purity:97.15% - 98.85%Color and Shape:SolidMolecular weight:251.33Rezatomidine
CAS:Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.Formula:C13H16N2SPurity:98.34%Color and Shape:SolidMolecular weight:232.34Bedoradrine
CAS:Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5Purity:>99.99%Color and Shape:SolidMolecular weight:428.52Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formula:C17H26FNO3Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:311.392Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formula:C14H20N4OPurity:98.58% - 99.53%Color and Shape:SolidMolecular weight:260.33Imiloxan
CAS:Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formula:C14H16N2O2Purity:98.13% - 99.8%Color and Shape:SolidMolecular weight:244.29Bedoradrine sulfate
CAS:Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5H2O4SPurity:99.31%Color and Shape:SolidMolecular weight:477.56ORM-10921
CAS:ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formula:C18H23NO2Purity:99.46% - 99.98%Color and Shape:SolidMolecular weight:285.38Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg369.00€5mg735.00€10mg938.00€25mg1,473.00€50mg1,882.00€100mg2,670.00€1mL*10mM (DMSO)929.00€JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formula:C24H24N4Purity:99.96%Color and Shape:SolidMolecular weight:368.47Oxyfedrine L-form HCl
CAS:Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Formula:C19H24ClNO3Purity:99.5% - 99.57%Color and Shape:SolidMolecular weight:349.85Ref: TM-T24579
1mg96.00€5mg188.00€10mg329.00€25mg512.00€50mg740.00€100mg944.00€200mg1,264.00€1mL*10mM (DMSO)215.00€Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Formula:C18H25N5O4Purity:99.76% - 99.97%Color and Shape:SolidMolecular weight:375.42Soquinolol
CAS:Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a longFormula:C17H26N2O3Purity:97.48% - 98.63%Color and Shape:SolidMolecular weight:306.4Midaglizole hydrochloride
CAS:Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formula:C16H19Cl2N3Purity:99.39% - 99.82%Color and Shape:SolidMolecular weight:324.25Ref: TM-T11015
1mg57.00€5mg126.00€10mg198.00€25mg324.00€50mg439.00€100mg562.00€200mg743.00€1mL*10mM (DMSO)160.00€Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formula:C10H11Cl2N3Purity:98.06% - 98.83%Color and Shape:SolidMolecular weight:244.12GP2-114
CAS:GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.Formula:C19H24N2O4Purity:99.32%Color and Shape:SolidMolecular weight:344.4Vadocaine
CAS:Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formula:C18H28N2O2Purity:99.7%Color and Shape:SolidMolecular weight:304.43ST 91
CAS:ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formula:C13H20ClN3Purity:99.83%Color and Shape:SolidMolecular weight:253.77Ref: TM-T23397
5mg52.00€10mg75.00€25mg150.00€50mg259.00€100mg374.00€200mg525.00€1mL*10mM (DMSO)52.00€Fipamezole
CAS:Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.Formula:C14H15FN2Purity:99.32% - 99.97%Color and Shape:SolidMolecular weight:230.28Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Formula:C15H22N2O2Purity:98.55%Color and Shape:SolidMolecular weight:262.35(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purity:98.27%Color and Shape:SolidMolecular weight:646.17Milveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formula:C25H30ClN3O4Purity:99.9%Color and Shape:SolidMolecular weight:471.98Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formula:C18H24N2O5SPurity:99.5%Color and Shape:SolidMolecular weight:380.46Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formula:C19H21ClFN5O2Purity:97.49% - >99.99%Color and Shape:SolidMolecular weight:405.85Taprizosin
CAS:Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Formula:C25H26N6O4SPurity:98.10% - 99.11%Color and Shape:SolidMolecular weight:506.58Bisaramil hydrochloride
CAS:Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.Formula:C17H24Cl2N2O2Purity:98.64% - 99.48%Color and Shape:SolidMolecular weight:359.29Palatrigine
CAS:Palatrigine (BW-A 256C) is a compound with angiotensin-converting enzyme inhibitory and beta-adrenergic receptor blocking properties.Formula:C12H13Cl2N5Purity:98.87%Color and Shape:SolidMolecular weight:298.17CL 316243
CAS:CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formula:C20H18ClNNa2O7Purity:98.00% - 99.68%Color and Shape:SolidMolecular weight:465.79Xamoterol hemifumarate
