Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 385 products of "Histamine Receptor"
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NP10679
CAS:NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Formula:C23H26F3N3O3Purity:99.43%Color and Shape:SolidMolecular weight:449.47Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formula:C21H26ClNOPurity:99.21%Color and Shape:SolidMolecular weight:343.89Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purity:99.21% - 99.65%Color and Shape:SolidMolecular weight:329.44Ref: TM-TQ0046
500mgTo inquire1mg43.00€1mL*10mM (DMSO)94.00€5mg96.00€10mg134.00€25mg221.00€50mg325.00€100mg465.00€Linetastine
CAS:Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formula:C35H40N2O6Purity:99.99%Color and Shape:SolidMolecular weight:584.7D18024
CAS:D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.Formula:C29H31ClFN3OPurity:99.86%Color and Shape:SolidMolecular weight:492.03Ref: TM-T10945
1mg349.00€5mg697.00€1mL*10mM (DMSO)880.00€10mg888.00€25mg1,395.00€50mg1,783.00€100mg2,530.00€Enerisant hydrochloride
CAS:Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteinsFormula:C22H31ClN4O3Purity:99.95%Color and Shape:SolidMolecular weight:434.96Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Formula:C23H24N4OPurity:98.17% - 98.49%Color and Shape:SolidMolecular weight:372.46KSK68
CAS:KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formula:C23H28N2O2Purity:99.11%Color and Shape:SolidMolecular weight:364.48Efletirizine
CAS:Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.Formula:C21H24F2N2O3Purity:99.39%Color and Shape:SolidMolecular weight:390.42Antihistamine-1
CAS:Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。Formula:C23H24FN5Purity:99.69%Color and Shape:SolidMolecular weight:389.47Eclazolast
CAS:Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.Formula:C12H12ClNO4Purity:98.29% - 98.61%Color and Shape:SolidMolecular weight:269.68Ref: TM-T25360
1mg112.00€1mL*10mM (DMSO)249.00€5mg261.00€10mg396.00€25mg655.00€50mg888.00€100mg1,251.00€500mg2,493.00€Irdabisant
CAS:Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.Formula:C18H23N3O2Purity:99.96%Color and Shape:SolidMolecular weight:313.39UCB-35440
CAS:UCB-35440, a 5-lipoxygenase inhibitor and a histamine H1 receptor antagonist, is used potentially for the treatment of dermatitis.Formula:C31H34ClN5O4Color and Shape:SolidMolecular weight:576.09Meclizine N-oxide
CAS:Meclizine N-oxide, a metabolite of the histamine H1 receptor antagonist meclizine (1), also acts as a degradation product and potential impurity in commercial meclizine preparations (2).Formula:C25H27ClN2OColor and Shape:SolidMolecular weight:407Levocabastine hydrochloride
CAS:Levocabastine HCl is an agent with antihistaminic activity.Formula:C26H30ClFN2O2Color and Shape:SolidMolecular weight:456.98Quinotolast sodium
CAS:Quinotolast sodium inhibits histamine, LTC4 and PGD2 release in a concentration-dependent manner in the concentration range of 1-100 μg/mL.Formula:C17H12N6NaO3Purity:98%Color and Shape:SolidMolecular weight:371.312A-349821
CAS:A-349821 is an H3 receptor agonist radioligand.Formula:C28H35F3N2O5Color and Shape:SolidMolecular weight:536.59CI-949
CAS:CI-949 inhibits LTC4/D4, histamine, TXB2 release (IC50: 0.5, 11.4, 0.1 μM).Formula:C20H20N6O3Purity:98%Color and Shape:SolidMolecular weight:392.41Ebrotidine
CAS:Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection.Formula:C14H17BrN6O2S3Purity:97.519%Color and Shape:SolidMolecular weight:477.42Minocromil
CAS:Minocromil is a new agent of Anti-asthmatic.Formula:C18H16N2O6Purity:98%Color and Shape:SolidMolecular weight:356.33
