Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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IPAG
CAS:193527-91-2
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
Formula:
C17H22IN3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
395.28
Ref: TM-T22870
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 454.00 € | ||
| 100mg | 655.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 723.00 € | ||
| 5mg | 1,510.00 € | ||
| 25mg | 2,023.00 € | ||
| 50mg | 2,452.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
Trimebutine CTB salt
CAS:1456509-46-8
Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.
Formula:
C29H36N2O8S2
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
604.74
Ref: TM-T27413
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,537.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
SCH-486757
CAS:524019-25-8
SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used …
Formula:
C24H23Cl2N3O
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
440.37
Ref: TM-T28728
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
GSK1521498 free base
CAS:1007573-18-3
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor.
Formula:
C24H20F2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T11478L
| 25mg | 1,206.00 € | ||
| 50mg | 1,568.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
ADL-5747
CAS:850176-30-6
ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the …
Formula:
C24H28N2O3
Purity:
100% - 99.44%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T29663
| 1mg | 140.00 € | ||
| 5mg | 343.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
ICI 204,448
CAS:121264-04-8
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of …
Formula:
C23H27Cl3N2O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
501.83
Ref: TM-T22850
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 620.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
Opioid receptor modulator 1
CAS:77514-44-4
Opioid receptor modulator 1 is a modulator of opioid receptor.
Formula:
C18H23NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T12314
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
GSK1521498
CAS:1426543-84-1
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H23F2N4O4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.43
Ref: TM-T11479
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
Bevenopran
CAS:676500-67-7
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies …
Formula:
C20H26N4O4
Purity:
98.14% - 98.76%
Color and Shape:
Solid
Molecular weight:
386.44
Ref: TM-T14551
| 1mg | 65.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 316.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 562.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Wednesday 4 Jun 2025
MOR agonist-1
CAS:2305781-14-8
MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and …
Formula:
C22H26ClFN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
404.91
Ref: TM-T79060
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 18 Jun 2025
Icalcaprant
CAS:2227384-17-8
Icalcaprant is a kappa-opioid receptor antagonist [1].
Formula:
C23H26N4O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
406.48
Ref: TM-T79848
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 18 Jun 2025
DPI-3290
CAS:182417-73-8
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 …
Formula:
C30H34FN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
487.61
Ref: TM-T15165
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Wednesday 18 Jun 2025
μ opioid receptor agonist 3
CAS:2378397-91-0
Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that …
Formula:
C22H28N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
352.47
Ref: TM-T79430
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 18 Jun 2025
Mu opioid receptor antagonist 7
CAS:2378397-30-7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid …
Formula:
C22H27ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.91
Ref: TM-T79431
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Wednesday 18 Jun 2025
Isotodesnitazene
CAS:2732926-27-9
Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 …
Formula:
C23H31N3O
Color and Shape:
Liquid
Molecular weight:
365.51
Ref: TM-T201840
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 16 Jul 2025
Nalmefene
CAS:55096-26-9
Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study …
Formula:
C21H25NO3
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
339.43
Ref: TM-T86954
| 2mg | 38.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 87.00 € |
Estimated delivery in United States, on Wednesday 16 Jul 2025
22-Thiocyanatosalvinorin A
CAS:1174223-49-4
22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 …
Formula:
C24H27NO8S
Color and Shape:
Liquid
Molecular weight:
489.54
Ref: TM-T201845
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 16 Jul 2025
Norbinaltorphimine dihydrochloride
CAS:113158-34-2
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses …
Formula:
C40H45Cl2N3O6
Purity:
99%
Color and Shape:
Solid
Molecular weight:
734.71
Ref: TM-T12241
| 1mg | 40.00 € | ||
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 16 Jul 2025
