Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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Sinomenine
CAS:115-53-7
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the …
Formula:
C19H23NO4
Purity:
99.02% - 99.89%
Color and Shape:
White Powder
Molecular weight:
329.39
Ref: TM-T2726
| 100mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
PZM21
CAS:1997387-43-5
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
Formula:
C19H27N3O2S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
361.5
Ref: TM-T4386
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 468.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 80.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 861.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,341.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
BMS986187
CAS:684238-37-7
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
Formula:
C31H34O4
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
470.6
Ref: TM-T8991
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 503.00 € | ||
| 500mg | 1,068.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
GR103545
CAS:126766-43-6
GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can …
Formula:
C23H29Cl2N3O7
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T9459
| 1mg | 96.00 € | ||
| 2mg | 141.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 278.00 € | ||
| 25mg | 499.00 € | ||
| 50mg | 715.00 € | ||
| 100mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
LY2795050
CAS:1346133-08-1
LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).
Formula:
C23H22ClN3O2
Purity:
97.77%
Color and Shape:
Solid
Molecular weight:
407.89
Ref: TM-TQ0091
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 292.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
DAMGO
CAS:78123-71-4
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity …
Formula:
C26H35N5O6
Purity:
98.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
513.59
Ref: TM-T4351
| 1mg | 50.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 609.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
Spinorphin
CAS:137201-62-8
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
Formula:
C45H64N8O10
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
877
Ref: TM-T8455
| 1mg | 129.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 373.00 € | ||
| 25mg | 622.00 € | ||
| 50mg | 887.00 € | ||
| 100mg | 1,201.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C50H72N15O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1326.26
Ref: TM-T7567L
| 1mg | 47.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 450.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 836.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
![[D-Ala2]leucine-enkephalin](https://static.cymitquimica.com/products/TM/thumb/TP1367.jpg)
[D-Ala2]leucine-enkephalin
CAS:64963-01-5
[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta …
Formula:
C29H39N5O7
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1367
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 460.00 € | ||
| 200mg | 643.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
Endomorphin 1
CAS:189388-22-5
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays …
Formula:
C34H38N6O5
Purity:
95.92%
Color and Shape:
Solid (Solid Powder )
Molecular weight:
610.7
Ref: TM-TQ0267
| 5mg | 49.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 94.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
ADL-5747
CAS:850176-30-6
ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the …
Formula:
C24H28N2O3
Purity:
100% - 99.44%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T29663
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,971.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
ORL1 antagonist 1
CAS:1174985-59-1
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 …
Formula:
C20H22ClN5
Purity:
97.87%
Color and Shape:
Solid
Molecular weight:
367.88
Ref: TM-T12320
| 1mg | 78.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 478.00 € | ||
| 100mg | 642.00 € | ||
| 200mg | 850.00 € | ||
| 1mL*10mM (DMSO) | 164.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
Opioid receptor modulator 1
CAS:77514-44-4
Opioid receptor modulator 1 is a modulator of opioid receptor.
Formula:
C18H23NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T12314
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 707.00 € | ||
| 5mg | 1,486.00 € | ||
| 25mg | 1,976.00 € | ||
| 50mg | 2,412.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
GR 89696 fumarate
CAS:126766-32-3
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with …
Formula:
C23H29Cl2N3O7
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T22810
| 5mg | 63.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 328.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
NNC 63-0532
CAS:250685-44-0
NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.
Formula:
C27H29N3O3
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T23074
| 1mg | 49.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 626.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
SCH 221510
CAS:322473-89-2
SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.
Formula:
C28H31NO
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
397.55
Ref: TM-T23335
| 1mg | 77.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 834.00 € | ||
| 100mg | 1,355.00 € | ||
| 200mg | 1,822.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
SCH-486757
CAS:524019-25-8
SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used …
Formula:
C24H23Cl2N3O
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
440.37
Ref: TM-T28728
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Wednesday 2 Apr 2025
