AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Read more
SEN12333
CAS:874450-44-9
SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist
Formula:
C20H25N3O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
339.43
Ref: TM-T23348
| 2mg | 46.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 504.00 € | ||
| 200mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
VU0152100
CAS:409351-28-6
VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 …
Formula:
C18H19N3O2S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
341.43
Ref: TM-T17238
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 487.00 € | ||
| 100mg | 731.00 € | ||
| 200mg | 1,023.00 € | ||
| 500mg | 1,542.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Aclidinium bromide
CAS:320345-99-1
Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant …
Formula:
C26H30NO4S2·Br
Purity:
98.93% - 99.69%
Color and Shape:
Solid
Molecular weight:
564.55
Ref: TM-T2555
| 2mg | 44.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 229.00 € | ||
| 100mg | 343.00 € | ||
| 500mg | 806.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Umeclidinium bromide
CAS:869113-09-7
Umeclidinium bromide (GSK573719A) is a novel mAChR antagonist.
Formula:
C29H34BrNO2
Purity:
98.40% - 99.09%
Color and Shape:
Solid
Molecular weight:
508.49
Ref: TM-T4997
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 514.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ursulcholic acid
CAS:88426-32-8
Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.
Formula:
C24H40O10S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
552.7
Ref: TM-T68019
| 5mg | 45.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 225.00 € | ||
| 500mg | 634.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Benzetimide hydrochloride
CAS:5633-14-7
Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.
Formula:
C23H27ClN2O2
Purity:
99.32%
Color and Shape:
Off-White Powder
Molecular weight:
398.93
Ref: TM-T7561
| 10mg | 35.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 62.00 € | ||
| 100mg | 84.00 € | ||
| 200mg | 109.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mepenzolate Bromide
CAS:76-90-4
Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.
Formula:
C21H26BrNO3
Purity:
95.73% - 99.21%
Color and Shape:
Solid
Molecular weight:
420.34
Ref: TM-T0794
| 100mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Propoxur
CAS:114-26-1
Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; …
Formula:
C11H15NO3
Purity:
98% - 98.15%
Color and Shape:
Minute Crystals (Niosh 2016)
Molecular weight:
209.24
Ref: TM-T0976
| 1g | 90.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 45.00 € | ||
| 500mg | 69.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CDD0102
CAS:146422-58-4
CDD0102 is a potent agonist of M1 Muscarinic receptor.
Formula:
C8H12N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
180.21
Ref: TM-T10731
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Posatirelin
CAS:78664-73-0
Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.
Formula:
C17H28N4O4
Purity:
97.41% - 98.22%
Color and Shape:
Solid
Molecular weight:
352.43
Ref: TM-T34114
| 1mg | 125.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 733.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,383.00 € | ||
| 500mg | 2,749.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Phenserine
CAS:101246-66-6
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
Formula:
C20H23N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
337.42
Ref: TM-T12446
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
JNJ-39393406
CAS:953428-73-4
JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco …
Formula:
C19H18F2N6O3
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
416.38
Ref: TM-T27679
| 1mg | 141.00 € | ||
| 5mg | 326.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,974.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CP-810123
CAS:439608-12-5
CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or …
Formula:
C14H18N4O
Purity:
98.63% - 99.23%
Color and Shape:
Solid
Molecular weight:
258.32
Ref: TM-T31079
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Thonzylamine hydrochloride
CAS:63-56-9
Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.
Formula:
C16H23ClN4O
Purity:
99.84%
Color and Shape:
White Crystalline Powder
Molecular weight:
322.83
Ref: TM-T21014
| 5mg | 54.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 267.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Otenzepad
CAS:102394-31-0
Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM …
Formula:
C24H31N5O2
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
421.54
Ref: TM-T16411
| 1mg | 46.00 € | ||
| 2mg | 36.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 266.00 € | ||
| 50mg | 427.00 € | ||
| 100mg | 631.00 € | ||
| 200mg | 530.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
MHP 133
CAS:147340-43-0
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
Formula:
C17H20ClN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.83
Ref: TM-T13772
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
9-CP-Ade Mesylate
CAS:189639-09-6
9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate …
Formula:
C11H17N5O3S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
299.35
Ref: TM-T23588
| 1mg | 66.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 389.00 € | ||
| 50mg | 575.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GP531
CAS:142344-87-4
GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.
Formula:
C16H21N5O4
Color and Shape:
Solid
Molecular weight:
347.37
Ref: TM-T13713
| 25mg | 1,406.00 € | ||
| 50mg | 1,854.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
N-0861 racemate
CAS:121241-87-0
N-0861 racemate is the racemate of N-0861.
Formula:
C13H17N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
243.31
Ref: TM-T12136
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Vesamicol hydrochloride
CAS:120447-62-3
Vesamicol hydrochloride ((±)-AH5183 hydrochloride) is a acetylcholine transport inhibitor.
Formula:
C17H26ClNO
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
295.85
Ref: TM-T22486
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 322.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
