Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
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Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Formula:C13H22N6Purity:99.84%Color and Shape:SolidMolecular weight:262.35FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.55ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Formula:C24H28ClNO2Purity:98%Color and Shape:SolidMolecular weight:397.94H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Formula:C11H11BrN8Color and Shape:SolidMolecular weight:335.16(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formula:C23H32N6O3SPurity:99.54%Color and Shape:SolidMolecular weight:472.6Ref: TM-T10000
1mg140.00€5mg269.00€1mL*10mM (DMSO)350.00€10mg389.00€25mg610.00€50mg820.00€100mg1,063.00€Azelastine
CAS:Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.Formula:C22H24ClN3OPurity:99.35% - 99.99%Color and Shape:White Crystal PowderMolecular weight:381.90Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Formula:C8H10N6SPurity:98%Color and Shape:SolidMolecular weight:222.27JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFormula:C13H15ClN4OColor and Shape:SolidMolecular weight:278.74Alimemazine
CAS:Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.Formula:C18H22N2SPurity:98%Color and Shape:Crystals SolidMolecular weight:298.45Aminopotentidine
CAS:H2 antagonistFormula:C26H35N7O2Purity:98%Color and Shape:SolidMolecular weight:477.6Zolantidine dimaleate
CAS:H2 receptor antagonistFormula:C26H31N3O5SPurity:98%Color and Shape:SolidMolecular weight:497.61BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Formula:C12H19N5O2S2Purity:98%Color and Shape:SolidMolecular weight:329.44ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Formula:C22H22N2OPurity:99.94%Color and Shape:SolidMolecular weight:330.42Ref: TM-T14087
1mg44.00€1mL*10mM (DMSO)90.00€5mg93.00€10mg133.00€25mg270.00€50mg409.00€100mg595.00€200mg833.00€(R)-Mequitazine
CAS:(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.Formula:C20H22N2SColor and Shape:SolidMolecular weight:322.47A-304121
CAS:A-304121 is a histamine H(3) receptor.Formula:C20H29N3O3Color and Shape:SolidMolecular weight:359.46OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98JNJ 10181457 dihydrochloride
CAS:JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.Formula:C20H28N2OPurity:98%Color and Shape:SolidMolecular weight:312.45Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Formula:C18H20N2Purity:99.85%Color and Shape:SolidMolecular weight:264.36Wy 49051
CAS:Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).Formula:C28H33N5O3Purity:99.89%Color and Shape:SolidMolecular weight:487.59Ref: TM-T13352
1mg99.00€5mg188.00€1mL*10mM (DMSO)250.00€10mg273.00€25mg427.00€50mg575.00€100mg743.00€200mg990.00€ROS 234
CAS:ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.Formula:C13H15N5Color and Shape:SolidMolecular weight:241.29