CAS:Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormula:C36H54N6O14Purity:99.79%Color and Shape:White SolidMolecular weight:794.37Rafabegron
CAS:Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formula:C21H23ClN2O4Purity:99.81%Color and Shape:SolidMolecular weight:402.87Prenalterol hydrochloride
CAS:Prenalterol HCl: beta 1-specific agonist; treats acute cardiac failure, shock, low-output post-MI, Shy-Drager syndrome.Formula:C12H20ClNO3Color and Shape:SolidMolecular weight:261.75RS 17053 hydrochloride
CAS:RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formula:C24H30Cl2N2O2Purity:99.27%Color and Shape:SolidMolecular weight:449.41AR-08
CAS:<p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>Formula:C12H12N6Purity:99.7%Color and Shape:SolidMolecular weight:240.26Mefenidil
CAS:Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.Formula:C12H11N3Purity:98.27%Color and Shape:SolidMolecular weight:197.24Nolomirole HCl
CAS:Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory effects on norepinephrine release, which can be used to studyFormula:C19H28ClNO4Purity:99.03% - >99.99%Color and Shape:SolidMolecular weight:369.88(±)-N-Methylcoclaurine
CAS:N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].Formula:C18H21NO3Purity:98%Color and Shape:SolidMolecular weight:299.36BU-E 75
CAS:BU-E 75 is an agonist of the histamine H2.Formula:C21H24F2N6Color and Shape:SolidMolecular weight:398.45RS100329 hydrochloride
CAS:RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.Formula:C20H26ClF3N4O3Purity:99.95%Color and Shape:SolidMolecular weight:462.89L-796568 free base
CAS:L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formula:C31H27F3N4O3S2Color and Shape:SolidMolecular weight:624.7LK 204-545
CAS:LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.Formula:C25H32N4O6Color and Shape:SolidMolecular weight:484.54Vatinoxan hydrochloride
CAS:Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.Formula:C20H27ClN4O4SPurity:98%Color and Shape:SolidMolecular weight:454.97NGD9002
CAS:NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.Formula:C20H31N5OPurity:98%Color and Shape:SolidMolecular weight:357.49Domesticine, (-)-
CAS:Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.Formula:C19H19NO4Purity:98%Color and Shape:SolidMolecular weight:325.36GW-597901
CAS:GW-597901, an β2 adrenergic receptor agonist, is used potentially for the treatment of asthma and chronic obstructive.Formula:C25H38N2O6SColor and Shape:SolidMolecular weight:494.64Epinephrine HCl
CAS:Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formula:C9H14ClNO3Purity:99.48%Color and Shape:SolidMolecular weight:219.67KUC-7322
CAS:Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.Formula:C21H27NO5Color and Shape:SolidMolecular weight:373.44Vemtoberant
CAS:Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.Formula:C29H37N3O8S2Color and Shape:SolidMolecular weight:619.75Abediterol
CAS:Abediterol (LAS100977): potent, long-acting beta-2 agonist for asthma and COPD treatment.Formula:C25H30F2N2O4Color and Shape:SolidMolecular weight:460.51BMS-194449
CAS:BMS-194449 is a full beta 3 agonist.Formula:C24H24F4N2O6SColor and Shape:SolidMolecular weight:544.52β3-AR agonist 1
CAS:β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/Formula:C22H28N4O4SPurity:98%Color and Shape:SolidMolecular weight:444.55L-796568 dihydrochloride
CAS:L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.Formula:C31H29Cl2F3N4O3S2Color and Shape:SolidMolecular weight:697.62Ritodrine
CAS:Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].Formula:C17H21NO3Color and Shape:SolidMolecular weight:287.35Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purity:98%Color and Shape:SolidMolecular weight:293.41Dibenamine hydrochloride
CAS:<p>Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.</p>Formula:C16H19Cl2NPurity:96.43%Color and Shape:Oily Liquid SolidMolecular weight:296.23Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurity:99.73%Color and Shape:SolidMolecular weight:555.65Pronetalol
CAS:Pronethalol ((±)-Pronethalol), a non-selective β-adrenergic antagonist, effectively inhibits Sox2 expression and offers protection against Digitalis-induced ventricular arrhythmias. Additionally, it can reverse such arrhythmias and limit the development of cerebral arteriovenous malformations (AVMs) [1] [2].Formula:C15H19NOColor and Shape:SolidMolecular weight:229.32SDZ-NVI-085
