Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
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Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFormula:C31H37N5O3Purity:96.68%Color and Shape:SolidMolecular weight:527.66CP-66948
CAS:CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.Formula:C13H20N6SPurity:99.14%Color and Shape:SolidMolecular weight:292.4PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Formula:C20H28F2N2OPurity:>99.99%Color and Shape:SolidMolecular weight:350.45Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Formula:C19H29N5O2Purity:98.30% - 98.36%Color and Shape:SolidMolecular weight:359.47H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Formula:C19H24ClN3O3Purity:98%Color and Shape:SolidMolecular weight:377.86Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Formula:C20H25ClN2OSColor and Shape:SolidMolecular weight:376.94Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Formula:C17H22Cl2N4OPurity:98.28% - 99.30%Color and Shape:SolidMolecular weight:369.29JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Formula:C17H19ClN4O5Purity:99.37%Color and Shape:SolidMolecular weight:394.81Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Formula:C20H22N2Purity:98%Color and Shape:SolidMolecular weight:290.4Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurity:98%Color and Shape:SolidMolecular weight:321.44VUF14862
CAS:VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C26H32N4O2Color and Shape:SolidMolecular weight:432.56Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColor and Shape:SolidMolecular weight:342.46Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22BL 6341A
CAS:BL 6341A is related to Tumor data and H2-antagonists or anti-histaminsFormula:C9H14N8OS3Color and Shape:SolidMolecular weight:346.46(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Formula:C19H22N2OSColor and Shape:SolidMolecular weight:326.46Noberastine maleate
CAS:Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.Formula:C25H29N5O9Color and Shape:SolidMolecular weight:543.53ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Formula:C17H19N5O8Purity:98%Color and Shape:SolidMolecular weight:421.37Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Formula:C15H15D5N2O2Color and Shape:SolidMolecular weight:265.36
