VEGFR
VEGFR (Vascular Endothelial Growth Factor Receptor) inhibitors are compounds that block the signaling of VEGFR, a key receptor in the VEGF pathway, which is crucial for angiogenesis. VEGFR inhibitors prevent the formation of new blood vessels that supply nutrients and oxygen to tumors, thereby inhibiting tumor growth. These inhibitors are widely used in cancer therapy and research to study the mechanisms of angiogenesis and develop anti-cancer treatments. At CymitQuimica, we provide a comprehensive range of high-quality VEGFR inhibitors to support your research in oncology, vascular biology, and angiogenesis.
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AMG-47a
CAS:882663-88-9
AMG-47a inhibits Lck, T cell growth, and degrades KRAS oncoprotein, affecting EGFP-KRASG12V but not EGFP.
Formula:
C29H28F3N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
535.56
Ref: TM-T7123
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 532.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Xanthatin
CAS:26791-73-1
Xanthatin exhibits cytotoxic, antibacterial, antifungal properties, may treat NSCLC, and inhibits melanoma by targeting Wnt/β-catenin …
Formula:
C15H18O3
Purity:
98% - 99.39%
Color and Shape:
Solid
Molecular weight:
246.3
Ref: TM-T3S0153
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Dovitinib lactate
CAS:692737-80-7
Dovitinib lactate (TKI-258 lactate)(TKI258) lactate is a potent inhibitor of fibroblast growth factor receptor 3 …
Formula:
C24H27FN6O4
Purity:
98.44% - 99.54%
Color and Shape:
Solid
Molecular weight:
482.51
Ref: TM-T7104
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 350.00 € | ||
| 200mg | 523.00 € | ||
| 500mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
AAL-993
CAS:269390-77-4
AAL-993: VEGFR inhibitor; IC50: 130 nM (1), 23 nM (2), 18 nM (3); weak on …
Formula:
C20H16F3N3O
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
371.36
Ref: TM-T21593
| 1mg | 45.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 427.00 € | ||
| 100mg | 631.00 € | ||
| 500mg | 1,328.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
RAF265
CAS:927880-90-8
RAF265 (CHIR-265) inhibits C-Raf/B-Raf/V600E (IC50: 3-60 nM), blocks VEGFR2 (EC50: 30 nM), in Phase 2 …
Formula:
C24H16F6N6O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
518.41
Ref: TM-T6296
| 1mg | 46.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 625.00 € | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
NVP-BAW2881
CAS:861875-60-7
NVP-BAW2881 (BAW2881) is a potent and selective VEGFR inhibitor with activity to inhibit chronic and …
Formula:
C22H15F3N4O2
Purity:
98.19% - 99.97%
Color and Shape:
Solid
Molecular weight:
424.38
Ref: TM-T3641
| 1mg | 36.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 490.00 € | ||
| 500mg | 1,087.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
SU5205
CAS:3476-86-6
SU5205 is a VEGFR2 inhibitor.
Formula:
C15H10FNO
Purity:
99.67% - 99.68%
Color and Shape:
Solid
Molecular weight:
239.24
Ref: TM-T3566
| 25mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Foretinib
CAS:849217-64-7
Foretinib (GSK1363089) is a broad-spectrum tyrosine kinase inhibitor with IC50s of 0.4 nM and 0.9 …
Formula:
C34H34F2N4O6
Purity:
98.07% - 99.7%
Color and Shape:
Solid
Molecular weight:
632.65
Ref: TM-T3113
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 349.00 € | ||
| 500mg | 829.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Vorolanib
CAS:1013920-15-4
Vorolanib (X-82) is an orally active VEGFR/PDGFR dual inhibitor.
