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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 643 products of "AChR"

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  • Tebanicline tosylate

    CAS:
    Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.
    Formula:C16H19ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.85

    Ref: TM-T3694L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD 0328

    CAS:
    AZD 0328 is a nicotinic receptor agonist for α7 neurons.
    Formula:C13H16N2O
    Color and Shape:Solid
    Molecular weight:216.28

    Ref: TM-T30247

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LRE1

    CAS:
    LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.
    Formula:C12H13ClN4S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:280.78

    Ref: TM-T15787

    10mg
    39.00€
    25mg
    71.00€
    50mg
    119.00€
    100mg
    172.00€
  • SIB 1508Y maleate

    CAS:
    neuronal nicotinic ACh receptor agonist
    Formula:C16H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.33

    Ref: TM-T23352

    50mg
    3,510.00€
  • Benzatropine

    CAS:
    Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.
    Formula:C21H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.43

    Ref: TM-T23781

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R,R)-Glycopyrrolate

    CAS:
    (R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.
    Formula:C19H28BrNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.34

    Ref: TM-T12640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Terodiline hydrochloride

    CAS:

    Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),

    Formula:C20H28ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:317.9

    Ref: TM-T13129

    25mg
    1,159.00€
    50mg
    1,510.00€
    100mg
    2,308.00€
  • Elucaine

    CAS:
    Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.
    Formula:C19H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.39

    Ref: TM-T15211

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • YM-46303

    CAS:
    YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia in
    Formula:C20H23ClN2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:358.86

    Ref: TM-T13370

    1mg
    630.00€
    5mg
    1,620.00€
  • CHF5407

    CAS:
    CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on
    Formula:C27H25BrF4N2O3S
    Purity:99.54% - >99.99%
    Color and Shape:Solid
    Molecular weight:613.46

    Ref: TM-T13992

    1mg
    138.00€
    5mg
    280.00€
    10mg
    416.00€
    25mg
    683.00€
    50mg
    964.00€
    100mg
    1,288.00€
  • AR-R 17779 hydrochloride

    CAS:
    AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.
    Formula:C9H15ClN2O2
    Color and Shape:Solid
    Molecular weight:218.68

    Ref: TM-T21857

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Biricodar dicitrate

    CAS:
    Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.
    Formula:C46H57N3O21
    Purity:97.78% - 99.78%
    Color and Shape:Solid
    Molecular weight:987.95

    Ref: TM-T67790

    1mg
    492.00€
    5mg
    1,111.00€
    25mg
    1,825.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • KL8604166

    CAS:
    KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.
    Formula:C12H21N5O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:267.33

    Ref: TM-T29038

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    1mL*10mM (DMSO)
    590.00€
  • PF-06767832

    CAS:
    PF-06767832: selective M1 PAM (EC50=60 nM), no M2-M5 activity, good CNS penetration, but has GI and cardiovascular risks.
    Formula:C22H23N3O3S
    Color and Shape:Solid
    Molecular weight:409.5

    Ref: TM-T33950

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Hadacidin

    CAS:
    Hadacidin is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.
    Formula:C3H5NO4
    Color and Shape:Solid
    Molecular weight:119.08

    Ref: TM-T68868

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bibn 140

    CAS:
    Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.
    Formula:C32H44N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.72

    Ref: TM-T26798

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon Receptor Antagonist I

    CAS:
    Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.
    Formula:C20H30N2OS
    Color and Shape:Solid
    Molecular weight:346.53

    Ref: TM-T37223

    1mg
    430.00€
    5mg
    1,549.00€
  • RJR-2403 oxalate

    CAS:
    RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.
    Formula:C14H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.308

    Ref: TM-T26096

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RJR-2429

    CAS:
    RJR-2429 is a potent AChR agonist.
    Formula:C12H16N2
    Color and Shape:Solid
    Molecular weight:188.27

