AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Dicyclomine hydrochloride
CAS:67-92-5
Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.
Formula:
C19H36ClNO2
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
345.95
Ref: TM-T1460
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Benzethonium chloride
CAS:121-54-0
Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum …
Formula:
C27H42ClNO2
Purity:
97.5%
Color and Shape:
White To Off-White Solid Solid Particulate/Powder
Molecular weight:
448.09
Ref: TM-T0401
| 50mg | 42.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 74.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
TAK-071
CAS:1820812-16-5
TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) …
Formula:
C24H24FN3O3
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
421.46
Ref: TM-T13066
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 229.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 545.00 € | ||
| 500mg | 2,040.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Homatropine Methylbromide
CAS:80-49-9
Homatropine Methylbromide is the methyl bromide salt of homatropine, a synthetic tertiary amine alkaloid with …
Formula:
C17H24BrNO3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
370.29
Ref: TM-T0427
| 25mg | 47.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 88.00 € | ||
| 500mg | 131.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
MK-7622
CAS:1227923-29-6
MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.
Formula:
C25H25N3O2
Purity:
99.77% - 99.8%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T15942
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Nebracetam hydrochloride
CAS:1177279-49-0
Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an …
Formula:
C12H17ClN2O
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
240.729
Ref: TM-T12201
| 5mg | 49.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 225.00 € | ||
| 200mg | 330.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Benactyzine hydrochloride
CAS:57-37-4
Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.
Formula:
C20H26ClNO3
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
363.88
Ref: TM-T2571
| 100mg | 53.00 € | ||
| 200mg | 69.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Darifenacin hydrobromide
CAS:133099-07-7
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and …
Formula:
C28H31BrN2O2
Purity:
100% - 99.71%
Color and Shape:
Solid
Molecular weight:
505.45
Ref: TM-T1534
| 50mg | 50.00 € | ||
| 100mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Tolterodine tartrate
CAS:124937-52-6
Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the …
Formula:
C22H31NO·C4H6O6
Purity:
99.62%
Color and Shape:
White-To-Off-White Crystalline Powder
Molecular weight:
475.58
Ref: TM-T0099
| 25mg | 51.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 122.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Pirenzepine dihydrochloride
CAS:29868-97-1
Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
Formula:
C19H21N5O2·2HCl
Purity:
99.62% - 99.68%
Color and Shape:
White Powder
Molecular weight:
424.32
Ref: TM-T1542
| 1ml | 62.00 € | ||
| 50mg | 47.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 88.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
nAChR agonist 1
CAS:1394371-75-5
nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine …
Formula:
C20H18ClNO3S2
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
419.94
Ref: TM-T12165
| 1mg | 92.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 413.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 754.00 € | ||
| 200mg | 998.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Loxeen
CAS:6856-31-1
Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.
Formula:
C20H25NO·CH4O3S
Purity:
99.72%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
391.52
Ref: TM-T1072
| 1g | 159.00 € | ||
| 25mg | 34.00 € | ||
| 50mg | 41.00 € | ||
| 100mg | 51.00 € | ||
| 500mg | 110.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Propantheline bromide
CAS:50-34-0
Propantheline bromide (Pro-Banthine) competitively antagonizes acetylcholine activity mediated by muscarinic receptors at neuroeffector sites on …
Formula:
C23H30BrNO3
Purity:
95% - ≥98%
Molecular weight:
448.4
Ref: TM-T1006
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 74.00 € | ||
| 500mg | 105.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Methacholine Chloride
CAS:62-51-1
Methacholine Chloride (Acetyl-β-methylcholine chloride) is a quaternary ammonium parasympathomimetic agent with the muscarinic actions of …
Formula:
C8H18ClNO2
Purity:
99.47% - 99.74%
Color and Shape:
White Hygroscopic Crystals With Slight Odor Of Dead Fish
Molecular weight:
195.69
Ref: TM-T1682
| 100mg | 64.00 € | ||
| 200mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Flavoxate hydrochloride
CAS:3717-88-2
Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various …
Formula:
C24H26ClNO4
Purity:
99.64%
Color and Shape:
White Solid
Molecular weight:
427.92
Ref: TM-T0703
| 1g | 96.00 € | ||
| 25mg | 35.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 68.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Diphenmanil methylsulfate
CAS:62-97-5
Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.
Formula:
C20H24N·CH3O4S
Purity:
98% - 99.85%
Color and Shape:
Solid
Molecular weight:
389.51
Ref: TM-T0594
| 25mg | 44.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 66.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 140.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Trospium chloride
CAS:10405-02-4
Trospium chloride treats urinary incontinence without causing liver damage.
Formula:
C25H30ClNO3
Purity:
100% - 99.92%
Color and Shape:
White To Off-White Powder
Molecular weight:
427.964
Ref: TM-T1472
| 1g | 86.00 € | ||
| 100mg | 35.00 € | ||
| 500mg | 59.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Clidinium bromide
CAS:3485-62-9
Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and …
Formula:
C22H26BrNO3
Purity:
98.89% - 99.86%
Color and Shape:
White Crystalline Solid
Molecular weight:
432.35
Ref: TM-T0786
| 50mg | 39.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 105.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Tropicamide
CAS:1508-75-4
Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for …
Formula:
C17H20N2O2
Purity:
99.75% - 99.78%
Color and Shape:
White Powder
Molecular weight:
284.35
Ref: TM-T1281
| 100mg | 52.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Orphenadrine Citrate
CAS:4682-36-4
Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system …
Formula:
C18H23NO·C6H8O7
Purity:
98% - 99.51%
Color and Shape:
White Solid
Molecular weight:
461.5
Ref: TM-T6618
| 50mg | 40.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
