Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
INCB38579
CAS:INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.Formula:C25H34N6OColor and Shape:SolidMolecular weight:434.58GSK 189254 HCl
CAS:GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.Formula:C21H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:387.9Nebidrazine
CAS:Nebidrazine is an alpha-adrenoceptor agonist.Formula:C9H8Cl2N6Color and Shape:SolidMolecular weight:271.11Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54Loratadine N-oxide
CAS:Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.Formula:C22H23ClN2O3Color and Shape:SolidMolecular weight:398.88MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Formula:C23H28Cl2F2N2O3Purity:98%Color and Shape:SolidMolecular weight:489.38Thioperamide
CAS:histamine H3 and H4 antagonist/inverse agonistFormula:C15H24N4SPurity:98%Color and Shape:White SolidMolecular weight:292.44VUF 5681 dihydrobromide
CAS:histamine H3 receptor silent antagonistFormula:C11H21Br2N3Purity:98%Color and Shape:SolidMolecular weight:355.11VUF 8430
CAS:VUF 8430 is a selective agonist for the H4 receptor.Formula:C4H11N5SPurity:98%Color and Shape:SolidMolecular weight:161.23UK-9040
CAS:UK-9040 inhibits gastric secretory.Formula:C23H31NSPurity:98%Color and Shape:SolidMolecular weight:353.56(R)-(-)-α-Methylhistamine dihydrobromide
CAS:(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).Formula:C6H13Br2N3Purity:99.98%Color and Shape:SolidMolecular weight:287Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Formula:C16H19ClN2OPurity:98%Color and Shape:LiquidMolecular weight:290.79PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.Formula:C19H26F2N2O3Purity:99.44%Color and Shape:SoildMolecular weight:368.42Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Formula:C8H14N4OPurity:98%Color and Shape:SolidMolecular weight:182.22JNJ-28610244
CAS:JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.Formula:C16H21N3OPurity:98%Color and Shape:SolidMolecular weight:271.36Setastine
CAS:Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.Formula:C22H28ClNOColor and Shape:SolidMolecular weight:357.92Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Formula:C13H19N3OSPurity:98.26%Color and Shape:SolidMolecular weight:265.37H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Formula:C20H27N3O2Purity:99.11%Color and Shape:SolidMolecular weight:341.45