    Ref: TM-T68362

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CC4

    CAS:
    Selective α6β2/α4β2 partial agonist; Ki: 12/26nM (rat); poor α3β4/α7 affinity; stimulates dopamine release; reduces nicotine self-admin in rats.
    Formula:C24H30N4O2
    Color and Shape:Solid
    Molecular weight:406.52

    Ref: TM-T37202

    50mg
    2,475.00€
  • Hadacidin sodium

    CAS:
    Hadacidin sodium is an inhibitor of AMP synthesis. Hadacidin and hadacidin analogues have anticancer activity and activity against adenylosuccinate synthetase.
    Formula:C3H4NNaO4
    Color and Shape:Solid
    Molecular weight:141.06

    Ref: TM-T69565

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dexetimide HCl

    CAS:
    Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.
    Formula:C23H27ClN2O2
    Color and Shape:Solid
    Molecular weight:398.93

    Ref: TM-T69825

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (E/Z)-VU0029767

    CAS:
    VU0029767 enhances M1 muscarinic receptor function, increasing acetylcholine potency and efficacy.
    Formula:C21H21N3O3
    Color and Shape:Solid
    Molecular weight:363.41

    Ref: TM-T29120

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Octamylamine sulfamate

    CAS:
    Octamylamine sulfamate is a P450 inhibitor.
    Formula:C13H32N2O3S
    Color and Shape:Solid
    Molecular weight:296.47

    Ref: TM-T68215

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adenylyl cyclase type 2 agonist-1

    CAS:
    Potent AC2 agonist with an EC50 of 90 nM, potential for respiratory disease treatment.
    Formula:C27H17BrClNO5
    Color and Shape:Solid
    Molecular weight:550.78

    Ref: TM-T63893

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Muscarine iodide

    CAS:
    Muscarinic acetylcholine receptor agonist
    Formula:C9H20INO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:301.17

    Ref: TM-T23034

    10mg
    1,071.00€
  • LY 2087101

    CAS:
    Allosteric potentiator of α7, α4β2 and α4β4 nAChRs
    Formula:C15H11FN2OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.39

    Ref: TM-T22939

    10mg
    767.00€
    50mg
    2,673.00€
  • Metanicotine

    CAS:
    Metanicotine is a selective nicotinic agonist with antinociceptive properties.
    Formula:C10H14N2
    Color and Shape:Solid
    Molecular weight:162.23

    Ref: TM-T69134

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Caramiphen hydrochloride

    CAS:
    Caramiphen hydrochloride: antimuscarinic, anticholinergic, NMDA receptor antagonist salt.
    Formula:C18H28ClNO2
    Color and Shape:Solid
    Molecular weight:325.88

    Ref: TM-T71107

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Flupyrimin

    CAS:
    Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].
    Formula:C13H9ClF3N3O
    Color and Shape:Solid
    Molecular weight:315.68

    Ref: TM-T60819

    2mg
    110.00€
    100mg
    1,153.00€
  • TC-1698 dihydrochloride

    CAS:
    TC-1698 dihydrochloride: selective α7 nicotinic agonist, with some β-receptor activity; neuroprotectant.
    Formula:C13H20Cl2N2
    Color and Shape:Solid
    Molecular weight:275.22

    Ref: TM-T68697

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Octamylamine hydrochloride

    CAS:
    Octamylamine hydrochloride is a P450 inhibitor.
    Formula:C13H30ClN
    Color and Shape:Solid
    Molecular weight:235.84

    Ref: TM-T69039

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Neopterin, L-erythro-

    CAS:
    Neopterin, L-erythro- can be used as a cholinergic receptor.
    Formula:C9H11N5O4
    Color and Shape:Solid
    Molecular weight:253.21

    Ref: TM-T33634

    25mg
    1,369.00€
  • Methacholine iodide

    CAS:
    Methacholine iodide is a muscarinic acetylcholine receptor agonist.
    Formula:C8H18INO2
    Color and Shape:Solid
    Molecular weight:287.14

    Ref: TM-T68975

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dimethyl-W84 (dibromide)