CAS:SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formula:C15H21NO2SColor and Shape:SolidMolecular weight:279.4Lidamidine
CAS:Lidamidine (Lidamidinum) is an effective antidiarrheal agent that inhibits intestinal secretion, reduces intestinal transit, and inhibits smooth muscleFormula:C11H16N4OPurity:99.98%Color and Shape:SolidMolecular weight:220.27Ref: TM-T25719
1mg115.00€2mg162.00€5mg249.00€10mg369.00€25mg562.00€50mg787.00€100mg1,054.00€200mg1,406.00€Ro-70-0004
CAS:Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formula:C20H24F4N4O3Color and Shape:SolidMolecular weight:444.42Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurity:99.96%Color and Shape:SolidMolecular weight:281.35Ref: TM-T12444
1mg86.00€5mg172.00€10mg259.00€25mg425.00€50mg598.00€100mg810.00€200mg1,074.00€1mL*10mM (DMSO)172.00€Bunazosin Hydrochloride
CAS:Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formula:C19H28ClN5O3Purity:99.12%Color and Shape:SolidMolecular weight:409.91N-5984
CAS:<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formula:C20H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:391.854-hydroxy Nebivolol hydrochloride
CAS:4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.Formula:C22H25F2NO5HClColor and Shape:SolidMolecular weight:457.9(-)-Isoproterenol hydrochloride
CAS:(-)-Isoproterenol hydrochloride is used as a β-adrenergic receptor agonist in the treatment of bradycardia and as a bronchodilator.Formula:C11H17NO3·CIHColor and Shape:SolidMolecular weight:247.72BI-167107
CAS:BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR, Kd of 84 pM).Formula:C21H26N2O4Color and Shape:SolidMolecular weight:370.44AGN 192836
CAS:AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).Formula:C12H13N3O2Color and Shape:SolidMolecular weight:231.25β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formula:C27H38N4O7SPurity:98%Color and Shape:SolidMolecular weight:562.68Bufuralol (hydrochloride)
CAS:Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Formula:C16H24ClNO2Color and Shape:SolidMolecular weight:297.82Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Formula:C11H13ClN4O2Purity:99.91%Color and Shape:SolidMolecular weight:268.7Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColor and Shape:White Crystalline SolidMolecular weight:415.96Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Formula:C16H23NO2Purity:98.26%Color and Shape:SolidMolecular weight:261.36Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColor and Shape:SolidMolecular weight:592.11N-5984 Hydrochloride
CAS:N-5984 Hydrochloride is a beta3-AR agonist.Formula:C20H23Cl2NO5Color and Shape:SolidMolecular weight:428.31Indacaterol xinafoate
CAS:Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C35H36N2O6Color and Shape:SolidMolecular weight:580.67Indacaterol acetate
CAS:Indacaterol acetate is an ultra-long-acting beta-adrenoceptor agonist.Formula:C26H32N2O5Color and Shape:SolidMolecular weight:452.54Talibegron hydrochloride
CAS:Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.Formula:C18H22ClNO4Purity:99.82%Color and Shape:SolidMolecular weight:351.83Deriglidole
CAS:Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.Formula:C16H21N3Purity:98.12% - 99.03%Color and Shape:SolidMolecular weight:255.36CGP-20712
CAS:CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.Formula:C23H25F3N4O5Purity:99.40% - 99.58%Color and Shape:SolidMolecular weight:494.46Ref: TM-T30846
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€0990CL
CAS:0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMPFormula:C21H21N5Purity:98.99%Color and Shape:SolidMolecular weight:343.42Ref: TM-T13983
1mg202.00€5mg512.00€10mg740.00€25mg1,121.00€50mg1,539.00€100mg2,072.00€1mL*10mM (DMSO)535.00€α1 adrenoceptor-MO-1
CAS:α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action.Formula:C20H24ClN5OPurity:99.20% - 99.29%Color and Shape:SolidMolecular weight:385.89Ref: TM-T10003
1mg198.00€5mg393.00€10mg542.00€25mg785.00€50mg1,074.00€100mg1,454.00€200mg1,967.00€1mL*10mM (DMSO)467.00€OPC-28326
CAS:OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.Formula:C26H35N3O2Purity:99.79%Color and Shape:SolidMolecular weight:421.58Ref: TM-T13804
