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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • NKY80
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    NKY80

    CAS:
    <p>NKY80 regulates the adenylyl cyclase catalytic activity in heart and lung tissues.</p>
    Formula:C12H11N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:229.23

    Ref: TM-T16333

  • Oxotremorine M iodide
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    Oxotremorine M iodide

    CAS:
    <p>Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.</p>
    Formula:C11H19IN2O
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:322.19

    Ref: TM-T12339

  • Iperoxo
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    Iperoxo

    CAS:
    <p>Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe activation-related conformational transitions of muscarinic receptors.</p>
    Formula:C10H17IN2O2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:324.16

    Ref: TM-T25538

  • Aceclidine
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    Aceclidine

    CAS:
    <p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>
    Formula:C9H15NO2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:169.22

    Ref: TM-T19870

  • Posatirelin
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    Posatirelin

    CAS:
    <p>Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.</p>
    Formula:C17H28N4O4
    Purity:98.08% - 98.87%
    Color and Shape:Solid
    Molecular weight:352.43

    Ref: TM-T34114

  • GSK233705
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    GSK233705

    CAS:
    <p>GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.</p>
    Formula:C24H29BrN2
    Purity:99.87% - 99.98%
    Color and Shape:Solid
    Molecular weight:425.4

    Ref: TM-T31207

  • Temiverine hydrochloride
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    Temiverine hydrochloride

    CAS:
    <p>Temiverine hydrochloride is a potential calcium channel antagonist with anticholinergic effects that inhibits some of the functions of atropine.</p>
    Formula:C24H36ClNO3
    Purity:99.26% - 99.43%
    Color and Shape:Solid
    Molecular weight:422

    Ref: TM-T13118

  • Zamifenacin fumarate
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    Zamifenacin fumarate

    CAS:
    <p>Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.</p>
    Formula:C31H33NO7
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:531.6

    Ref: TM-T13385

  • LG 50643
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    LG 50643

    CAS:
    <p>LG 50643 is a muscarinic antagonist.</p>
    Formula:C24H34INO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.44

    Ref: TM-T25706

  • LY2033298
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    LY2033298

    CAS:
    <p>LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.</p>
    Formula:C13H14ClN3O2S
    Purity:99.06%
    Color and Shape:Solid
    Molecular weight:311.79

    Ref: TM-T27931

  • ICL-CCIC-0019
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    ICL-CCIC-0019

    CAS:
    <p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>
    Formula:C26H44Br2N4
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:572.46

    Ref: TM-T27579

  • PTAC oxalate
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    PTAC oxalate

    CAS:
    <p>muscarinic receptor ligand</p>
    Formula:C14H21N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.46

    Ref: TM-T23205

  • N-Demethyl MK-6884
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    N-Demethyl MK-6884

    CAS:
    <p>N-Demethyl MK-6884 (compound 34) is an M4 mAChR modulator for Alzheimer's and related disease research.</p>
    Formula:C24H23N5O
    Color and Shape:Solid
    Molecular weight:397.47

    Ref: TM-T61878

  • Adenylyl cyclase-IN-1
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    Adenylyl cyclase-IN-1

    CAS:
    <p>Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].</p>
    Formula:C9H8N2S3
    Color and Shape:Solid
    Molecular weight:240.37

    Ref: TM-T83169

  • Tiotropium Bromide hydrate
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    Tiotropium Bromide hydrate

    CAS:
    <p>Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for muscarinic receptors M1, M2, and M3.</p>
    Formula:C19H24BrNO5S2
    Purity:98.44% - 99.41%
    Color and Shape:Solid
    Molecular weight:490.43

    Ref: TM-T6707

  • Timepidium bromide
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    Timepidium bromide

    CAS:
    <p>Timepidium bromide is an agent of anticholinergic.</p>
    Formula:C17H22BrNOS2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.4

    Ref: TM-T12825

  • APS3
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    APS3

    CAS:
    <p>APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].</p>
    Formula:C18H7Cl2F6N5O5S2
    Color and Shape:Solid
    Molecular weight:622.31

    Ref: TM-T82981

  • VU0453595
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    VU0453595

    CAS:
    <p>VU0453595 is a M1 positive allosteric modulator (PAM).</p>
    Formula:C18H15FN4O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:322.34

    Ref: TM-T29137

  • VU 0255035
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    VU 0255035

    CAS:
    <p>VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with an IC50 of 130 nM.</p>
    Formula:C18H20N6O3S2
    Purity:98.09% - 98.1%
    Color and Shape:Solid
    Molecular weight:432.52

    Ref: TM-T23508

  • ABT-418 hydrochloride
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    ABT-418 hydrochloride

    CAS:
    <p>ABT-418 HCl enhances cognition and reduces anxiety as a selective nAChRs agonist, researched for Alzheimer's.</p>
    Formula:C9H15ClN2O
    Color and Shape:Solid
    Molecular weight:202.68

    Ref: TM-T10224