    CAS:
    Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.
    Formula:C34H48Br2N4O4
    Color and Shape:Solid
    Molecular weight:736.59

    Ref: TM-T38111

    5mg
    447.00€
  • 5-Iodo-A-85380 dihydrochloride

    CAS:
    α4β2 and α6β2 nicotinic acetylcholine receptors agonist
    Formula:C9H13Cl2IN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.02

    Ref: TM-T22521

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Anabasine hydrochloride

    CAS:
    neuronal nicotinic ACh receptor partial agonist
    Formula:C10H15ClN2
    Purity:98%
    Color and Shape:White To Off-White Solid
    Molecular weight:198.693

    Ref: TM-T22571

    50mg
    477.00€
  • CDD0102

    CAS:
    CDD0102 is a potent agonist of M1 Muscarinic receptor.
    Formula:C8H12N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:180.21

    Ref: TM-T10731

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AQ-RA 721

    CAS:
    AQ-RA 721 is a selective muscarinic antagonist with high affinity for M1- and M3-receptors. AQ-RA 721 may be used as a bronchodilator.
    Formula:C22H23N3O2
    Color and Shape:Solid
    Molecular weight:361.44

    Ref: TM-T70797

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Ethybenztropine

    CAS:
    Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.
    Formula:C22H27NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.46

    Ref: TM-T27295

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD-9164 bromide

    CAS:
    AMG-221, a selective 11β-HSD1 inhibitor, suppresses enzyme activity, lowers glucose/insulin, and reduces weight in obese mice.
    Formula:C29H38BrFN2O2
    Color and Shape:Solid
    Molecular weight:545.53

    Ref: TM-T26724

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UH-AH 37

    CAS:
    UH-AH 37 is a antagonist of human muscarinic acetylcholine receptor.
    Formula:C21H23Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.33

    Ref: TM-T29047

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DAU 5884 HCl

    CAS:
    DAU 5884 HCl is an M3 receptor antagonist
    Formula:C17H21N3O3
    Color and Shape:Solid
    Molecular weight:315.37

    Ref: TM-T71962

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ethybenztropine HBr

    CAS:
    Ethybenztropine HBr is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.
    Formula:C22H28BrNO
    Color and Shape:Solid
    Molecular weight:402.37

    Ref: TM-T69614

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Atropine Oxide Hydrochloride

    CAS:
    Atropine Oxide, a derivative of anticholinergic Atropine, treats poisonings, slow heart rate, and reduces saliva during surgery.
    Formula:C17H24ClNO4
    Color and Shape:Solid
    Molecular weight:341.83

    Ref: TM-T69232

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • YM-58790

    CAS:
    YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.
    Formula:C27H31N3O2
    Purity:99.87%
    Color and Shape:Soild
    Molecular weight:429.55

    Ref: TM-T72038

    1mg
    64.00€
    5mg
    126.00€
    10mg
    195.00€
    25mg
    374.00€
    50mg
    533.00€
  • α7 nAchR-JAK2-STAT3 agonist 1

    CAS:
    α7 nAchR-JAK2-STAT3 agonist 1 is a potent inhibitor of the α7 nAchR-JAK2-STAT3 pathway that acts on nitric oxide (NO) (IC50: 0.32 μM).
    Formula:C25H30O6
    Color and Shape:Solid
    Molecular weight:426.5

    Ref: TM-T62317

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Metixene hydrochloride

    CAS:
    Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
    Formula:C20H24ClNS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.93

    Ref: TM-T12020

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AC-42

    CAS:

    AC-42 is an allosteric agonist of M1 muscarinic receptor.

    Formula:C20H31NO
    Color and Shape:Solid
    Molecular weight:301.47

    Ref: TM-T26541

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • (R)-Oxybutynin

    CAS:

    (R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.

