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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • Isopropamide Iodide
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    Isopropamide Iodide

    CAS:
    <p>Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.</p>
    Formula:C23H33IN2O
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:480.43

    Ref: TM-T5051

  • Mc-​Val-​Ala-​PAB
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    Mc-​Val-​Ala-​PAB

    CAS:
    <p>Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).</p>
    Formula:C25H34N4O6
    Purity:98.34% - 99.24%
    Color and Shape:Solid
    Molecular weight:486.56

    Ref: TM-T4289

  • Donepezil Hydrochloride
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    Donepezil Hydrochloride

    CAS:
    <p>Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).</p>
    Formula:C24H29NO3·HCl
    Purity:99.55% - 99.8%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:415.96

    Ref: TM-T6478

  • Nitenpyram
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    Nitenpyram

    CAS:
    <p>Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.</p>
    Formula:C11H15ClN4O2
    Purity:99.03%
    Color and Shape:Light-Yellow Crystal
    Molecular weight:270.72

    Ref: TM-T6607

  • Mecamylamine hydrochloride
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    Mecamylamine hydrochloride

    CAS:
    <p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>
    Formula:C11H22ClN
    Purity:99.76% - >99.99%
    Color and Shape:White Solid
    Molecular weight:203.75

    Ref: TM-T2141

  • Solifenacin hydrochloride
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    Solifenacin hydrochloride

    CAS:
    <p>Solifenacin Hcl is a muscarinic receptor antagonist.</p>
    Formula:C23H27ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.93

    Ref: TM-T23379

  • Encenicline
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    Encenicline

    CAS:
    <p>Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.</p>
    Formula:C16H17ClN2OS
    Purity:99.20%
    Color and Shape:Solid
    Molecular weight:320.84

    Ref: TM-T7193

  • Harman hydrochloride
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    Harman hydrochloride

    CAS:
    <p>Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.</p>
    Formula:C12H11ClN2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:218.68

    Ref: TM-T3158L

  • Oxyphencyclimine Hydrochloride
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    Oxyphencyclimine Hydrochloride

    CAS:
    <p>Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.</p>
    Formula:C20H29ClN2O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:380.91

    Ref: TM-T2138

  • Mecamylamine
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    Mecamylamine

    CAS:
    <p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>
    Formula:C11H21N
    Color and Shape:Solid
    Molecular weight:167.29

    Ref: TM-T69019

  • Propiverine
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    Propiverine

    CAS:
    <p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>
    Formula:C23H29NO3
    Color and Shape:Solid
    Molecular weight:367.48

    Ref: TM-T61438

  • NS 1738
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    NS 1738

    CAS:
    <p>NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)</p>
    Formula:C14H9Cl2F3N2O2
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:365.13

    Ref: TM-T7884

  • Mivacurium dichloride
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    Mivacurium dichloride

    CAS:
    <p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>
    Formula:C58H80Cl2N2O14
    Purity:99.2% - 99.48%
    Color and Shape:Off-White Solid
    Molecular weight:1100.17

    Ref: TM-T22371

  • Fesoterodine
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    Fesoterodine

    CAS:
    <p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>
    Formula:C26H37NO3
    Purity:97.1%
    Color and Shape:Solid
    Molecular weight:411.58

    Ref: TM-T9419

  • Oxyphenonium bromide
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    Oxyphenonium bromide

    CAS:
    <p>Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.</p>
    Formula:C21H34BrNO3
    Purity:98.96%
    Color and Shape:Solid
    Molecular weight:428.404

    Ref: TM-T33846

  • Cyclopentolate Hydrochloride
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    Cyclopentolate Hydrochloride

    CAS:
    <p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>
    Formula:C17H26ClNO3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:327.85

    Ref: TM-T8383

  • A-867744
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    A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Formula:C20H19ClN2O3S
    Purity:95.66%
    Color and Shape:Solid
    Molecular weight:402.89

    Ref: TM-TQ0117

  • DMAB-anabaseine dihydrochloride
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    DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Formula:C19H23Cl2N3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:364.31

    Ref: TM-T22735

  • Propantheline
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    Propantheline

    CAS:
    <p>Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.</p>
    Formula:C23H30NO3
    Color and Shape:Solid
    Molecular weight:368.49

    Ref: TM-T61453

  • MC-Val-Cit-PABC-PNP
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    MC-Val-Cit-PABC-PNP

    CAS:
    <p>MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.</p>
    Formula:C35H43N7O11
    Purity:97.2% - 98.055%
    Color and Shape:Solid
    Molecular weight:737.76

    Ref: TM-T3503