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Adrenergic Receptor

Adrenergic Receptor

Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.

Subcategories of "Adrenergic Receptor"

Found 645 products of "Adrenergic Receptor"

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  • Metipranolol

    CAS:
    <p>Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.</p>
    Formula:C17H27NO4
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:309.4
  • Oxaprotiline hydrochloride

    CAS:
    <p>Oxaprotiline hydrochloride is an antidepressant.</p>
    Formula:C20H24ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.86
  • Yohimbine

    CAS:
    <p>Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)</p>
    Formula:C21H26N2O3
    Purity:99.78% - 99.89%
    Color and Shape:Solid
    Molecular weight:354.4
  • Adrenergic Receptor-Targeted Compound Library


    <p>A unique collection of 193 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;</p>
    Color and Shape:Odour Solid
  • Terazosin dimer impurity dihydrochloride

    CAS:
    <p>Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.</p>
    Formula:C24H30Cl2N8O4
    Color and Shape:Solid
    Molecular weight:565.46
  • (±)5(6)-EET

    CAS:
    <p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.473
  • ARC 239 dihydrochloride

    CAS:
    <p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>
    Formula:C24H31Cl2N3O3
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:480.43
  • Abediterol napadisylate

    CAS:
    <p>Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.</p>
    Formula:C60H68F4N4O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1209.32
  • 5-Bromoimidazo[1,2-A]Pyrazine

    CAS:
    <p>5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.</p>
    Formula:C6H4BrN3
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:198.02
  • (R)-(+)-Atenolol

    CAS:
    <p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>
    Formula:C14H22N2O3
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:266.34
  • Metaraminol

    CAS:
    <p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>
    Formula:C9H13NO2
    Color and Shape:Solid
    Molecular weight:167.21
  • S(-)-Bisoprolol fumarate

    CAS:
    <p>S(-)-Bisoprolol fumarate is a selective β1-blocker for hypertension and heart research.</p>
    Formula:C18H31NO4·xC4H4O4
    Color and Shape:Solid
    Molecular weight:441.521
  • Meluadrine tartrate

    CAS:
    <p>Meluadrine tartrate is an endogenous metabolite.</p>
    Formula:C16H24ClNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.82
  • O-Desmethyl Mebeverine alcohol

    CAS:
    <p>Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.</p>
    Formula:C15H25NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:251.36
  • Propranolol hydrochloride

    CAS:
    <p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>
    Formula:C16H22ClNO2
    Purity:99.94% - >99.99%
    Color and Shape:White Or Almost White Powder White Powder
    Molecular weight:295.80
  • Detomidine carboxylic acid

    CAS:
    <p>Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.</p>
    Formula:C12H12N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:216.24
  • AdTx1


    <p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>
    Formula:C310H481N87O100S8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:7283.22
  • Carvedilol

    CAS:
    <p>Carvedilol (SKF 105517) Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intrinsic sympathomimetic activity. The S enantiomer of carvedilol nonselectively binds to and blocks beta-adrenergic receptors, thereby exerting negative inotropic and chronotropic effects, and leading to a reduction in cardiac output. In addition, both enantiomers of carvedilol bind to and block alpha 1-adrenergic receptors, thereby causing vasodilation and reducing peripheral vascular resistance.</p>
    Formula:C24H26N2O4
    Purity:99.73% - 99.97%
    Color and Shape:Colourless Crystalline Powder
    Molecular weight:406.47
  • Besipirdine hydrochloride

    CAS:
    <p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>
    Formula:C16H18ClN3
    Purity:98.45%
    Color and Shape:Soild
    Molecular weight:287.79
  • Acrinor

    CAS:
    <p>Acrinor is a adrenergic beta receptor agonist.</p>
    Formula:C35H46Cl2N10O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:805.72