    Formula:C22H31NO3
    Color and Shape:Solid
    Molecular weight:357.49

    Ref: TM-T61309

    25mg
    2,033.00€
    50mg
    2,645.00€
    100mg
    3,345.00€
  • Ethybenztropine HCl

    CAS:
    Ethybenztropine HCl is an anticholinergic which is used as an antiparkinsonian agent. Ethybenztropine may also act as a dopamine reuptake inhibitor.
    Formula:C22H28ClNO
    Color and Shape:Solid
    Molecular weight:357.92

    Ref: TM-T69549

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Esoxybutynin Chloride

    CAS:
    (S)-oxybutynin, with antimuscarinic effects, is being developed for urinary incontinence.
    Formula:C22H32ClNO3
    Color and Shape:Solid
    Molecular weight:393.95

    Ref: TM-T71889

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK575594A

    CAS:
    GSK575594A is a selective agonist of GPR55.
    Formula:C24H23F2N3O3S
    Color and Shape:Solid
    Molecular weight:471.52

    Ref: TM-T27483

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Arecaidine but-2-ynyl ester tosylate

    CAS:
    mAChR M2 agonist
    Formula:C18H23NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:365.44

    Ref: TM-T22584

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 9-CP-Ade Mesylate

    CAS:
    9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.
    Formula:C11H17N5O3S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:299.35

    Ref: TM-T23588

    1mg
    63.00€
    5mg
    137.00€
    10mg
    205.00€
    25mg
    378.00€
    50mg
    557.00€
  • PQCA

    CAS:
    PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.
    Formula:C22H20N4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:388.42

    Ref: TM-T12531

    1mg
    51.00€
    5mg
    116.00€
    10mg
    192.00€
    25mg
    304.00€
    50mg
    420.00€
    100mg
    560.00€
  • TMPH hydrochloride

    CAS:
    neuronal nicotinic ACh receptors (nAChRs) antagonist
    Formula:C16H32ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.88

    Ref: TM-T23462

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ENS-163 phosphate

    CAS:
    Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.
    Formula:C11H19N2O5PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.32

    Ref: TM-T11204

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tridihexethyl chloride

    CAS:
    Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.
    Formula:C21H36ClNO
    Color and Shape:Solid
    Molecular weight:353.97

    Ref: TM-T34936

    25mg
    888.00€
    50mg
    1,215.00€
    100mg
    1,791.00€
  • UB 165 fumarate

    CAS:
    UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.
    Formula:C17H19ClN2O4
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:350.8

    Ref: TM-T13241

    1mg
    315.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TC 2559 difumarate

    CAS:
    partial agonist of α4β2 nicotinic acetylcholine receptor
    Formula:C12H18N2OC4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.39

    Ref: TM-T23425

    1mg
    81.00€
    25mg
    1,198.00€
  • TC299423

    CAS:
    TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.
    Formula:C11H15N3
    Color and Shape:Solid
    Molecular weight:189.26

    Ref: TM-T70022

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Temiverine hydrochloride

    CAS:
    Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.
    Formula:C24H36ClNO3
    Purity:99.26% - 99.43%
    Color and Shape:Solid
    Molecular weight:422

    Ref: TM-T13118

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • NB001

    CAS:
    NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.
    Formula:C12H20N6O
    Purity:99.69%
    Color and Shape:Off-White To Pale Pink Solid
    Molecular weight:264.33

    Ref: TM-T16275

    1mg
    74.00€
    5mg
    200.00€
    10mg
    295.00€
    25mg
    497.00€
    50mg
    710.00€
    100mg
    964.00€
    500mg
    1,935.00€
    1mL*10mM (DMSO)
    173.00€
  • Oxotremorine M iodide

    CAS:
    Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.
    Formula:C11H19IN2O
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:322.19

    Ref: TM-T12339

    10mg
    48.00€
    50mg
    To inquire
    1mL*10mM (DMSO)
    50.00€
  • JNJ-39393406

    CAS:
    JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco dependence and Alzheimer's disease.
    Formula:C19H18F2N6O3
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:416.38

