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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • Solifenacin succinate

    CAS:
    <p>Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.</p>
    Formula:C23H26N2O2·C4H6O4
    Purity:99.85% - 99.98%
    Color and Shape:Solid
    Molecular weight:480.56
  • Diphenmanil methylsulfate

    CAS:
    <p>Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.</p>
    Formula:C20H24N·CH3O4S
    Purity:98% - 99.27%
    Color and Shape:Solid
    Molecular weight:389.51
  • Pirenzepine dihydrochloride

    CAS:
    <p>Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.</p>
    Formula:C19H21N5O2·2HCl
    Purity:99.48% - 99.62%
    Color and Shape:White Powder
    Molecular weight:424.32
  • Temephos

    CAS:
    <p>Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.</p>
    Formula:C16H20O6P2S3
    Purity:≥95%
    Color and Shape:White Crystalline Solid Or Liquid
    Molecular weight:466.47
  • Carbetapentane citrate

    CAS:
    <p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>
    Formula:C20H31NO3·C6H8O7
    Purity:99.46%
    Color and Shape:White To Off-White Solid
    Molecular weight:525.59
  • Zelminemab

    CAS:
    <p>Zelminemab (AMG-301) is a human monoclonal antibody designed to target and inhibit the PACAP type I (PAC1) receptor [1].</p>
    Purity:98.8% (SDS-PAGE); 97% (SEC-HPLC) - 98.8% (SDS-PAGE); 97% (SEC-HPLC)
    Color and Shape:Liquid
  • Rivastigmine tartrate

    CAS:
    <p>Rivastigmine (SDZ-ENA 713), a CNS-selective carbamate, treats dementia in Alzheimer's and Parkinson's.</p>
    Formula:C14H22N2O2·C4H6O6
    Purity:98% - 99.66%
    Color and Shape:White To Off-White Powder
    Molecular weight:400.43
  • Dequalinium chloride

    CAS:
    <p>Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.</p>
    Formula:C30H40Cl2N4
    Purity:99.79% - 99.9%
    Color and Shape:Solid
    Molecular weight:527.59
  • Cotinine

    CAS:
    <p>Cotinine (NIH-10498) is an alkaloid found in tobacco and is also the predominant metabolite of nicotine.</p>
    Formula:C10H12N2O
    Purity:98% - 99.89%
    Color and Shape:Viscous Oil Solid
    Molecular weight:176.22
  • MK-7622

    CAS:
    <p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>
    Formula:C25H25N3O2
    Purity:99.77% - 99.8%
    Color and Shape:Solid
    Molecular weight:399.48
  • Dicyclomine hydrochloride

    CAS:
    <p>Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.</p>
    Formula:C19H36ClNO2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:345.95
  • Benactyzine hydrochloride

    CAS:
    <p>Benactyzine hydrochloride (Neuroleptone) is a centrally acting muscarinic antagonist.</p>
    Formula:C20H26ClNO3
    Purity:99.03% - 99.94%
    Color and Shape:Solid
    Molecular weight:363.88
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Formula:C21H25NO·CH4SO3
    Purity:98.41% - 99.96%
    Color and Shape:White Crystalline Powder; Odourless Or Almost Odourless
    Molecular weight:403.53
  • Procainamide hydrochloride

    CAS:
    <p>Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analog</p>
    Formula:C13H21N3O·HCl
    Purity:99.83% - 99.97%
    Color and Shape:White To Slightly Yellow Powder
    Molecular weight:271.79
  • VU 0365114

    CAS:
    <p>VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).</p>
    Formula:C22H14F3NO3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:397.35
  • Fipexide

    CAS:
    <p>Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983.</p>
    Formula:C20H21ClN2O4
    Purity:97.6% - 99.95%
    Color and Shape:Solid
    Molecular weight:388.84
  • (Rac)-ABT-202 dihydrochloride

    CAS:
    <p>(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.</p>
    Formula:C9H15Cl2N3
    Purity:97.4%
    Color and Shape:Solid
    Molecular weight:236.142
  • Lysipressin acetate(50-57-7(fb_acetate))

    CAS:
    <p>Lysipressin acetate (50-57-7), triggers rabbit bladder contraction &amp; activates adenylate cyclase, is an antidiuretic in pigs &amp; marsupials.</p>
    Formula:C48H69N13O14S2
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:1116.28
  • Nebracetam hydrochloride

    CAS:
    <p>Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.</p>
    Formula:C12H17ClN2O
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:240.729
  • nAChR agonist 1

    CAS:
    <p>nAChR agonist 1 (DUN71755) is a brain-permeable and orally efficacious positive allosteric α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.</p>
    Formula:C20H18ClNO3S2
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:419.94