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Glucagon Receptor

Glucagon Receptor

Glucagon receptors are GPCRs that mediate the effects of glucagon, a hormone involved in regulating glucose homeostasis by promoting glycogen breakdown and glucose release from the liver. These receptors are critical in the management of blood sugar levels and are of particular interest in the study of diabetes and metabolic disorders. Glucagon receptor antagonists are being explored as potential treatments for hyperglycemia in type 2 diabetes. At CymitQuimica, we offer a variety of high-quality glucagon receptor modulators to support your research in endocrinology, diabetes, and metabolic regulation.

Found 164 products of "Glucagon Receptor"

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  • GLP-1R agonist 3
    Targetmol
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    GLP-1R agonist 3

    CAS:
    <p>GLP-1R agonist 3 is a GLP-1R agonist, an imidazole derivative.GLP-1R agonist 3 can be used to study diabetes and obesity.</p>
    Formula:C31H28FN5O4
    Purity:97.19%
    Color and Shape:Solid
    Molecular weight:553.58

    Ref: TM-T63909

  • GLP-1R agonist 10
    Targetmol
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    GLP-1R agonist 10

    CAS:
    <p>GLP-1R agonist 10 is a GLP-1 agonist (EC50: 0.051 nM).</p>
    Formula:C29H29ClFN5O4
    Color and Shape:Solid
    Molecular weight:566.02

    Ref: TM-T64007

  • LGD-6972
    Targetmol
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    LGD-6972

    CAS:
    <p>LGD-6972 is an antagonist of glucagon receptor.</p>
    Formula:C43H46N2O5S
    Purity:98.8% - 99.62%
    Color and Shape:Solid
    Molecular weight:702.9

    Ref: TM-T11845

  • Lotiglipron
    Targetmol
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    Lotiglipron

    CAS:
    <p>Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.</p>
    Formula:C31H31ClN4O5
    Purity:98.3%
    Color and Shape:Solid
    Molecular weight:575.05

    Ref: TM-T77781

  • Adomeglivant
    Targetmol
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    Adomeglivant

    CAS:
    <p>Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.</p>
    Formula:C32H36F3NO4
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:555.63

    Ref: TM-T14130

  • PF-06372222
    Targetmol
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    PF-06372222

    CAS:
    <p>PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.</p>
    Formula:C26H28F3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.53

    Ref: TM-T24620

  • GLP-1 receptor agonist 11
    Targetmol
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    GLP-1 receptor agonist 11

    CAS:
    <p>GLP-1 Receptor Agonist 11 (compound 3) acts as an effective agonist for the GLP Receptor, finding use in research related to conditions like diabetes and non-alc. fatty liver disease [1].</p>
    Formula:C31H31ClFN3O4
    Color and Shape:Solid
    Molecular weight:564.05

    Ref: TM-T86503

  • GLP-1 receptor agonist 16
    Targetmol
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    GLP-1 receptor agonist 16

    CAS:
    <p>GLP-1 receptoragonist 16 (Example 53) is a GLP-1 agonist applicable for research in diabetes, obesity, or diseases related to non-alcoholic steatohepatitis.</p>
    Formula:C33H31ClFN3O4
    Color and Shape:Solid
    Molecular weight:588.068

    Ref: TM-T204526

  • GLP-1 receptor agonist 15
    Targetmol
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    GLP-1 receptor agonist 15

    CAS:
    <p>GLP-1 receptor agonist 15 (Example 4) is a GLP receptor agonist with an EC50 of 0.74 nM. It exhibits an IC50 of 10.1 μM against the hERG potassium ion channel. This compound is applicable for research in the diabetes field.</p>
    Formula:C32H31ClFN3O5
    Color and Shape:Solid
    Molecular weight:592.057

    Ref: TM-T204742

  • SCH-900822
    Targetmol
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    SCH-900822

    CAS:
    <p>SCH-900822 is a potent and selective glucagon receptor antagonist.</p>
    Formula:C34H43Cl2N7O2
    Color and Shape:Solid
    Molecular weight:652.66

    Ref: TM-T71201

  • GLP-1R agonist 8
    Targetmol
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    GLP-1R agonist 8

    CAS:
    <p>GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 &lt; 2 nM).</p>
    Formula:C33H32N4O5
    Color and Shape:Solid
    Molecular weight:564.63

    Ref: TM-T63999

  • DS79932728
    Targetmol
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    DS79932728

    CAS:
    <p>DS79932728 is an orally active inhibitor of G9a and GLP, with IC50 values of 12.6 nM and 75.7 nM, respectively. It induces the production of γ-globin, thereby increasing fetal hemoglobin (HbF) levels. In cynomolgus monkey models, DS79932728 enhances the proportion of F-reticulocytes (F-rets) and shows good oral absorption characteristics.</p>
    Formula:C19H25N3O
    Color and Shape:Solid
    Molecular weight:311.421

    Ref: TM-T205011

  • DA-302168S
    Targetmol
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    DA-302168S

    CAS:
    <p>DA-302168S is an orally active, selective GLP-1R agonist with an EC50 value of 1.32 nM. It promotes insulin secretion and has a hypoglycemic effect. Additionally, DA-302168S reduces food intake. It primarily activates GLP-1R in humans and monkeys, with minimal effect on GLP-1R in rats, mice, and dogs. DA-302168S can be used for research in type 2 diabetes and obesity.</p>
    Formula:C33H24ClF2N3O5
    Color and Shape:Solid
    Molecular weight:616.011

    Ref: TM-T206917

  • LSN3318839
    Targetmol
    + Info

    LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:480.39

    Ref: TM-T63166