VEGFR
VEGFR (Vascular Endothelial Growth Factor Receptor) inhibitors are compounds that block the signaling of VEGFR, a key receptor in the VEGF pathway, which is crucial for angiogenesis. VEGFR inhibitors prevent the formation of new blood vessels that supply nutrients and oxygen to tumors, thereby inhibiting tumor growth. These inhibitors are widely used in cancer therapy and research to study the mechanisms of angiogenesis and develop anti-cancer treatments. At CymitQuimica, we provide a comprehensive range of high-quality VEGFR inhibitors to support your research in oncology, vascular biology, and angiogenesis.
Read more
CP-547632
CAS:252003-65-9
CP-547632 is an oral ATP-competitive inhibitor of VEGFR-2/FGF kinase with IC50s of 11/9 nM, highly …
Formula:
C20H24BrF2N5O3S
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
532.4
Ref: TM-T10870L
| 1mg | 36.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 241.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
VEGFR-3-IN-1
CAS:2756668-73-0
VEGFR-3-IN-1, a potent VEGFR3 inhibitor (IC50=110.4 nM), hinders tumor growth and VEGFR3 signaling, affecting HDLEC …
Formula:
C29H29ClF3N7OS
Purity:
99.52%
Color and Shape:
Liquid
Molecular weight:
616.1
Ref: TM-T72924
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 579.00 € | ||
| 100mg | 928.00 € | ||
| 500mg | 1,850.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
MMPP
CAS:1895957-18-2
MMPP is a VEGFR2 inhibitor with anti-inflammatory activity, inhibits STAT3 , inhibits angiogenesis, and can …
Formula:
C17H18O3
Purity:
100% - 99.22%
Color and Shape:
Solid
Molecular weight:
270.32
Ref: TM-T28077
| 1mg | 238.00 € | ||
| 5mg | 590.00 € | ||
| 10mg | 843.00 € | ||
| 25mg | 1,266.00 € | ||
| 50mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
PKI-166
CAS:187724-61-4
PKI-166: oral EGF-R tyrosine kinase inhibitor (IC50: 0.7 nM), halts growth & spread of many …
Formula:
C20H18N4O
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
330.38
Ref: TM-T16549
| 1mg | 42.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 189.00 € | ||
| 25mg | 370.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 985.00 € | ||
| 200mg | 1,332.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
AMG-Tie2-1
CAS:870223-96-4
AMG-Tie2-1 is a Tie2 and VEGFR2 inhibitor with anticancer and antitumor activity for the study …
Formula:
C25H20F3N5O2
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
479.45
Ref: TM-T22259
| 1mg | 52.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 366.00 € | ||
| 50mg | 623.00 € | ||
| 100mg | 1,017.00 € | ||
| 200mg | 1,527.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Chiauranib
CAS:1256349-48-0
Chiauranib, a potent anticancer agent, inhibits angiogenesis kinases (VEGFR1-3, PDGFRα, c-Kit), Aurora B, and CSF1R …
Formula:
C27H21N3O3
Purity:
96.25%
Color and Shape:
Solid
Molecular weight:
435.47
Ref: TM-T35570
| 1mg | 89.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 508.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,003.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
(E)-FeCP-oxindole
CAS:884338-18-5
(E)-FeCP-oxindole is an inhibitor of VEGFR2 with IC50 of 214 nM.
Formula:
C19H15FeNO
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
329.17
Ref: TM-T22755
| 1mg | 72.00 € | ||
| 5mg | 147.00 € | ||
| 10mg | 214.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 509.00 € | ||
| 100mg | 693.00 € | ||
| 200mg | 912.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
DMH4
CAS:515880-75-8
DMH4 is a potent and selective inhibitor of VEGFR2 with an IC50 of 0.16 µM.
Formula:
C24H24N4O2
Purity:
98.68%
Color and Shape:
Solid
Molecular weight:
400.47
Ref: TM-T22737
| 1mg | 41.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 244.00 € | ||
| 100mg | 361.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Naphazoline
CAS:835-31-4
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity.
