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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 575 products of "AChR"

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  • Azacyclonol hydrochloride
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    Azacyclonol hydrochloride

    CAS:
    <p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>
    Formula:C18H22ClNO
    Color and Shape:Off White Crystalline Powder
    Molecular weight:303.83

    Ref: TM-T0318L

  • Diphenidol
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    Diphenidol

    CAS:
    <p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>
    Formula:C21H27NO
    Color and Shape:Needles From Petroleum Ether Solid
    Molecular weight:309.45

    Ref: TM-T21420

  • Sulindac sulfide
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    Sulindac sulfide

    CAS:
    <p>Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.</p>
    Formula:C20H17FO2S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:340.41

    Ref: TM-T13037

  • N-0861 racemate
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    N-0861 racemate

    CAS:
    <p>N-0861 racemate is the racemate of N-0861.</p>
    Formula:C13H17N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:243.31

    Ref: TM-T12136

  • Sulfoxaflor
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    Sulfoxaflor

    CAS:
    <p>Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.</p>
    Formula:C10H10F3N3OS
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:277.27

    Ref: TM-T19940

  • Sch412348
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    Sch412348

    CAS:
    <p>Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, &gt;1000-fold selectivity vs. other adenosine receptors.</p>
    Formula:C22H21F2N9O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.46

    Ref: TM-T12868

  • SR 16584
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    SR 16584

    CAS:
    <p>α3β4 nAChR antagonist</p>
    Formula:C17H22N2O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:270.37

    Ref: TM-T23388

  • Tarafenacin
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    Tarafenacin

    CAS:
    <p>Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.</p>
    Formula:C21H20F4N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.39

    Ref: TM-T16990

  • Meseclazone
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    Meseclazone

    CAS:
    <p>Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.</p>
    Formula:C11H10ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.65

    Ref: TM-T16353

  • 4-DAMP
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    4-DAMP

    CAS:
    <p>4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in the study of allergic rhinitis and cardiovascular disease.</p>
    Formula:C21H26INO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451.34

    Ref: TM-T22511

  • mAChr-in-1
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    mAChr-in-1

    CAS:
    <p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>
    Formula:C23H25IN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.36

    Ref: TM-T5476

  • Darenzepine
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    Darenzepine

    CAS:
    <p>Darenzepine is a muscarinic receptor inhibitor.</p>
    Formula:C21H21N3O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:347.41

    Ref: TM-T10961

  • UB 165 fumarate
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    UB 165 fumarate

    CAS:
    <p>UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.</p>
    Formula:C17H19ClN2O4
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:350.8

    Ref: TM-T13241

  • CDD0102
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    CDD0102

    CAS:
    <p>CDD0102 is a potent agonist of M1 Muscarinic receptor.</p>
    Formula:C8H12N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:180.21

    Ref: TM-T10731

  • 5-Iodo-A-85380 dihydrochloride
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    5-Iodo-A-85380 dihydrochloride

    CAS:
    <p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>
    Formula:C9H13Cl2IN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.02

    Ref: TM-T22521

  • Dimethyl-W84 (dibromide)
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    Dimethyl-W84 (dibromide)

    CAS:
    <p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>
    Formula:C34H48Br2N4O4
    Color and Shape:Solid
    Molecular weight:736.59

    Ref: TM-T38111

  • LY 2087101
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    LY 2087101

    CAS:
    <p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>
    Formula:C15H11FN2OS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.39

    Ref: TM-T22939

  • AR-R 17779 hydrochloride
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    AR-R 17779 hydrochloride

    CAS:
    <p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>
    Formula:C9H15ClN2O2
    Color and Shape:Solid
    Molecular weight:218.68

    Ref: TM-T21857

  • Elucaine
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    Elucaine

    CAS:
    <p>Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.</p>
    Formula:C19H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.39

    Ref: TM-T15211

  • (R,R)-Glycopyrrolate
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    (R,R)-Glycopyrrolate

    CAS:
    <p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>
    Formula:C19H28BrNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.34

    Ref: TM-T12640