    Ref: TM-T27679

    1mg
    64.00€
    5mg
    137.00€
    10mg
    200.00€
    25mg
    324.00€
    50mg
    470.00€
    100mg
    662.00€
    200mg
    893.00€
  • AQW051

    CAS:
    AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.
    Formula:C19H22N2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:294.39

    Ref: TM-T26646

    1mg
    34.00€
    2mg
    46.00€
    5mg
    66.00€
    10mg
    99.00€
    25mg
    205.00€
    50mg
    313.00€
    100mg
    439.00€
    500mg
    954.00€
    1mL*10mM (DMSO)
    67.00€
  • CP-810123

    CAS:
    CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.
    Formula:C14H18N4O
    Purity:98.63% - 99.60%
    Color and Shape:Solid
    Molecular weight:258.32

    Ref: TM-T31079

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • McN-A 343

    CAS:
    McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.
    Formula:C14H18Cl2N2O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:317.21

    Ref: TM-T22963

    25mg
    54.00€
    50mg
    87.00€
    100mg
    To inquire
  • Tribendimidine

    CAS:
    Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.
    Formula:C28H32N6
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:452.59

    Ref: TM-T62769

    5mg
    50.00€
    10mg
    85.00€
    25mg
    155.00€
    50mg
    225.00€
    100mg
    336.00€
    1mL*10mM (DMSO)
    85.00€
  • Xanomeline

    CAS:
    Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.
    Formula:C14H23N3OS
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:281.42

    Ref: TM-T36640

    2mg
    34.00€
    5mg
    50.00€
    10mg
    84.00€
    25mg
    152.00€
    50mg
    236.00€
    1mL*10mM (DMSO)
    55.00€
  • PHA 543613

    CAS:
    PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.
    Formula:C15H17N3O2
    Purity:99.43% - 99.96%
    Color and Shape:Solid
    Molecular weight:271.31

    Ref: TM-T23145

    1mg
    52.00€
    5mg
    102.00€
    10mg
    166.00€
    25mg
    358.00€
    50mg
    610.00€
    100mg
    895.00€
    500mg
    1,945.00€
    1mL*10mM (DMSO)
    100.00€
  • ASM-024

    CAS:
    ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.
    Formula:C15H25N2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:233.37

    Ref: TM-T26666

    1mg
    144.00€
    2mg
    207.00€
    5mg
    346.00€
    10mg
    494.00€
    25mg
    740.00€
    1mL*10mM (DMSO)
    289.00€
  • Desformylflustrabromine hydrochloride

    CAS:
    Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.
    Formula:C17H12INO5
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:437.19

    Ref: TM-T11004

    2mg
    34.00€
    5mg
    50.00€
    10mg
    80.00€
    25mg
    145.00€
    50mg
    225.00€
    100mg
    353.00€
    200mg
    550.00€
    1mL*10mM (DMSO)
    57.00€
  • Posatirelin

    CAS:
    Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.
    Formula:C17H28N4O4
    Purity:99.43% - 99.95%
    Color and Shape:Solid
    Molecular weight:352.43

    Ref: TM-T34114

    1mg
    122.00€
    5mg
    289.00€
    10mg
    432.00€
    25mg
    707.00€
    50mg
    973.00€
    100mg
    1,333.00€
    500mg
    2,665.00€
  • Xanomeline oxalate

    CAS:
    Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.
    Formula:C16H25N3O5S
    Purity:99.1%
    Color and Shape:Solid
    Molecular weight:371.45

    Ref: TM-T13353

    5mg
    35.00€
    10mg
    55.00€
    25mg
    100.00€
    50mg
    159.00€
    100mg
    245.00€
    200mg
    353.00€
    1mL*10mM (DMSO)
    39.00€
  • GSK233705

    CAS:
    GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.
    Formula:C24H29BrN2
    Purity:99.87% - 99.98%
    Color and Shape:Solid
    Molecular weight:425.4

    Ref: TM-T31207

    1mg
    81.00€
    5mg
    172.00€
    10mg
    259.00€
    25mg
    424.00€
    50mg
    620.00€
    100mg
    884.00€
    500mg
    1,773.00€
  • Otenzepad