1mg187.00€5mg455.00€10mg620.00€25mg940.00€50mg1,264.00€100mg1,663.00€200mg2,252.00€1mL*10mM (DMSO)567.00€(±)-Prenalterol
CAS:(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.Formula:C12H19NO3Purity:99.73%Color and Shape:SolidMolecular weight:225.28Teoprolol
CAS:Teoprolol is a blocker of β-adrenergic receptor.Formula:C23H30N6O4Purity:98%Color and Shape:SolidMolecular weight:454.52LK 11
CAS:LK-11, an alkaloid derivative, inhibits the passive uptake of norepinephrine (NA) by synaptic vesicles in the thalamus, similarly to cocaine.Formula:C15H26N2O3Color and Shape:SolidMolecular weight:282.38(±)-Penbutolol
CAS:(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic receptor antagonist. (±)-Penbutolol mitigates the tachycardia induced by exercise, reduces the increase in peak expiratory flow rate (PEFR) caused by physical activity, and decreases plasma renin activity (PRA) at rest. The peak plasma concentration of this compound is achieved one hour after oral administration, with a half-life of 4.5 hours, and it is metabolized into active metabolites in the body. This compound is utilized in research related to cardiovascular diseases.Formula:C18H29NO2Color and Shape:SolidMolecular weight:291.43Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Formula:C26H28N4O3Color and Shape:SolidMolecular weight:444.53Nipradolol
CAS:Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.Formula:C15H22N2O6Color and Shape:SolidMolecular weight:326.35Sulfinalol hydrochloride
CAS:Sulfinalol hydrochloride is an orally active β-adrenoceptor (β-adrenoceptor) antagonist that exhibits direct vasodilatory activity. It is also classified as an antihypertensive agent.Formula:C20H28ClNO4SColor and Shape:SolidMolecular weight:413.96TAAR1 agonist 3
CAS:TAAR1 agonist 3 is a potent agonist of Trace Amine-Associated Receptor 1 (TAAR1) with a pEC50 value of 7.6. Additionally, it acts as a full agonist at the α2AR with a pEC50 of 6. TAAR1 agonist 3 is utilized in the research of neuropsychiatric disorders.Formula:C10H13NOColor and Shape:SolidMolecular weight:163.22Metrazoline
CAS:<p>Metrazoline (o-Methyl-tracizoline) acts as a ligand for adrenergic receptors (low affinity) and imidazoline I2 receptors.</p>Formula:C14H16N2O4Color and Shape:SolidMolecular weight:276.288PF-9404C
CAS:PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.Formula:C16H25N3O9Purity:98%Color and Shape:SolidMolecular weight:403.38SAR-150640
CAS:SAR-150640, a selective β3-adrenergic receptor agonist, prevents an increase in MMP activity and production observed after LPS stimulation or in cases of chorioamnionitis.Formula:C25H35ClN2O7SColor and Shape:SolidMolecular weight:543.07Ersentilide
CAS:Ersentilide, a benzamide derivative, functions as both a β1-adrenergic receptor antagonist and an Ikr blocker. It has demonstrated efficacy in animal models of cardiac arrhythmias.Formula:C21H26N4O5SColor and Shape:SolidMolecular weight:446.52Carazolol hydrochloride
CAS:Carazolol (BM 51052) hydrochloride is a potent antagonist of β1/β2-adrenoceptors and also serves as a powerful and selective agonist of β3-adrenoceptors. It is utilized in research focusing on hypertension.Formula:C18H23ClN2O2Molecular weight:334.84Anti-MRSA agent 19
CAS:Anti-MRSA agent 19 (Compound 1) is an antibiotic that exhibits activity against Staphylococcus aureus. It is active against 40 clinical isolates from the CDC, representing diverse bacterial species with various resistance factors, including resistance to vancomycin, aminoglycoside/tetracycline, and oxazolidinone (median MIC=4 μg/mL).Formula:C15H10Cl3NO4Color and Shape:SolidMolecular weight:374.6(S)-Bucindolol
CAS:(S)-Bucindolol is an enantiomer of bucindolol, specifically a β1-adrenergic receptor antagonist. It is primarily utilized in research related to heart failure.Formula:C22H25N3O2Color and Shape:SolidMolecular weight:363.45Mafoprazine
CAS:Mafoprazine, a phenylpiperazine derivative, exhibits varying affinities for neuronal receptors, primarily exerting its antipsychotic effects through blocking D2 receptors and enhancing α-adrenergic activity. It also increases the activity of dopamine metabolites.Formula:C22H28FN3O3Color and Shape:SolidMolecular weight:401.472,3-MDMA hydrochloride
