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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 296 products of "Opioid Receptor"

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  • β-Naltrexamine dihydrochloride
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    β-Naltrexamine dihydrochloride

    CAS:
    <p>β-Naltrexamine dihydrochloride is an orally administered, irreversible opioid receptor antagonist. Its derivatives exhibit optimised subtype selectivity and can be used for pain research.</p>
    Formula:C20H28Cl2N2O3
    Purity:95.98%
    Color and Shape:Soild
    Molecular weight:415.35

    Ref: TM-T204075L

  • Biphalin TFA
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    Biphalin TFA

    CAS:
    <p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>
    Formula:C46H56N10O10·xC2HF3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:909.00 (free base)

    Ref: TM-T80074

  • CTOP
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    CTOP

    CAS:
    <p>Potent μ-receptor antagonist, Ki=0.96nM, ineffective at δ (&gt;10,000nM). Alters behavior in vivo, boosts K+ currents in rat neurons in vitro, μ-independent.</p>
    Formula:C50H67N11O11S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1062.28

    Ref: TM-TP2052

  • Cebranopadol hemicitrate
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    Cebranopadol hemicitrate

    CAS:
    <p>Cebranopadol hemicitrate is a NOP and opioid receptor agonist that targets human NOP, MOP, KOP, and δ-opioid peptide (DOP) receptors, with Ki/EC50 values of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, and 18 nM/110 nM, respectively. It is used in studies of acute and chronic pain.</p>
    Color and Shape:Solid

    Ref: TM-T206647

  • [DPro10] Dynorphin A (1-11)acetate,porcine
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    [DPro10] Dynorphin A (1-11)acetate,porcine

    <p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>
    Formula:C65H107N21O15
    Purity:99.05%
    Color and Shape:Soild
    Molecular weight:1422.7

    Ref: TM-T76341L

  • Nociceptin (1-13), amide
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    Nociceptin (1-13), amide

    CAS:
    <p>Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain</p>
    Formula:C61H100N22O15
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1381.59

    Ref: TM-TP1793

  • Ro 64-6198
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    Ro 64-6198

    CAS:
    <p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP&gt;opioid affinity.</p>
    Formula:C26H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.54

    Ref: TM-T16772

  • [Arg14,Lys15]Nociceptin
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    [Arg14,Lys15]Nociceptin

    CAS:
    <p>Potent NOP agonist (EC50 = 1 nM), &gt;875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.</p>
    Formula:C82H137N31O22
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1909.18

    Ref: TM-TP1986

  • N-Desmethyl Loperamide
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    N-Desmethyl Loperamide

    CAS:
    <p>N-Desmethyl Loperamide is the major metabolite of loperamide. It is also used as the precusor for radiolabelled loperamide.</p>
    Formula:C28H31ClN2O2
    Color and Shape:Solid
    Molecular weight:463.01

    Ref: TM-T33615

  • MT-7716 free base
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    MT-7716 free base

    CAS:
    <p>MT-7716: selective NOP agonist, potential in preventing alcohol abuse/relapse.</p>
    Formula:C27H28N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.54

    Ref: TM-T12120L

  • Neurotransmitter Receptor Compound Library
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    Neurotransmitter Receptor Compound Library

    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>
    Color and Shape:Odour Solid

    Ref: TM-L2610

  • BAM-22P
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    BAM-22P

    CAS:
    <p>Bovine adrenal medulla docosapeptide (BAM-22P) is a potent opioid agonist, derived from the proenkephalin A gene, which is present in the adrenal medulla.</p>
    Formula:C130H184N38O31S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2839.22

    Ref: TM-TP1211

  • TAN67
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    TAN67

    CAS:
    <p>TAN67 is the first effective selective non-peptide delta1 opioid receptor.</p>
    Formula:C23H26Br2N2O
    Color and Shape:Solid
    Molecular weight:506.282

    Ref: TM-T34784

  • Boc-ypgflt(O-tbu)
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    Boc-ypgflt(O-tbu)

    CAS:
    <p>Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.</p>
    Formula:C44H64N6O11
    Color and Shape:Solid
    Molecular weight:853.01

    Ref: TM-T25168

  • UFP-101
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    UFP-101

    CAS:
    <p>Strong, selective NOP receptor antagonist with pKi=10.24; &gt;3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.</p>
    Formula:C82H138N32O21
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1908.19

    Ref: TM-TP2105

  • CymitQuimica logo
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    N-terminally acetylated Endomorphin-1

    <p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>
    Formula:C36H40N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:652.74

    Ref: TM-TP1251

  • (Rac)-SNC80
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    (Rac)-SNC80

    CAS:
    <p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>
    Formula:C28H39N3O2
    Color and Shape:Solid
    Molecular weight:449.63

    Ref: TM-T73631

  • DAMGO (TFA)
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    DAMGO (TFA)

    CAS:
    <p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>
    Formula:C28H36F3N5O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:627.61

    Ref: TM-TP1607

  • Deltorphin acetate
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    Deltorphin acetate

    <p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>
    Formula:C46H66N10O12S2
    Purity:98.93%
    Color and Shape:Solid
    Molecular weight:1015.21

    Ref: TM-T20166L

  • N-Phenethylnoroxymorphone
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    N-Phenethylnoroxymorphone

    CAS:
    <p>N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.</p>
    Formula:C24H25NO4
    Color and Shape:Solid
    Molecular weight:391.46

    Ref: TM-T203674