AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Darenzepine
CAS:84629-61-8
Darenzepine is a muscarinic receptor inhibitor.
Formula:
C21H21N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
347.41
Ref: TM-T10961
| 1mg | 210.00 € | ||
| 5mg | 417.00 € | ||
| 10mg | 585.00 € | ||
| 25mg | 869.00 € | ||
| 50mg | 1,161.00 € | ||
| 100mg | 1,569.00 € | ||
| 1mL*10mM (DMSO) | 469.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
UB 165 fumarate
CAS:2454492-43-2
UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM …
Formula:
C17H19ClN2O4
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T13241
| 1mg | 327.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,321.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Tematropium
CAS:113932-41-5
Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.
Formula:
C21H31NO8S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
457.54
Ref: TM-T10732
| 1mg | 209.00 € | ||
| 2mg | 279.00 € | ||
| 5mg | 441.00 € | ||
| 10mg | 606.00 € | ||
| 25mg | 914.00 € | ||
| 50mg | 1,224.00 € | ||
| 100mg | 1,663.00 € | ||
| 1mL*10mM (DMSO) | 499.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
TZ3O
CAS:2218754-19-7
TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type …
Formula:
C18H13NO4S
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
339.37
Ref: TM-T77678
| 1mg | 183.00 € | ||
| 5mg | 453.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,395.00 € | ||
| 100mg | 1,844.00 € | ||
| 500mg | 3,679.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
VU0453595
CAS:1432436-13-9
VU0453595 is a M1 positive allosteric modulator (PAM).
Formula:
C18H15FN4O
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
322.34
Ref: TM-T29137
| 2mg | 44.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 175.00 € | ||
| 50mg | 271.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Timepidium bromide
CAS:35035-05-3
Timepidium bromide is an agent of anticholinergic.
Formula:
C17H22BrNOS2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
400.4
Ref: TM-T12825
| 25mg | 1,688.00 € | ||
| 50mg | 2,226.00 € | ||
| 100mg | 2,899.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Tiotropium Bromide hydrate
CAS:411207-31-3
Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for …
Formula:
C19H24BrNO5S2
Purity:
98.44% - 99.41%
Color and Shape:
Solid
Molecular weight:
490.43
Ref: TM-T6707
| 25mg | 43.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 131.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
BuChE-IN-TM-10
CAS:2313524-95-5
TM-10: Potent BuChE inhibitor, IC50 8.9 nM, disaggregates Aβ, antioxidant, BBB penetrant, may treat Alzheimer's.
Formula:
C32H38N2O3
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
498.66
Ref: TM-T10630
| 1mg | 183.00 € | ||
| 2mg | 272.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 615.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,290.00 € | ||
| 100mg | 1,755.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
VU 0255035
CAS:1135243-19-4
VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with …
Formula:
C18H20N6O3S2
Purity:
96.53% - 98.26%
Color and Shape:
Solid
Molecular weight:
432.52
Ref: TM-T23508
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 532.00 € | ||
| 500mg | 1,095.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
ICL-CCIC-0019
CAS:936498-64-5
ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.
Formula:
C26H44Br2N4
Purity:
97.62%
Color and Shape:
Solid
Molecular weight:
572.46
Ref: TM-T27579
| 1mg | 183.00 € | ||
| 5mg | 410.00 € | ||
| 10mg | 606.00 € | ||
| 25mg | 926.00 € | ||
| 50mg | 1,295.00 € | ||
| 100mg | 1,745.00 € | ||
| 500mg | 3,475.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
3-Bromocytisine
CAS:207390-14-5
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for …
Formula:
C11H13BrN2O
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
269.14
Ref: TM-T10108
| 1mg | 93.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 302.00 € | ||
| 25mg | 509.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,007.00 € | ||
| 1mL*10mM (DMSO) | 207.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Zamifenacin fumarate
CAS:127308-98-9
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
Formula:
C31H33NO7
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
531.6
Ref: TM-T13385
| 1mg | 40.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 618.00 € | ||
| 500mg | 1,299.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
LY2033298
CAS:886047-13-8
LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.
Formula:
C13H14ClN3O2S
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
311.79
Ref: TM-T27931
| 1mg | 96.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 343.00 € | ||
| 25mg | 776.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,420.00 € | ||
| 500mg | 2,759.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
AChE/BChE-IN-10
CAS:2924824-48-4
AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.
Formula:
C26H30N2O2
Purity:
99.75%
Color and Shape:
Soild
Molecular weight:
402.53
Ref: TM-T61969
| 5mg | 46.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 301.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Levamisole hydrochloride
CAS:16595-80-5
Levamisole hydrochloride ((-)-Tetramisole hydrochloride) is an antihelminthic drug that has been tried experimentally in rheumatic …
Formula:
C11H12N2S·HCl
Purity:
99.89%
Color and Shape:
White To Almost White Crystalline Powder
Molecular weight:
240.75
Ref: TM-T0944
| 5g | Discontinued | Request information | |
| 10g | Discontinued | Request information | |
| 10mg | Discontinued | Request information |
Carbachol
CAS:51-83-2
Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation …
Formula:
C6H15ClN2O2
Purity:
100% - 90%
Color and Shape:
Liquid
Molecular weight:
182.65
Ref: TM-T0105
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
Scopolamine butylbromide
CAS:149-64-4
Scopolamine butylbromide ((-)-Scopolamine butylbromide) is a competitive antagonist of mAChR (IC50: 55.3 ± 4.3 nM).
Formula:
C21H30NO4·Br
Purity:
99.95%
Color and Shape:
White Powder
Molecular weight:
440.37
Ref: TM-T2183
| 20mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
