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Adrenergic Receptor

Adrenergic Receptor

Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.

Subcategories of "Adrenergic Receptor"

Found 717 products of "Adrenergic Receptor"

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  • Celiprolol hydrochloride

    CAS:
    Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.
    Formula:C20H33N3O4·HCl
    Color and Shape:White Crystalline Solid
    Molecular weight:415.96
  • Bufuralol (hydrochloride)

    CAS:
    Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.
    Formula:C16H24ClNO2
    Color and Shape:Solid
    Molecular weight:297.82
  • Mefenidil

    CAS:
    Mefenidil (McN-2378), a selective cerebral vasodilator, was shown to increase CBF in healthy brains without stimulating O2 uptake in a dog anesthesia model.
    Formula:C12H11N3
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:197.24
  • Todralazine hydrochloride

    CAS:
    Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.
    Formula:C11H13ClN4O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:268.7
  • RS100329 hydrochloride

    CAS:
    RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.
    Formula:C20H26ClF3N4O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:462.89
  • NGD9002

    CAS:
    NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.
    Formula:C20H31N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:357.49
  • AR-08

    CAS:
    <p>AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.</p>
    Formula:C12H12N6
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:240.26
  • Vatinoxan hydrochloride

    CAS:
    <p>Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.</p>
    Formula:C20H27ClN4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.97
  • BMS-194449

    CAS:
    BMS-194449 is a full beta 3 agonist.
    Formula:C24H24F4N2O6S
    Color and Shape:Solid
    Molecular weight:544.52
  • β3-AR agonist 1

    CAS:
    β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/
    Formula:C22H28N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.55
  • LK 204-545

    CAS:
    LK 204-545 is a highly selective antagonist of beta1-adrenoceptor.
    Formula:C25H32N4O6
    Color and Shape:Solid
    Molecular weight:484.54
  • Bufuralol

    CAS:
    Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.
    Formula:C16H23NO2
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:261.36
  • Vemtoberant

    CAS:
    Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.
    Formula:C29H37N3O8S2
    Color and Shape:Solid
    Molecular weight:619.75
  • L-796568 dihydrochloride

    CAS:
    L-796568: potent β3 agonist (EC50 = 3.6 nM), >600-fold selectivity vs β1/β2, good oral bioavailability, long action.
    Formula:C31H29Cl2F3N4O3S2
    Color and Shape:Solid
    Molecular weight:697.62
  • N-5984

    CAS:
    <p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>
    Formula:C20H22ClNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.85
  • 4-hydroxy Nebivolol hydrochloride

    CAS:
    <p>4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.</p>
    Formula:C22H25F2NO5HCl
    Color and Shape:Solid
    Molecular weight:457.9
  • Ritodrine

    CAS:
    Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].
    Formula:C17H21NO3
    Color and Shape:Solid
    Molecular weight:287.35
  • Binedaline

    CAS:
    Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.
    Formula:C19H23N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.41
  • 0990CL

    CAS:
    0990CL is an effective heterotrimer Gαi subunit specific inhibitor, which can interact with purified Go± in GDP-bound state, and can block α2AR mediated cAMP
    Formula:C21H21N5
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:343.42
  • Talibegron hydrochloride

    CAS:
    Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.
    Formula:C18H22ClNO4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:351.83