Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 358 products of "Histamine Receptor"
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FR-A 19
CAS:<p>FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.</p>Formula:C25H34Cl3F2N5Color and Shape:SolidMolecular weight:548.93VUF 8328
CAS:<p>VUF 8328 is an agonist of histamine H(3) receptor.</p>Formula:C7H12N4SPurity:98%Color and Shape:SolidMolecular weight:184.26Adriforant
CAS:<p>Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.</p>Formula:C13H22N6Purity:99.84%Color and Shape:SolidMolecular weight:262.35FRG8701
CAS:<p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.55ReN-1869 hydrochloride
CAS:<p>ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.</p>Formula:C24H28ClNO2Purity:98%Color and Shape:SolidMolecular weight:397.94H4R antagonist 1
CAS:<p>H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.</p>Formula:C11H11BrN8Color and Shape:SolidMolecular weight:335.16(±)-Tazifylline
CAS:<p>(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.</p>Formula:C23H32N6O3SPurity:99.54%Color and Shape:SolidMolecular weight:472.6Noberastine
CAS:<p>Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.</p>Formula:C17H21N5OPurity:99.72% - >99.99%Color and Shape:SolidMolecular weight:311.38KSK68
CAS:<p>KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.</p>Formula:C23H28N2O2Purity:99.11%Color and Shape:SolidMolecular weight:364.48Immethridine dihydrobromide
CAS:<p>Immethridine dihydrobromide is a histamine H3 receptor agonist.</p>Formula:C9H11Br2N3Purity:97.61% - 98.14%Color and Shape:SolidMolecular weight:321.01D18024
CAS:<p>D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.</p>Formula:C29H31ClFN3OPurity:99.86%Color and Shape:SolidMolecular weight:492.03Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Formula:C14H26Cl3N7SPurity:99.82%Color and Shape:SolidMolecular weight:430.83Enerisant hydrochloride
CAS:<p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>Formula:C22H31ClN4O3Purity:99.95%Color and Shape:SolidMolecular weight:434.96Linetastine
CAS:<p>Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.</p>Formula:C35H40N2O6Purity:99.76%Color and Shape:SolidMolecular weight:584.7Pitolisant
CAS:<p>Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Formula:C17H26ClNOPurity:99.84%Color and Shape:SolidMolecular weight:295.85KSK94
CAS:<p>KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.</p>Formula:C25H26N4OPurity:99.60%Color and Shape:SolidMolecular weight:398.5Irdabisant
CAS:<p>Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.</p>Formula:C18H23N3O2Purity:99.96%Color and Shape:SolidMolecular weight:313.39Efletirizine
CAS:<p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>Formula:C21H24F2N2O3Purity:99.39%Color and Shape:SolidMolecular weight:390.42Antihistamine-1
CAS:<p>Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。</p>Formula:C23H24FN5Purity:99.69%Color and Shape:SolidMolecular weight:389.47NP10679
CAS:<p>NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.</p>Formula:C23H26F3N3O3Purity:99.43%Color and Shape:SolidMolecular weight:449.47
