Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 296 products of "Opioid Receptor"
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Leumorphin, human
CAS:<p>Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-</p>Formula:C150H224N42O46Purity:98%Color and Shape:SolidMolecular weight:3351.64Deltorphin acetate
<p>Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid</p>Formula:C46H66N10O12S2Purity:98.93%Color and Shape:SolidMolecular weight:1015.21CJ-15208
CAS:<p>CJ-15208: κ-opioid antagonist, IC50: 47 nM kappa, 260 nM mu, 2600 nM delta, reverses asimadoline effects in rabbits (ED50 1.3 µM).</p>Formula:C34H35N5O4Color and Shape:SolidMolecular weight:577.67N-terminally acetylated Endomorphin-1
<p>N-terminally acetylated Endomorphin-1 is a modified Endomorphin-1.</p>Formula:C36H40N6O6Purity:98%Color and Shape:SolidMolecular weight:652.74Opioid receptor agonist 1
<p>Opioid receptor agonist1 (Compound 2638-28) is an orally active opioid receptor agonist that shows strong affinity for MOR, DOR, and KOR, with Ki values of 5, 24, and 212 nM, respectively. It exhibits analgesic activity in both the mouse warm water tail-flick model and the acetic acid writhing model.</p>Formula:C32H45N5OColor and Shape:SolidMolecular weight:515.73Neuropeptide AF (human) acetate
<p>Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,</p>Purity:99.89%Color and Shape:SoildCTOP acetate
<p>CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.</p>Formula:C52H71N11O13S2Purity:99.87%Color and Shape:SoildMolecular weight:1122.32UFP-101 acetate
<p>UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.</p>Formula:C84H142N32O23Purity:95.92%Color and Shape:SolidMolecular weight:1968.23difelikefalin acetate(1024828-77-0 Free base)
CAS:<p>is a ketone and a building block.</p>Formula:C38H57N7O8Purity:96.94%Color and Shape:SolidMolecular weight:739.9[(pF)Phe4]Nociceptin(1-13)NH2 acetate
<p>[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and a pEC50 of 9.31.</p>Formula:C63H103FN22O17Purity:98.03%Color and Shape:SolidMolecular weight:1459.63[D-Ala2]leucine-enkephalin acetate
<p>[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of</p>Formula:C31H43N5O9Purity:98%Color and Shape:SolidMolecular weight:629.65β-Endorphin (1-27) (human) acetate
<p>β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.</p>Formula:C141H221N33O42SPurity:96.52%Color and Shape:SolidMolecular weight:3082.52β-Endorphin (6-31), human
CAS:<p>β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors.</p>Formula:C131H218N34O40Purity:98%Color and Shape:SolidMolecular weight:2909.38Deltorphin
CAS:<p>Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity to the opioid receptor.</p>Formula:C44H62N10O10S2Purity:98.96%Color and Shape:SolidMolecular weight:955.15Loperamide phenyl
CAS:<p>Loperamide phenyl, an impurity detected in Loperamide, is an opioid receptor agonist.</p>Formula:C35H37ClN2O2Color and Shape:SolidMolecular weight:553.14BMS-986121
CAS:<p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>Formula:C15H9Cl2N3O2SPurity:99.67%Color and Shape:SolidMolecular weight:366.22[Leu5]-Enkephalin
CAS:<p>[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM</p>Formula:C28H37N5O7Purity:99.87% - 99.88%Color and Shape:SolidMolecular weight:555.62Porcine dynorphin A(1-13)
CAS:<p>Porcine dynorphin A (1-13) is a potent κ opioid receptor agonist; it's antinociceptive and raises [Ca2+]i in neurons like NMDA.</p>Formula:C75H126N24O15Purity:98%Color and Shape:SolidMolecular weight:1603.95Endomorphin 2 TFA
CAS:<p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>Formula:C34H38F3N5O7Color and Shape:SolidMolecular weight:685.69BAN ORL 24 dihydrochloride
CAS:<p>BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that can be used to study neurological diseases.</p>Formula:C27H37Cl2N3O2Purity:95.03%Color and Shape:SolidMolecular weight:506.51Alvimopan dihydrate (LY246736 dihydrate)
CAS:<p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>Formula:C25H36N2O6Color and Shape:SolidMolecular weight:460.56Asimadoline
CAS:<p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54GR103545
CAS:<p>GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.</p>Formula:C23H29Cl2N3O7Purity:99.75%Color and Shape:SolidMolecular weight:530.4Endomorphin 1
