Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 297 products of "Opioid Receptor"
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AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Formula:C23H29ClN2OPurity:98.66%Color and Shape:SolidMolecular weight:384.94Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Formula:C32H37N5O5Purity:99.64%Color and Shape:SolidMolecular weight:571.67Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formula:C26H25N3O2·HClPurity:99.27% - 99.59%Color and Shape:SolidMolecular weight:447.96BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Formula:C132H188N38O33S2Purity:99.87%Color and Shape:SoildMolecular weight:2899.27BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78ADL-5859
CAS:<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Formula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Formula:C101H159N31O25Purity:99.69%Color and Shape:SolidMolecular weight:2207.58(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Formula:C33H46N6O10Purity:94.17%Color and Shape:SoildMolecular weight:686.75Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formula:C19H23NO4Purity:99.02% - 99.73%Color and Shape:White PowderMolecular weight:329.39Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Formula:C77H130N24O17Purity:99.14%Color and Shape:SolidMolecular weight:1664Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55Endomorphin 1
CAS:<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Formula:C34H38N6O5Purity:95.92%Color and Shape:Solid (Solid Powder )Molecular weight:610.7Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Formula:C76H119N21O19Purity:99.72%Color and Shape:SolidMolecular weight:1630.89ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formula:C24H29ClN2O3Color and Shape:SolidMolecular weight:428.95