    CAS:
    Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.
    Formula:C24H31N5O2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:421.54

    Ref: TM-T16411

    1mg
    44.00€
    5mg
    79.00€
    10mg
    114.00€
    25mg
    222.00€
    50mg
    356.00€
    100mg
    572.00€
    200mg
    803.00€
    1mL*10mM (DMSO)
    87.00€
  • Aceclidine

    CAS:
    Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular
    Formula:C9H15NO2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:169.22

    Ref: TM-T19870

    200mg
    34.00€
    500mg
    54.00€
    1mL*10mM (DMSO)
    33.00€
  • SCH-900271

    CAS:
    SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.
    Formula:C14H16N2O4
    Purity:98.82% - 99.93%
    Color and Shape:Solid
    Molecular weight:276.29

    Ref: TM-T34573

    1mg
    112.00€
    5mg
    261.00€
    10mg
    396.00€
    25mg
    655.00€
    50mg
    888.00€
    100mg
    1,251.00€
    500mg
    2,493.00€
    1mL*10mM (DMSO)
    249.00€
  • Thonzylamine hydrochloride

    CAS:
    Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.
    Formula:C16H23ClN4O
    Purity:99.67%
    Color and Shape:White Crystalline Powder
    Molecular weight:322.83

    Ref: TM-T21014

    5mg
    52.00€
    10mg
    78.00€
    25mg
    119.00€
    50mg
    172.00€
    100mg
    259.00€
  • SAK3

    CAS:
    SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.
    Formula:C20H23N3O4
    Purity:98.37% - 99.43%
    Color and Shape:Solid
    Molecular weight:369.41

    Ref: TM-T26174

    1mg
    120.00€
    5mg
    259.00€
    10mg
    393.00€
    25mg
    623.00€
  • Iperoxo

    CAS:
    Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.
    Formula:C10H17IN2O2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:324.16

    Ref: TM-T25538

    1mg
    50.00€
    5mg
    106.00€
    10mg
    168.00€
    25mg
    339.00€
    50mg
    512.00€
    100mg
    748.00€
    200mg
    1,026.00€
    1mL*10mM (DMSO)
    117.00€
  • rel-(1R,2R)-Vesamicol Hydrochloride

    CAS:
    rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.
    Formula:C17H26ClNO
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:295.85

    Ref: TM-T22486

    2mg
    37.00€
    5mg
    54.00€
    10mg
    82.00€
    25mg
    147.00€
    50mg
    212.00€
    100mg
    313.00€
  • Dimethindene

    CAS:
    Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.
    Formula:C20H24N2
    Purity:98.3% - 98.99%
    Color and Shape:Solid
    Molecular weight:292.42

    Ref: TM-T31488

    1mg
    34.00€
    5mg
    111.00€
    10mg
    163.00€
  • NKY80

    CAS:
    NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.
    Formula:C12H11N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:229.23

    Ref: TM-T16333

    2mg
    47.00€
    5mg
    67.00€
    10mg
    96.00€
    25mg
    187.00€
    50mg
    325.00€
    100mg
    497.00€
    200mg
    715.00€
    1mL*10mM (DMSO)
    105.00€
  • PF-03635659

    CAS:
    PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.
    Formula:C28H32N2O3
    Purity:98.39% - 99.85%
    Color and Shape:Solid
    Molecular weight:444.57

    Ref: TM-T33941

    1mg
    229.00€
    5mg
    560.00€
    10mg
    800.00€
    25mg
    1,216.00€
    50mg
    1,644.00€
    100mg
    2,213.00€
    500mg
    4,436.00€
    1mL*10mM (DMSO)
    640.00€
  • UFP-512

    CAS:
    UFP-512 is a selective delta-opioid (DOP) receptor agonist.
    Formula:C31H33N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:555.62

