Serine Protease
Serine protease inhibitors are compounds that target and inhibit serine proteases, a group of enzymes characterized by a serine residue at their active site. These proteases are involved in numerous physiological processes, including digestion, immune response, blood coagulation, and inflammation. Serine protease inhibitors are important for studying diseases where these enzymes are dysregulated, such as cardiovascular diseases, cancer, and inflammatory conditions. At CymitQuimica, we provide serine protease inhibitors to support your research in enzymology, disease mechanisms, and therapeutic interventions.
Found 85 products for "Serine Protease".
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TAO Kinase inhibitor 2
CAS:TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.Formula:C25H24N2O3Purity:98.58%Color and Shape:SolidMolecular weight:400.4697Chlorobenzothiazolinone
CAS:Chlorobenzothiazolinone blocks human chymase at 90 μM, assessed by fluorescence using a specific peptide substrate after 1 hr.Formula:C7H4ClNOSPurity:99.42% - 99.77%Color and Shape:SolidMolecular weight:185.631BAY-85-8501
CAS:BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Formula:C22H17F3N4O3SPurity:99.16%Color and Shape:SolidMolecular weight:474.456Tilpisertib fosmecarbil TFA
CAS:Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.Formula:C37H37ClF3N8O9PColor and Shape:SolidMolecular weight:861.16Chymotrypsinogen
CAS:Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .Color and Shape:SolidLonodelestat TFA
Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.Formula:C73H112F3N15O21Color and Shape:SolidMolecular weight:1592.75Roseltide rT1
CAS:Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.Formula:C110H177N31O31S6Color and Shape:SolidMolecular weight:2622.16KKI-5
CAS:KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.Formula:C35H55N11O9Purity:98%Color and Shape:SolidMolecular weight:773.88α 1 Antichymotrypsin, Human Plasma
CAS:Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.Color and Shape:SolidSafflower oil (from Carthamus tinctorius seed)
CAS:Safflower oil (from Carthamus tinctorius seed) contains unsaturated fatty acids, tocopherols and phenolic compounds, which has antioxidant and lipid metabolism regulating activities, can scavenge free radicals and inhibit collagenase and elastase activities, and is often used in skin aging, atherosclerosis and functional oil-related research.CDD-3290
CDD-3290 serves as a functional therapeutic tool specifically designed to enable the precise detection and inhibition of the proteolytic activity of PSA which plays a pivotal role in the progression of prostate cancer during strictly monitored laboratory observation periods and molecular investigations to evaluate the pharmacological potential of targeted kallikrein inhibition in specialized preclinical research environments.Formula:C17H14N6O2Purity:99.06% - 99.13%Color and Shape:White SolidMolecular weight:334.33Kallikrein 5-IN-2 TFA
Kallikrein5-IN-2 TFA is the trifluoroacetate salt form of Kallikrein5-IN-2. It acts as a selective inhibitor of kallikrein5 (KLK5), with a pIC50 value of 7.1. Kallikrein5-IN-2 TFA exhibits no phototoxicity at 100 μg/mL and is non-irritating. The compound remains stable in non-oxidative conditions within a pH range of 4 to 8. Kallikrein5-IN-2 shows potential for improving Netherton syndrome.Formula:C25H23F3N6O3Color and Shape:SolidMolecular weight:512.17837hCAXII-IN-10
hCAXII-IN-10 (Compound 18b) acts as a dual inhibitor of human carbonic anhydrase isoenzyme XII (hCAXII) and cathepsin B, with a Ki value of 2.2 nM. It inhibits the function of hCAXII in creating a pH microenvironment conducive to tumor growth, showing promise for use in cancer research.Color and Shape:Odour SolidSuc-AAP-Abu-pNA
CAS:Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Formula:C25H34N6O9Color and Shape:SolidMolecular weight:562.57Tiprelestat
CAS:Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.Formula:C254H416N72O75S10Color and Shape:SolidMolecular weight:5999.09Z-APF-CMK
CAS:Z-APF-CMK is a selective inhibitor of the calcium (Ca2+)-regulated nuclear scaffold protease (CRNSP), as reported in reference [1].Formula:C26H30ClN3O5Color and Shape:SolidMolecular weight:499.99SFTI-1
CAS:SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.Formula:C67H104N18O18S2Color and Shape:SolidMolecular weight:1513.78Protease Inhibitor Library
A unique collection of xnum protease and proteasome inhibitors for research in chemical genomics, and drug screening;Color and Shape:Odour SolidMeOSuc-AAPA-CMK
MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].Formula:C20H31ClN4O8Color and Shape:SolidMolecular weight:490.94Dansyl-Glu-Gly-Arg-Chloromethylketone
CAS:Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activatedFormula:C26H36ClN7O7SColor and Shape:SolidMolecular weight:626.12
