AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Vecuronium bromide
CAS:50700-72-6
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting mono-quaternary steroid and non-depolarizing neuromuscular blocking …
Formula:
C34H57BrN2O4
Purity:
99.63% - 99.92%
Color and Shape:
White Powder
Molecular weight:
637.73
Ref: TM-T1594
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 97.00 € | ||
| 500mg | 207.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Homatropine Methylbromide
CAS:80-49-9
Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with …
Formula:
C17H24BrNO3
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
370.29
Ref: TM-T0427
| 25mg | 43.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 65.00 € | ||
| 200mg | 88.00 € | ||
| 500mg | 133.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Darifenacin hydrobromide
CAS:133099-07-7
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and …
Formula:
C28H31BrN2O2
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
505.45
Ref: TM-T1534
| 50mg | 49.00 € | ||
| 100mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Pirenzepine dihydrochloride
CAS:29868-97-1
Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
Formula:
C19H21N5O2·2HCl
Purity:
99.48% - 99.62%
Color and Shape:
White Powder
Molecular weight:
424.32
Ref: TM-T1542
| 1ml | 63.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 88.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Tolterodine tartrate
CAS:124937-52-6
Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the …
Formula:
C22H31NO·C4H6O6
Purity:
99.95%
Color and Shape:
White-To-Off-White Crystalline Powder
Molecular weight:
475.58
Ref: TM-T0099
| 25mg | 52.00 € | ||
| 50mg | 84.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 126.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Ipratropium bromide monohydrate
CAS:66985-17-9
Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.
Formula:
C20H32BrNO4
Purity:
97.85%
Color and Shape:
Solid
Molecular weight:
430.38
Ref: TM-T0098
| 25mg | 50.00 € | ||
| 50mg | 77.00 € | ||
| 100mg | 108.00 € | ||
| 500mg | 264.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
nAChR agonist 1
CAS:1394371-75-5
nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine …
Formula:
C20H18ClNO3S2
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
419.94
Ref: TM-T12165
| 1mg | 94.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 775.00 € | ||
| 200mg | 1,026.00 € | ||
| 1mL*10mM (DMSO) | 192.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Neostigmine methyl sulfate
CAS:51-60-5
Neostigmine methyl sulfate (Syntostigmin) is a reversible inhibitor of acetylcholinesterase used in the treatment of …
Formula:
C13H22N2O6S
Purity:
99.34% - 99.53%
Color and Shape:
Crystalline Solid
Molecular weight:
334.39
Ref: TM-T1612
| 100mg | 55.00 € | ||
| 200mg | 66.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
MK-7622
CAS:1227923-29-6
MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.
Formula:
C25H25N3O2
Purity:
99.77% - 99.8%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T15942
| 2mg | 49.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Loxeen
CAS:6856-31-1
Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.
Formula:
C20H25NO·CH4O3S
Purity:
99.46%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
391.52
Ref: TM-T1072
| 1g | 165.00 € | ||
| 25mg | 34.00 € | ||
| 50mg | 42.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 114.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Propantheline bromide
CAS:50-34-0
Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on …
Formula:
C23H30BrNO3
Purity:
95% - ≥98%
Molecular weight:
448.4
Ref: TM-T1006
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 74.00 € | ||
| 500mg | 107.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Benactyzine hydrochloride
CAS:57-37-4
Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.
Formula:
C20H26ClNO3
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
363.88
Ref: TM-T2571
| 100mg | 48.00 € | ||
| 200mg | 65.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Pancuronium dibromide
CAS:15500-66-0
Pancuronium dibromide (Pavulon), a competitive AChR antagonist, acts as a skeletal muscle relaxant. Pancuronium dibromide …
Formula:
C35H60Br2N2O4
Purity:
99.86%
Color and Shape:
solid
Molecular weight:
732.67
Ref: TM-T0166
| 5mg | 38.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 115.00 € | ||
| 100mg | 188.00 € | ||
| 200mg | 235.00 € | ||
| 500mg | 394.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Fesoterodine fumarate
CAS:286930-03-8
Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic …
Formula:
C26H37NO3·C4H4O4
Purity:
98% - 98.55%
Color and Shape:
White Solid
Molecular weight:
527.65
Ref: TM-T1475
| 5mg | 51.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 153.00 € | ||
| 100mg | 227.00 € | ||
| 500mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Gallamine triethiodide
CAS:65-29-2
Gallamine triethiodide (Benzkurin), a synthetic inhibiting drug, is nondepolarizing.
Formula:
C30H60I3N3O3
Purity:
98.90%
Color and Shape:
White Amorphous Powder Solid
Molecular weight:
891.53
Ref: TM-T0720
| 100mg | 48.00 € | ||
| 200mg | 70.00 € | ||
| 500mg | 114.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
(Rac)-ABT-202 dihydrochloride
CAS:1258641-38-1
(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist …
Formula:
C9H15Cl2N3
Purity:
97.4%
Color and Shape:
Solid
Molecular weight:
236.142
Ref: TM-T12653
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 497.00 € | ||
| 100mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 119.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Temephos
CAS:3383-96-8
Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.
Formula:
C16H20O6P2S3
Purity:
≥95%
Color and Shape:
White Crystalline Solid Or Liquid
Molecular weight:
466.47
Ref: TM-T0997
| 25mg | 49.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 7 Apr 2025
Methacholine Chloride
CAS:62-51-1
Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of …
Formula:
C8H18ClNO2
Purity:
99.37% - 99.74%
Color and Shape:
White Hygroscopic Crystals With Slight Odor Of Dead Fish
Molecular weight:
195.69
Ref: TM-T1682
| 100mg | 65.00 € | ||
| 200mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Atropine methyl bromide
CAS:2870-71-5
Atropine methyl bromide (Methylatropine bromide) is a quaternary ammonium salt of atropine, characterized as a …
Formula:
C18H26BrNO3
Purity:
99.70%
Color and Shape:
Solid
Molecular weight:
384.308
Ref: TM-T14345
| 1mg | 40.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 432.00 € | ||
| 1mL*10mM (DMSO) | 131.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
Flavoxate hydrochloride
CAS:3717-88-2
Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various …
Formula:
C24H26ClNO4
Purity:
99.78%
Color and Shape:
White Solid
Molecular weight:
427.92
Ref: TM-T0703
| 1g | 87.00 € | ||
| 25mg | 35.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 69.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
