GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
Read more
Pomaglumetad methionil anhydrous
CAS:635318-55-7
LY2140023, potential schizophrenia treatment, is an oral prodrug of LY404039, a selective mGlu2/3 agonist.
Formula:
C12H18N2O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
366.41
Ref: TM-T11907
| 10mg | 1,400.00 € | ||
| 25mg | 2,987.00 € | ||
| 50mg | 4,698.00 € | ||
| 100mg | 7,142.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
NBQX Disodium
CAS:479347-86-9
NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and …
Formula:
C12H6N4Na2O6S
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
380.24
Ref: TM-T25853
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 464.00 € | ||
| 100mg | 677.00 € | ||
| 200mg | 938.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
(S)-AMPA HCl
(S)-AMPA HCl (L-AMPA HCl) is a selective AMPA receptor agonist with potential antidepressant activity. It …
Formula:
C7H11ClN2O4
Color and Shape:
Liquid
Molecular weight:
222.63
Ref: TM-T21271L
| 1mg | 264.00 € | ||
| 5mg | 571.00 € | ||
| 10mg | 857.00 € | ||
| 25mg | 1,443.00 € | ||
| 50mg | 2,097.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
EGLU
CAS:170984-72-2
EGLU, an antidepressant and potent mGluR-2 antagonist, binds with a 66 μM Kd to (lS,3S)-ACPD …
Formula:
C7H13NO4
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
175.18
Ref: TM-T11165
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
AMN082
CAS:97075-46-2
AMN082 is an mGluR7 agonist with antidepressant effects. Neuroprotective effect of AMN082 on neuronal apoptosis …
Formula:
C28H30Cl2N2
Purity:
97.23% - 98.34%
Color and Shape:
Solid
Molecular weight:
465.46
Ref: TM-T21935
| 1mg | 42.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 216.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
(S)-4CPG
CAS:134052-73-6
(S)-4CPG ((S)-4-Carboxyphenylglycine) is a competitive mGlu1 receptor antagonist that attenuates nociceptive hypersensitivity and nociceptive abnormalities …
Formula:
C9H9NO4
Color and Shape:
Solid
Molecular weight:
195.17
Ref: TM-T5507
| 1mg | 40.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 373.00 € | ||
| 200mg | 546.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
LY341495
CAS:201943-63-7
LY341495 is a potent metabotropic glutamate receptor antagonist and can be used to study neurological …
Formula:
C20H19NO5
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
353.37
Ref: TM-T15816
| 1mg | 47.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Mar 2025
NS-102
CAS:136623-01-3
NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2) and inhibits …
Formula:
C12H11N3O4
Purity:
98.73% - 98.95%
Color and Shape:
Liquid
Molecular weight:
261.23
Ref: TM-T38779
| 1mg | 156.00 € | ||
| 5mg | 376.00 € | ||
| 10mg | 628.00 € | ||
| 25mg | 1,035.00 € | ||
| 50mg | 1,396.00 € | ||
| 100mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
γ-DGG
CAS:6729-55-1
gamma-DGG is a competitive blocker of AMPA receptor.
Formula:
C7H12N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
204.18
Ref: TM-T15369
| 5mg | 47.00 € | ||
| 10mg | 60.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
GYKI 52466 dihydrochloride
CAS:2319722-40-0
GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used …
Formula:
C17H17Cl2N3O2
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
366.24
Ref: TM-T11522
| 2mg | 111.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
VU0422288
CAS:1630936-95-6
VU0422288 (ML396) is a type III mGlu receptor (mGlus) orthosteric modulator with inhibitory effects on …
Formula:
C17H11Cl2N3O2
Purity:
95.48%
Color and Shape:
Solid
Molecular weight:
360.19
Ref: TM-T29135
| 5mg | 80.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 376.00 € | ||
| 100mg | 612.00 € | ||
| 500mg | 1,264.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
JNJ-46778212
CAS:1363281-27-9
JNJ-46778212 (VU 0409551) is a selective and potent mGlu5 allosteric modulator (EC50: 260 nM) for …
Formula:
C20H17FN2O3
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
352.36
Ref: TM-T15619
| 5mg | 62.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 344.00 € | ||
| 100mg | 552.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CX717
CAS:867276-98-0
CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.
Formula:
C11H11N3O3
Purity:
100%
Color and Shape:
Soild
Molecular weight:
233.23
Ref: TM-T60201
| 10mg | 46.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 117.00 € | ||
| 100mg | 187.00 € | ||
| 200mg | 279.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
GYKI 53655 hydrochloride
CAS:143692-48-2
GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the …
Formula:
C19H21ClN4O3
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
388.85
Ref: TM-T15456
| 1mg | 58.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
CX516
CAS:154235-83-3
CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as …
Formula:
C14H15N3O
Purity:
99.29% - ≥95%
Color and Shape:
Tan Solid
Molecular weight:
241.29
Ref: TM-T1884
| 10mg | 34.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 65.00 € | ||
| 100mg | 84.00 € | ||
| 200mg | 133.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
DNQX
CAS:2379-57-9
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 …
Formula:
C8H4N4O6
Purity:
97.15% - 99.10%
Color and Shape:
Off-White Powder With A Yellow Tinge
Molecular weight:
252.14
Ref: TM-T7304
| 25mg | 56.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
VU0364770
CAS:61350-00-3
VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 …
Formula:
C12H9ClN2O
Purity:
99.66% - 99.92%
Color and Shape:
Solid
Molecular weight:
232.67
Ref: TM-T6727
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 62.00 € | ||
| 50mg | 99.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 221.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
XAP044
CAS:196928-50-4
XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.
Formula:
C15H9IO4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
380.13
Ref: TM-T21995
| 1mg | 62.00 € | ||
| 2mg | 87.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 557.00 € | ||
| 100mg | 797.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Lu AF21934
CAS:1445605-23-1
Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, …
Formula:
C14H16Cl2N2O2
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
315.2
Ref: TM-T3539
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 588.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
DL-AP3
CAS:20263-06-3
DL-AP3 is a competitive group I metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase.
Formula:
C3H8NO5P
Purity:
98.18% - ≥98%
Color and Shape:
White Powder
Molecular weight:
169.07
Ref: TM-T22730
| 5mg | 34.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