CAS:<p>Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).</p>Formula:C34H38N6O5Purity:95.92%Color and Shape:Solid (Solid Powder )Molecular weight:610.7DPDPE TFA (88373-73-3 free base)
CAS:<p>DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.</p>Formula:C32H40F3N5O9S2Purity:99.39%Color and Shape:SolidMolecular weight:759.81CTAP(TFA) (103429-32-9 free base)
<p>CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.</p>Formula:C53H70F3N13O13S2Purity:99.62%Color and Shape:SolidMolecular weight:1218.33Gluten Exorphin C
CAS:<p>Gluten exorphin C is an opioid peptide derived from wheat gluten.</p>Formula:C29H45N5O8Purity:99.39%Color and Shape:SolidMolecular weight:591.7ADL-5747 (HCl)
CAS:<p>ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.</p>Formula:C24H29ClN2O3Color and Shape:SolidMolecular weight:428.95PZM21
CAS:<p>PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).</p>Formula:C19H27N3O2SPurity:99.93% - >99.99%Color and Shape:SolidMolecular weight:361.5Asimadoline hydrochloride
CAS:<p>Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.</p>Formula:C27H31ClN2O2Purity:98.94% - 99.32%Color and Shape:SolidMolecular weight:451.01Hemorphin-7 acetate(152685-85-3 free base)
<p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16DAMGO
CAS:<p>DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.</p>Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59MCOPPB
CAS:<p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>Formula:C26H40N4Color and Shape:SolidMolecular weight:408.62Deltorphin 2
CAS:<p>Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.</p>Formula:C38H54N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:782.88DAMGO TFA (78123-71-4(Free base))
<p>DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.</p>Formula:C28H36F3N5O8Purity:98.67% - 99.76%Color and Shape:SolidMolecular weight:627.6BW-180C
CAS:<p>BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.</p>Formula:C29H39N5O7Purity:>99.99%Color and Shape:SolidMolecular weight:569.65N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8GR 89696 free base
CAS:<p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>Formula:C19H25Cl2N3O3Color and Shape:SolidMolecular weight:414.33Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Formula:C26H27FN2O2Purity:99.53% - 99.93%Color and Shape:SolidMolecular weight:418.5EST73502 hydrochloride
CAS:<p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>Formula:C19H27ClF2N2O2Color and Shape:SolidMolecular weight:388.88Leuphasyl TFA
CAS:<p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.</p>Formula:C31H40F3N5O9Purity:98.79%Color and Shape:SolidMolecular weight:683.67Nociceptin (1-13) amide TFA
<p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>Formula:C63H101F3N22O17Purity:97.64%Color and Shape:SolidMolecular weight:1495.61Ac-RYYRIK-NH2 acetate
<p>Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.</p>Formula:C46H74N14O11Purity:99.84%Color and Shape:SolidMolecular weight:999.17BMS986188
CAS:<p>BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.</p>Formula:C30H31BrO4Purity:98.76%Color and Shape:SolidMolecular weight:535.47Adrenorphin 3TFA(88377-68-8(free base))
<p>Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).</p>Formula:C50H72N15O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1326.26Corydaline
CAS:<p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>Formula:C22H27NO4Purity:98.97% - 99.86%Color and Shape:SolidMolecular weight:369.45Dynorphin A 1-10 acetate(79994-24-4 free base)
<p>Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.</p>Formula:C59H95N19O14Purity:99.88%Color and Shape:SolidMolecular weight:1294.53[D-Ala2]leucine-enkephalin
CAS:<p>[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.</p>Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65[Leu5]-Enkephalin, amide acetate
<p>[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.</p>Formula:C30H42N6O8Purity:99.36%Color and Shape:SolidMolecular weight:614.69Difelikefalin acetate
CAS:<p>Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.</p>Formula:C38H57N7O8Purity:99.55%Color and Shape:SolidMolecular weight:739.9
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