    Ref: TM-T29046

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • 3-Bromocytisine

    CAS:
    3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7).
    Formula:C11H13BrN2O
    Purity:99.974%
    Color and Shape:Solid
    Molecular weight:269.14

    Ref: TM-T10108

    1mg
    95.00€
    5mg
    202.00€
    10mg
    293.00€
    25mg
    494.00€
    50mg
    710.00€
    100mg
    973.00€
    200mg
    1,305.00€
    1mL*10mM (DMSO)
    178.00€
  • APS3

    CAS:
    APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].
    Formula:C18H7Cl2F6N5O5S2
    Color and Shape:Solid
    Molecular weight:622.31

    Ref: TM-T82981

    5mg
    To inquire
    50mg
    To inquire
  • Muscarine tosylate

    CAS:
    Muscarine ((+)-Muscarine) tosylate, a prototype mAChR agonist, serves as a parasympathetic nervous system stimulant and is recognized for its toxic properties [1] [2].
    Formula:C16H27NO5S
    Color and Shape:Solid
    Molecular weight:345.45

    Ref: TM-T84726

    10mg
    To inquire
    50mg
    To inquire
  • LG 50643

    CAS:
    LG 50643 is a muscarinic antagonist.
    Formula:C24H34INO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.44

    Ref: TM-T25706

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • VU0453595

    CAS:

    VU0453595 is a M1 positive allosteric modulator (PAM).

    Formula:C18H15FN4O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:322.34

    Ref: TM-T29137

    2mg
    46.00€
    5mg
    64.00€
    10mg
    97.00€
    25mg
    182.00€
    50mg
    281.00€
  • VU 0255035

    CAS:

    VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.

    Formula:C18H20N6O3S2
    Purity:98.09% - 98.1%
    Color and Shape:Solid
    Molecular weight:432.52

    Ref: TM-T23508

    1mg
    35.00€
    5mg
    74.00€
    10mg
    111.00€
    25mg
    235.00€
    50mg
    359.00€
    100mg
    533.00€
    200mg
    743.00€
  • PTAC oxalate

    CAS:
    muscarinic receptor ligand
    Formula:C14H21N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.46

    Ref: TM-T23205

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • AR420626

    CAS:
    AR420626: selective FA3R agonist, guards against SALS, effects blocked by BHB, a FA3R antagonist.
    Formula:C21H18Cl2N2O3
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:417.29

    Ref: TM-T26647

    1mg
    34.00€
    5mg
    74.00€
    10mg
    113.00€
    25mg
    245.00€
    50mg
    394.00€
    100mg
    585.00€
    1mL*10mM (DMSO)
    82.00€
  • mAChR antagonist 1

    CAS:
    Compound 4a, a mAChR antagonist, exhibits K i values of 255 nM for M1 and M5 subtypes, and lower values of 121 nM and 158 nM for M3 and M4 subtypes,
    Formula:C19H22N2O2
    Color and Shape:Solid
    Molecular weight:310.39

    Ref: TM-T81888

    5mg
    To inquire
    50mg
    To inquire
  • Cynandione A

    CAS:
    Cynandione A is an acetophenone derived from Cynanchum wilfordii with anti-inflammatory activity.
    Formula:C16H14O6
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:302.28

    Ref: TM-T70277

    1mg
    467.00€
    5mg
    1,054.00€
    10mg
    1,288.00€
    25mg
    1,728.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • ICL-CCIC-0019

    CAS:
    ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.
    Formula:C26H44Br2N4
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:572.46

    Ref: TM-T27579

    2mg
    43.00€
    5mg
    70.00€
    10mg
    92.00€
    25mg
    132.00€
    50mg
    200.00€
    100mg
    344.00€
    200mg
    505.00€
    1mL*10mM (DMSO)
    88.00€
  • N-Demethyl MK-6884

    CAS:
    N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.
    Formula:C24H23N5O
    Color and Shape:Solid
    Molecular weight:397.47

    Ref: TM-T61878

    25mg
    1,288.00€
    50mg
    1,674.00€
    100mg
    2,512.00€