Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 358 products of "Histamine Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Proxyfan
CAS:<p>Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.</p>Formula:C13H16N2OPurity:99.68%Color and Shape:SolidMolecular weight:216.28ReN-1869
CAS:<p>ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseases</p>Formula:C24H27NO2Purity:99.83% - 99.98%Color and Shape:SolidMolecular weight:361.48DF-1111301
CAS:<p>DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.</p>Formula:C15H25Cl2N3OPurity:99.17%Color and Shape:SolidMolecular weight:334.29Eclazolast
CAS:<p>Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.</p>Formula:C12H12ClNO4Purity:98.36% - 98.58%Color and Shape:SolidMolecular weight:269.68KP136
CAS:<p>KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).</p>Formula:C16H18N4O3Purity:98.3% - 98.61%Color and Shape:SolidMolecular weight:314.34Bavisant
CAS:<p>Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.</p>Formula:C19H27N3O2Purity:99.21% - 99.65%Color and Shape:SolidMolecular weight:329.44Abt-288
CAS:<p>ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.</p>Formula:C23H24N4OPurity:98.17% - 98.49%Color and Shape:SolidMolecular weight:372.46Clemastine
CAS:<p>Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.</p>Formula:C21H26ClNOPurity:99.21%Color and Shape:SolidMolecular weight:343.89JZP-361
CAS:<p>JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.</p>Formula:C22H20ClN5OPurity:99.82%Color and Shape:SolidMolecular weight:405.88JNJ-28583867
CAS:<p>JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake.</p>Formula:C24H32N2O2SColor and Shape:SolidMolecular weight:412.59Cipralisant maleate
CAS:<p>Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.</p>Formula:C18H24N2O4Color and Shape:SolidMolecular weight:332.39CI-949
CAS:<p>CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).</p>Formula:C20H20N6O3Purity:98%Color and Shape:SolidMolecular weight:392.41Ebrotidine
CAS:<p>Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection.</p>Formula:C14H17BrN6O2S3Purity:97.519%Color and Shape:SolidMolecular weight:477.42GSK-1004723
CAS:<p>GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.</p>Formula:C39H49ClN4O2Color and Shape:SolidMolecular weight:641.28Quinotolast sodium
CAS:<p>Quinotolast sodium inhibits histamine, LTC4 and PGD2 release in a concentration-dependent manner in the concentration range of 1-100 μg/mL.</p>Formula:C17H12N6NaO3Purity:98%Color and Shape:SolidMolecular weight:371.312UCB-35440
CAS:<p>UCB-35440, a 5-lipoxygenase inhibitor and a histamine H1 receptor antagonist, is used potentially for the treatment of dermatitis.</p>Formula:C31H34ClN5O4Color and Shape:SolidMolecular weight:576.09Minocromil
CAS:<p>Minocromil is a new agent of Anti-asthmatic.</p>Formula:C18H16N2O6Purity:98%Color and Shape:SolidMolecular weight:356.33A-349821
CAS:<p>A-349821 is an H3 receptor agonist radioligand.</p>Formula:C28H35F3N2O5Color and Shape:SolidMolecular weight:536.59GT-2331
CAS:<p>GT-2331 is a histamine H3 receptor antagonist.</p>Formula:C14H20N2Color and Shape:SolidMolecular weight:216.32Levocabastine
CAS:<p>Levocarbastine: 2nd-gen H1 antagonist, treats allergic conjunctivitis, selective NTS2 neurotensin inhibitor.</p>Formula:C26H29FN2O2Color and Shape:SolidMolecular weight:420.52
