Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
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GSK-239512
CAS:GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Formula:C23H27N3O2Purity:99.62% - 99.74%Color and Shape:SolidMolecular weight:377.48S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFormula:C6H11NO2SPurity:98%Color and Shape:SolidMolecular weight:161.22Dacemazine
CAS:Dacemazine is used to treat depression.Formula:C16H16N2OSColor and Shape:SolidMolecular weight:284.38VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C25H32N4O2Color and Shape:SolidMolecular weight:420.55Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Formula:C19H17NO7Purity:95% - 97.34%Color and Shape:SolidMolecular weight:371.34Dothiepin HCl
CAS:Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.Formula:C19H22ClNSColor and Shape:SolidMolecular weight:331.9FR-A 19
CAS:FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.Formula:C25H34Cl3F2N5Color and Shape:SolidMolecular weight:548.93KY 234
CAS:KY 234 is a thromboxane synthetase antagonist.Formula:C33H35N5O2Color and Shape:SolidMolecular weight:533.676(S)-Azelastine
CAS:(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9VUF 8328
CAS:VUF 8328 is an agonist of histamine H(3) receptor.Formula:C7H12N4SPurity:98%Color and Shape:SolidMolecular weight:184.26ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormula:C24H27NO2Purity:99.83% - 99.98%Color and Shape:SolidMolecular weight:361.48Immethridine dihydrobromide
CAS:Immethridine dihydrobromide is a histamine H3 receptor agonist.Formula:C9H11Br2N3Purity:97.61% - 98.14%Color and Shape:SolidMolecular weight:321.01Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formula:C13H16N2OPurity:99.68%Color and Shape:SolidMolecular weight:216.28DF-1111301
CAS:DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.Formula:C15H25Cl2N3OPurity:99.17%Color and Shape:SolidMolecular weight:334.29Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Formula:C17H21N5OPurity:99.72% - >99.99%Color and Shape:SolidMolecular weight:311.38KP136
CAS:KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Formula:C16H18N4O3Purity:98.3% - 98.61%Color and Shape:SolidMolecular weight:314.34JZP-361
CAS:JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.Formula:C22H20ClN5OPurity:99.82%Color and Shape:SolidMolecular weight:405.88Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C17H26ClNOPurity:99.84%Color and Shape:SolidMolecular weight:295.85Ref: TM-T60636
5mg46.00€1mL*10mM (DMSO)49.00€10mg66.00€25mg114.00€50mg178.00€100mg295.00€500mg708.00€KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formula:C25H26N4OPurity:99.60%Color and Shape:SolidMolecular weight:398.5Impromidine hydrochloride
CAS:Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.Formula:C14H26Cl3N7SPurity:99.82%Color and Shape:SolidMolecular weight:430.83