CAS:2,3-MDMA hydrochloride is an inhibitor of the noradrenalin transporter and serotonin transporter, with IC50 values of 6.2 μM and 82 μM, respectively.Formula:C11H16ClNO2Molecular weight:229.703RU 52583
CAS:RU 52583 is an alpha 2-adrenergic receptor antagonist.Formula:C18H20N2Purity:98%Color and Shape:SolidMolecular weight:264.36Org-6906
CAS:DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.Formula:C13H16ClNPurity:98%Color and Shape:SolidMolecular weight:221.73Meluadrine
CAS:Meluadrine, a potent agonist of the β2 adrenergic receptor, is one of the metabolites of Tulobuterol [1].Formula:C12H18ClNO2Molecular weight:243.73L-654284
CAS:L-654284 is an α2-adrenergic receptor antagonist characterized by its notable selectivity. It competes with 3H-clonidine and 3H-rauwolscine for binding in vitro, exhibiting Ki values of 0.8 nM and 1.1 nM, respectively. L-654284 effectively blocks the pre-ejaculatory effects of clonidine in isolated rat vas deferens, with a pA2 value of 9.1. The compound demonstrates significant selectivity for α2 over α1 adrenergic receptors, with a Ki value of 110 nM against 3H-prazosin binding. In vivo, L-654284 significantly increases the turnover of norepinephrine in the rat cerebral cortex, indicating its activity in blocking α2-adrenergic receptors within the central nervous system.Formula:C18H24N2O4SColor and Shape:SolidMolecular weight:364.46Aclidinium
CAS:Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, exhibiting bronchodilator properties. It effectively reduces lung hyperinflation, enhances lung function, and prolongs exercise endurance time. This compound is commonly utilized in studies focusing on chronic obstructive pulmonary disease (COPD).Formula:C26H30NO4S2Color and Shape:SolidMolecular weight:484.65Bometolol Hydrochloride
CAS:Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.Formula:C25H33ClN2O7Purity:98%Color and Shape:SolidMolecular weight:508.99Butopamine hydrochloride
CAS:Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart rate compared to Dobutamine.Formula:C18H24ClNO3Color and Shape:SolidMolecular weight:337.84(Rac)-Nebivolol
CAS:(Rac)-Nebivolol, a racemic β1-adrenergic blocker (IC50=0.8 nM), has vasodilatory properties and mitigates ethanol-induced cardiac harm.Formula:C22H25F2NO4Color and Shape:SolidMolecular weight:405.43BRL-37344
CAS:<p>BRL-37344 is a selective β3-adrenergic receptor agonist. It significantly reduces the body weight of obese mice.</p>Formula:C19H22ClNO4Color and Shape:SolidMolecular weight:363.84AA 497 (Free Base)
CAS:AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.Formula:C14H21NO3Purity:98%Color and Shape:SolidMolecular weight:251.32HOKU-81
CAS:HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.Formula:C12H18ClNO2Color and Shape:SolidMolecular weight:243.73N-methyl-2-AI (hydrochloride)
CAS:N-methyl-2-AI (hydrochloride) is a useful organic compound for research related to life sciences. The catalog number is T66396 and the CAS number is 10408-85-2.Formula:C10H14ClNColor and Shape:SolidMolecular weight:183.68SKF 89748
CAS:SKF 89748 is an agonists of alpha 1-adrenoceptor.Formula:C12H17NOSPurity:98%Color and Shape:SolidMolecular weight:223.334-Hydroxypropranolol hydrochloride
CAS:4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).Formula:C16H22ClNO3Purity:98%Color and Shape:SolidMolecular weight:311.8Picumeterol
CAS:<p>Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth muscle relaxation. Picumeterol is a pure R enantiomer that can be used to improve lung function and reduce airway hyperreactivity in patients with asthma.</p>Formula:C21H29Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:426.384-Hydroxyatomoxetine
CAS:4-Hydroxyatomoxetine, an active metabolite of Atomoxetine, is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.Formula:C17H21NO2Purity:98%Color and Shape:SolidMolecular weight:271.351-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol
CAS:1-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol is a useful organic compound for research related to life sciences. The catalog number is T65156 and the CAS number is 24155-42-8.Formula:C11H10Cl2N2OColor and Shape:SolidMolecular weight:257.11SB251023
CAS:SB251023 is an agonist of β3-adrenoceptor.Formula:C28H34NO6PColor and Shape:SolidMolecular weight:511.55