Formula:
C23H26FN5O3
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
439.48
Ref: TM-T8491
| 1mg | 111.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 618.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Fruquintinib
CAS:1194506-26-7
Fruquintinib (HMPL-013) is an orally available, small molecule inhibitor of vascular endothelial growth factor receptors …
Formula:
C21H19N3O5
Purity:
98.84% - 99.89%
Color and Shape:
Solid
Molecular weight:
393.39
Ref: TM-T2656
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 245.00 € | ||
| 500mg | 609.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Orantinib
CAS:252916-29-3
Orantinib (NSC 702827) , a excellent effective against PDGFR autophosphorylation with Ki of 8 nM, …
Formula:
C18H18N2O3
Purity:
100% - 98.01%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T6184
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 480.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
AG-13958
CAS:319460-94-1
AG-13958 (AG-013958) (AG-013958), a potent VEGFR tyrosine kinase inhibitor, for the treatment of age-related macular …
Formula:
C26H22FN7O
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
467.5
Ref: TM-T7493
| 1mg | 94.00 € | ||
| 5mg | 257.00 € | ||
| 10mg | 396.00 € | ||
| 25mg | 637.00 € | ||
| 50mg | 918.00 € | ||
| 100mg | 1,220.00 € | ||
| 1mL*10mM (DMSO) | 268.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Motesanib
CAS:453562-69-1
Motesanib (AMG 706) orally blocks VEGFR, PDGFR, Kit, Ret; curbing angiogenesis and cancer cell growth.
Formula:
C22H23N5O
Purity:
98% - 98.87%
Color and Shape:
Solid
Molecular weight:
373.45
Ref: TM-T2288
| 5mg | 44.00 € | ||
| 10mg | 58.00 € | ||
| 50mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
KRN-633
CAS:286370-15-8
KRN-633 is an effective VEGFR inhibitor. The IC50s of KRN-633(KRN633) for VEGFR1, VEGFR2, and VEGFR3 …
Formula:
C20H21ClN4O4
Purity:
99.22% - 99.65%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T6137
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 430.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
JI-101
CAS:900573-88-8
JI-101 (CGI-1842) is an oral multi-kinase inhibitor that targets VEGFR-2, PDGFR-β, and EphB4.
Formula:
C22H20BrN5O2
Purity:
99.35% - 99.41%
Color and Shape:
Solid
Molecular weight:
466.33
Ref: TM-T3476
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Ilorasertib
CAS:1227939-82-3
Ilorasertib (ABT-348) inhibits Aurora kinases A/B/C & RET, PDGFRβ, Flt1 (IC50: 1-120 nM).
Formula:
C25H21FN6O2S
Purity:
96.17% - 98.03%
Color and Shape:
Solid
Molecular weight:
488.54
Ref: TM-TQ0059
| 1mg | 39.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 397.00 € | ||
| 200mg | 552.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Cediranib
CAS:288383-20-0
Cediranib (AZD2171) is a potent KDR tyrosine kinase inhibitor (IC50 < 1nM), also targets Flt1/4, PDGFRβ, …
Formula:
C25H27FN4O3
Purity:
97.21% - 99.94%
Color and Shape:
Solid
Molecular weight:
450.51
Ref: TM-T2500
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 175.00 € | ||
| 100mg | 248.00 € | ||
| 200mg | 454.00 € | ||
| 500mg | 729.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
SCR-1481B1
CAS:1174161-86-4
SCR-1481B1 (c-Met inhibitor 2) has activity against cancers dependent on Met activation and also has …
Formula:
C32H40ClF2N6O13P
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
821.12
Ref: TM-T5349
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 206.00 € | ||
| 50mg | 344.00 € | ||
| 100mg | 510.00 € | ||
| 1mL*10mM (DMSO) | 107.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Oglufanide
CAS:38101-59-6
Oglufanide (H-Glu-Trp-OH) is a naturally occurring thymic immunomodulator,and inhibits vascular endothelial growth factor (VEGF).
Formula:
C16H19N3O5
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
333.34
Ref: TM-T7203
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 523.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
EOC317
CAS:939805-30-8
EOC317 (ACTB-1003) is an oral kinase inhibitor (IC50: 6/2/4 nM, for FGFR1/VEGFR2/Tie-2).
Formula:
C27H26F5N7O3
Purity:
98.00% - 99.26%
Color and Shape:
Solid
Molecular weight:
591.53
Ref: TM-T4318
| 1mg | 90.00 € | ||
| 2mg | 132.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,077.00 € | ||
| 1mL*10mM (DMSO) | 253.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
