GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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CDPPB
CAS:781652-57-1
CDPPB is a modulator of mGluR5 positive allosteric(with an EC50 of 27 nM in Chinese …
Formula:
C23H16N4O
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
364.4
Ref: TM-T22641
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 410.00 € | ||
| 100mg | 613.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU0155094
CAS:731006-86-3
VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group …
Formula:
C24H24N2O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
436.52
Ref: TM-T9011
| 1mg | 96.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 466.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 932.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU 0357121
CAS:433967-28-3
VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly …
Formula:
C17H17F2NO2
Purity:
99% - 99.99%
Color and Shape:
Solid
Molecular weight:
305.32
Ref: TM-T6725
| 5mg | 59.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 521.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MPEP
CAS:96206-92-7
MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable …
Formula:
C14H11N
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
193.24
Ref: TM-T6598
| 10mg | 47.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 206.00 € | ||
| 200mg | 305.00 € | ||
| 500mg | 512.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
NBQX
CAS:118876-58-7
NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active …
Formula:
C12H8N4O6S
Purity:
97.66% - 99.42%
Color and Shape:
Solid
Molecular weight:
336.28
Ref: TM-T4113
| 1mg | 40.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 492.00 € | ||
| 100mg | 514.00 € | ||
| 200mg | 740.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CX614
CAS:191744-13-5
CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.
Formula:
C13H13NO4
Purity:
97.43%
Color and Shape:
Solid
Molecular weight:
247.25
Ref: TM-T19698
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 405.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU0361737
CAS:1161205-04-4
VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), …
Formula:
C13H11ClN2O2
Purity:
99.09% - 99.86%
Color and Shape:
Solid
Molecular weight:
262.69
Ref: TM-T6726
| 10mg | 36.00 € | ||
| 25mg | 62.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CFMTI
CAS:864864-17-5
CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.
Formula:
C19H16FN5O
Purity:
97.23%
Color and Shape:
Solid
Molecular weight:
349.36
Ref: TM-T3482
| 1mg | 60.00 € | ||
| 2mg | 86.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 179.00 € | ||
| 25mg | 319.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 630.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JNJ-42153605
CAS:1254977-87-1
JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).
Formula:
C22H23F3N4
Purity:
97.25% - 98.57%
Color and Shape:
Solid
Molecular weight:
400.44
Ref: TM-T3451
| 1mg | 34.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 382.00 € | ||
| 200mg | 536.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU 0364439
CAS:1246086-78-1
VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).
Formula:
C18H13Cl2N3O3S
Purity:
97.90%
Color and Shape:
Solid
Molecular weight:
422.29
Ref: TM-T6160
| 1mg | 47.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 206.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 528.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CX516
CAS:154235-83-3
CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as …
Formula:
C14H15N3O
Purity:
99.29% - ≥95%
Color and Shape:
Tan Solid
Molecular weight:
241.29
Ref: TM-T1884
| 10mg | 34.00 € | ||
| 25mg | 44.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 81.00 € | ||
| 200mg | 128.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
FITM
CAS:932737-65-0
FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).
Formula:
C18H18FN5OS
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
371.43
Ref: TM-T7292
| 1mg | 36.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 280.00 € | ||
| 100mg | 413.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Cyclothiazide
CAS:2259-96-3
Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).
Formula:
C14H16ClN3O4S2
Purity:
98.23% - 98.74%
Color and Shape:
Crystals From Dilute Alcohol Solid
Molecular weight:
389.88
Ref: TM-T4573
| 5mg | 52.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 230.00 € | ||
| 100mg | 341.00 € | ||
| 200mg | 503.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
IDRA-21
CAS:22503-72-6
IDRA-21 is a positive AMPA receptor modulator.
Formula:
C8H9ClN2O2S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
232.69
Ref: TM-T7823
| 50mg | 44.00 € | ||
| 100mg | 63.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
HBT1
CAS:489408-02-8
HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and …
Formula:
C16H17F3N4O2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
386.39
Ref: TM-T8779
| 10mg | 46.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 112.00 € | ||
| 100mg | 182.00 € | ||
| 200mg | 272.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ADX-47273
CAS:851881-60-2
ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor …
Formula:
C20H17F2N3O2
Purity:
97% - 99.18%
Color and Shape:
Solid
Molecular weight:
369.36
Ref: TM-T2053
| 2mg | 39.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 294.00 € | ||
| 100mg | 528.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Caroverine hydrochloride
CAS:55750-05-5
Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.
Formula:
C22H28ClN3O2
Purity:
98.37% - 98.75%
Color and Shape:
Solid
Molecular weight:
401.9
Ref: TM-T9133
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 369.00 € | ||
| 200mg | 544.00 € | ||
| 500mg | 848.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AMN082 free base
CAS:83027-13-8
AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.
Formula:
C28H28N2
Purity:
97.75% - 97.79%
Color and Shape:
Solid
Molecular weight:
392.54
Ref: TM-T21935L
| 1mg | 41.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 553.00 € | ||
| 500mg | 1,160.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ADX88178
CAS:1235318-89-4
ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 …
Formula:
C12H12N6S
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
272.33
Ref: TM-T4500
| 2mg | 37.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 345.00 € | ||
| 200mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU0155041
CAS:1093757-42-6
VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, …
Formula:
C14H15Cl2NO3
Purity:
99.52% - 99.56%
Color and Shape:
Solid
Molecular weight:
316.18
Ref: TM-T3565
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 290.00 € | ||
| 200mg | 419.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