Formula:
C14H14N2
Purity:
99.25%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
210.27
Ref: TM-T21445
| 5mg | 54.00 € | ||
| 10mg | 76.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 231.00 € | ||
| 500mg | 497.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Pz-1
CAS:1800505-64-9
Pz-1 is an inhibitor of VEGFR2 and RET (rearranged during transfection) tyrosine kinase that blocks …
Formula:
C26H26N6O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
454.52
Ref: TM-T12598
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 255.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
AMPK-IN-3
CAS:2417674-27-0
AMPK-IN-3: potent, selective AMPK (α2/α1) & KDR inhibitor; IC50: 60.7/107/3820 nM; anticancer in K562 cells.
Formula:
C25H33N5O3
Purity:
99.13%
Color and Shape:
Liquid
Molecular weight:
451.56
Ref: TM-T62745
| 1mg | 108.00 € | ||
| 5mg | 246.00 € | ||
| 10mg | 395.00 € | ||
| 25mg | 810.00 € | ||
| 50mg | 1,086.00 € | ||
| 100mg | 1,473.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
VEGFR-2-IN-6
CAS:444731-47-9
VEGFR-2-IN-6 (WO 02/059110, example 64) is a potent inhibitor of VEGFR2, a crucial receptor involved …
Formula:
C20H21N7O2S
Purity:
99.01%
Color and Shape:
Liquid
Molecular weight:
423.49
Ref: TM-T37078
| 1mg | 95.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 244.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
TG 100572
CAS:867334-05-2
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src …
Formula:
C26H26ClN5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
475.97
Ref: TM-T13156
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
Ansornitinib
CAS:1448874-96-1
Ansornitinib (ANG-3070) is a KDR and PDGF receptor inhibitor with antifibrotic activity for the study …
Formula:
C30H32N6O4
Color and Shape:
Liquid
Molecular weight:
540.61
Ref: TM-T63809
| 1mg | 138.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 993.00 € | ||
| 50mg | 1,568.00 € | ||
| 100mg | 2,319.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
(Z)-FeCP-oxindole
CAS:1137967-28-2
(Z)-FeCP-oxindole is a selective inhibitor of VEGFR2 with an IC50 of 200 nM for human. …
Formula:
C19H15FeNO
Purity:
100% - 98.13%
Color and Shape:
Solid
Molecular weight:
329.17
Ref: TM-T23554
| 1mg | 42.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 543.00 € | ||
| 500mg | 1,144.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
CGP60474
CAS:164658-13-3
CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive …
Formula:
C18H18ClN5O
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
355.82
Ref: TM-T14943
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 537.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
TG 100801 Hydrochloride
CAS:1018069-81-2
TG 100801: prodrug for macular degeneration. TG 100572: inhibits kinases (VEGFRs, FGFRs, PDGFRβ, Src family), …
Formula:
C33H31Cl2N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
616.54
Ref: TM-T13157L
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
BMS-605541
CAS:639858-32-5
BMS-605541 is a potent and selective inhibitor of vascular endothelial growth factor receptor-2 (VEGFR-2) kinase …
Formula:
C19H17F2N5OS
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
401.43
Ref: TM-T26852
| 5mg | 49.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 239.00 € | ||
| 100mg | 353.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Tuesday 4 Feb 2025
WAY-600
CAS:1062159-35-6
WAY-600 is a potent, ATP-competitive and selective inhibitor of mTOR with IC50 of 9 nM; …
Formula:
C28H30N8O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
494.59
Ref: TM-T6730
| 1mg | 38.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 355.00 € | ||
| 100mg | 495.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Brolucizumab
CAS:1531589-13-5
Brolucizumab (DLX1008) is a single-chain anti-VEGF-A antibody fragment exhibiting low picomolar affinity (K D = …
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T80593
| 1mg | 233.00 € | ||
| 5mg | 607.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,439.00 € | ||
| 50mg | 1,862.00 € | ||
| 100mg | 2,623.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
