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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • Benzetimide hydrochloride

    CAS:
    <p>Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.</p>
    Formula:C23H27ClN2O2
    Purity:99.32%
    Color and Shape:Off-White Powder
    Molecular weight:398.93
  • mAChR-IN-1 hydrochloride

    CAS:
    <p>mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.</p>
    Formula:C23H26ClIN2O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:524.82
  • Pirmenol

    CAS:
    <p>Pirmenol is a new antiarrhythmic drug</p>
    Formula:C22H30N2O
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:338.49
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Formula:C22H21O2P
    Purity:97.985%
    Color and Shape:White Or Slight Yellow Powder
    Molecular weight:348.37
  • LY2119620

    CAS:
    <p>LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.</p>
    Formula:C19H24ClN5O3S
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:437.94
  • DMAB-anabaseine dihydrochloride

    CAS:
    <p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>
    Formula:C19H23Cl2N3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:364.31
  • Batefenterol

    CAS:
    <p>Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).</p>
    Formula:C40H42ClN5O7
    Purity:97.94% - 98.4%
    Color and Shape:Solid
    Molecular weight:740.24
  • Ilmetropium iodide

    CAS:
    <p>Ilmetropium iodide is a bronchodilator.</p>
    Formula:C20H30INO3
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:459.36
  • Brompheniramine

    CAS:
    <p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>
    Formula:C16H19BrN2
    Color and Shape:Solid
    Molecular weight:319.24
  • Darifenacin

    CAS:
    <p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>
    Formula:C28H30N2O2
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:426.55
  • Nor-benzetimide

    CAS:
    <p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>
    Formula:C16H20N2O2
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:272.34
  • W-84 dibromide

    CAS:
    <p>W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.</p>
    Formula:C32H44Br2N4O4
    Purity:95.56%
    Color and Shape:Solid
    Molecular weight:708.52
  • Ursulcholic acid

    CAS:
    <p>Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.</p>
    Formula:C24H40O10S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:552.7
  • Mivacurium dichloride

    CAS:
    <p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>
    Formula:C58H80Cl2N2O14
    Purity:99.2% - 99.48%
    Color and Shape:Off-White Solid
    Molecular weight:1100.17
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Formula:C19H15Cl2N3O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:388.25
  • Glycopyrrolate

    CAS:
    <p>Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.</p>
    Formula:C19H28BrNO3
    Purity:99.41% - 99.64%
    Color and Shape:Solid
    Molecular weight:398.33
  • Nitrocaramiphen hydrochloride

    CAS:
    <p>Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.</p>
    Formula:C18H27ClN2O4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:370.87
  • Fesoterodine

    CAS:
    <p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>
    Formula:C26H37NO3
    Purity:97.1%
    Color and Shape:Solid
    Molecular weight:411.58
  • 9-Ethyladenine

    CAS:
    <p>9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].</p>
    Formula:C7H9N5
    Purity:99.35% - 99.41%
    Color and Shape:Solid
    Molecular weight:163.18
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Formula:C20H25N3O2
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:339.43