Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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Endomorphin 2 TFA
CAS:Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.Formula:C34H38F3N5O7Color and Shape:SolidMolecular weight:685.69BMS-986121
CAS:BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.Formula:C15H9Cl2N3O2SPurity:99.67%Color and Shape:SolidMolecular weight:366.22Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:768.86MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purity:99.89% - 99.91%Color and Shape:SolidMolecular weight:518.01Ref: TM-T2071
2mg33.00€5mg52.00€10mg82.00€25mg155.00€50mg241.00€100mg355.00€200mg507.00€1mL*10mM (DMSO)55.00€LY2940094 tartrate
CAS:LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.Formula:C26H29ClF2N4O8SColor and Shape:SolidMolecular weight:631.04LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Ref: TM-TQ0091
1mg50.00€2mg71.00€5mg110.00€10mg172.00€25mg281.00€50mgTo inquire1mL*10mM (DMSO)120.00€Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purity:99.75%Color and Shape:SolidMolecular weight:530.4Ref: TM-T9459
1mg93.00€2mg136.00€5mg178.00€10mg268.00€25mg482.00€50mg688.00€100mg964.00€1mL*10mM (DMSO)236.00€Naloxegol (NKTR-118)
CAS:Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].Formula:C34H53NO11Color and Shape:SolidMolecular weight:651.78b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Ref: TM-T21660L
5mg42.00€10mg57.00€25mg87.00€50mg131.00€100mg190.00€200mg285.00€1mL*10mM (DMSO)55.00€Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16Nalmefene hydrochloride
CAS:Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.Formula:C21H26ClNO3Purity:98% - 99.85%Color and Shape:SolidMolecular weight:375.89Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26EST73502 hydrochloride
CAS:EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.Formula:C19H27ClF2N2O2Color and Shape:SolidMolecular weight:388.88Sec-O-Glucosylhamaudol
CAS:Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.Formula:C21H26O10Purity:99.79%Color and Shape:SolidMolecular weight:438.43GR 89696 free base
CAS:GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.Formula:C19H25Cl2N3O3Color and Shape:SolidMolecular weight:414.33Naloxegol oxalate
CAS:Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.Formula:C36H55NO15Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:741.83Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purity:99.09%Color and Shape:SolidMolecular weight:470.6MCOPPB
CAS:MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.Formula:C26H40N4Color and Shape:SolidMolecular weight:408.62
