Bombesin Receptor
Bombesin receptors are a group of GPCRs that are activated by bombesin-like peptides, which are involved in regulating gastrointestinal function, energy balance, and cell proliferation. These receptors are of particular interest in cancer research, as they are often overexpressed in certain types of tumors. Bombesin receptor antagonists are studied for their potential as cancer therapeutics. At CymitQuimica, we provide a selection of high-quality bombesin receptor modulators to support your research in oncology, gastrointestinal physiology, and receptor signaling.
Found 35 products of "Bombesin Receptor"
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Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29Kuwanon H
CAS:Kuwanon H is a potent non-peptide GRP receptor antagonist with a Ki of 290 nM, useful in GRP-related studies.Formula:C45H44O11Purity:97.09% - 97.99%Color and Shape:SolidMolecular weight:760.82Bombesin acetate(31362-50-2 free base)
CAS:Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).Formula:C73H114N24O20SPurity:98.44%Color and Shape:SolidMolecular weight:1679.92BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.Formula:C59H80N14O13Purity:95.3%Color and Shape:SolidMolecular weight:1193.35[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C77H118N22O20Purity:98.41% - 99.14%Color and Shape:SolidMolecular weight:1671.9[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C76H116N22O20SPurity:99.81%Color and Shape:SolidMolecular weight:1689.94kuwanon G
CAS:Kuwanon G (Moracenin B) may be used to treat the type II diabetes mellitus as a dual inhibitor of PTP1B and α-glucosidase and as an insulin sensitiser.Formula:C40H36O11Purity:98% - 99.57%Color and Shape:SolidMolecular weight:692.71Ref: TM-T3S1612
1mg63.00€5mg138.00€1mL*10mM (DMSO)178.00€10mg198.00€25mg321.00€50mg465.00€100mg627.00€200mg845.00€Litorin
CAS:Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.Formula:C51H68N14O11SColor and Shape:White PowderMolecular weight:1085.24MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurity:98.56%Color and Shape:SolidMolecular weight:444.37DSO-5a
CAS:DSO-5a, a potent and selective orally active BB3 agonist, is a DMAKO-00 derivative that enhances ppar-γ activity via BB3 and stimulates ERK1/2 phosphorylation.Formula:C23H24N2O7Purity:98%Color and Shape:SolidMolecular weight:440.45Bag-1
CAS:Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.Formula:C22H27N3Color and Shape:SolidMolecular weight:333.47PD 168368
CAS:PD 168368 is a mixed neuromodulin B receptor (NMB-R) antagonist and potent FPR1/FPR2/FPR3 agonist that inhibits the gastrin-releasing peptide receptor.Formula:C31H34N6O4Purity:98.11% - 99.87%Color and Shape:SolidMolecular weight:554.64Ref: TM-T8691
1mg84.00€5mg167.00€1mL*10mM (DMSO)197.00€10mg245.00€25mg492.00€50mg737.00€100mg1,054.00€PD 165929
CAS:PD 165929 is a selective antagonist of Bombesin BB1.Formula:C37H47N5O2Purity:98%Color and Shape:SolidMolecular weight:593.8GRPR antagonist-1
GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.Formula:C29H33F3N4O4Color and Shape:SolidMolecular weight:558.59GRPR antagonist-2
GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).Formula:C28H32F3N5O4Color and Shape:SolidMolecular weight:559.58
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