Cholecystokinin
Cholecystokinin (CCK) receptors are a class of G protein-coupled receptors (GPCRs) that bind to the peptide hormone cholecystokinin. These receptors are involved in digestive processes, such as stimulating the release of digestive enzymes from the pancreas and bile from the gallbladder, as well as in regulating appetite and satiety. Cholecystokinin receptor modulators are studied for their potential roles in treating gastrointestinal disorders, obesity, and anxiety. At CymitQuimica, we provide a range of high-quality cholecystokinin receptor modulators to support your research in digestive health, endocrinology, and neurobiology.
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Proglumide
CAS:6620-60-6
Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal …
Formula:
C18H26N2O4
Purity:
99.44%
Color and Shape:
White Crystalline Powder
Molecular weight:
334.41
Ref: TM-T1052
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
WAY-620645
CAS:742116-45-6
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
Formula:
C22H22N4O2
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
374.44
Ref: TM-T9991
| 1mg | 62.00 € | ||
| 5mg | 132.00 € | ||
| 10mg | 186.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 553.00 € | ||
| 100mg | 802.00 € | ||
| 500mg | 1,558.00 € | ||
| 1mL*10mM (DMSO) | 176.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GV-150013X
CAS:151386-96-8
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Soild
Molecular weight:
534.65
Ref: TM-T27503L
| 1mg | 183.00 € | ||
| 5mg | 444.00 € | ||
| 10mg | 608.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,235.00 € | ||
| 100mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 638.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 152.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 876.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,214.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Lintitript
CAS:136381-85-6
Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and …
Formula:
C20H14ClN3O3S
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
411.86
Ref: TM-T15759
| 1mg | 113.00 € | ||
| 2mg | 154.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 549.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 258.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Pranazepide
CAS:150408-73-4
Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders …
Formula:
C26H19FN4O2
Purity:
98.20% - 99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T34123
| 1mg | 513.00 € | ||
| 5mg | 1,129.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
N-Cbz-DL-tryptophan
CAS:13058-16-7
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
Formula:
C19H18N2O4
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
338.36
Ref: TM-T9343
| 5mg | 41.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 198.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 495.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PHA-767491
CAS:845714-00-3
PHA-767491 (CAY10572) is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and …
Formula:
C12H11N3O
Purity:
100.00% - 99.49%
Color and Shape:
Solid
Molecular weight:
213.24
Ref: TM-T6206
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 396.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Loxiglumide
CAS:107097-80-3
Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.
Formula:
C21H30Cl2N2O5
Purity:
98% - 99.81%
Color and Shape:
Solid
Molecular weight:
461.38
Ref: TM-T2312
| 10mg | 40.00 € | ||
| 25mg | 76.00 € | ||
| 50mg | 120.00 € | ||
| 100mg | 196.00 € | ||
| 200mg | 337.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Nastorazepide
CAS:209219-38-5
Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic …
Formula:
C29H36N4O5
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
520.62
Ref: TM-TQ0062
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 178.00 € | ||
| 25mg | 341.00 € | ||
| 50mg | 519.00 € | ||
| 100mg | 749.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
XL413
CAS:1169558-38-6
XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell …
Formula:
C14H12ClN3O2
Purity:
100% - 99.38%
Color and Shape:
Solid
Molecular weight:
289.72
Ref: TM-T3352
| 1mg | 52.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 643.00 € |
Estimated delivery in United States, on Wednesday 8 Jan 2025
A-65186
CAS:119295-94-2
A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.
Formula:
C25H35N3O4
Purity:
98.37% - 99.94%
Color and Shape:
Solid
Molecular weight:
441.56
Ref: TM-T26483
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CCK-A receptor inhibitor 1
CAS:137004-80-9
CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: …
Formula:
C25H35NO6S
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
477.61
Ref: TM-T12404
| 1mg | 654.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Lorglumide sodium salt
CAS:1021868-76-7
Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).
Formula:
C22H31Cl2N2NaO4
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
481.39
Ref: TM-T11868
| 5mg | 34.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
L-365260
CAS:118101-09-0
L-365260 is a nonpeptide gastrin and cerebral cholecystokinin receptor (CCK-B) antagonist used in the study …
Formula:
C24H22N4O2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
398.46
Ref: TM-T22895
| 2mg | 293.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Itriglumide
CAS:201605-51-8
Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, …
Formula:
C33H38N2O4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T27640
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 915.00 € | ||
| 25mg | 1,409.00 € | ||
| 50mg | 1,836.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
(Iso)-FK-480
CAS:167820-10-2
(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic …
Formula:
C26H19FN4O2
Purity:
98.92% - 99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T10055
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
XL413 hydrochloride
CAS:2062200-97-7
XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7. XL413 …
Formula:
C14H13Cl2N3O2
Purity:
98.81% - 99.82%
Color and Shape:
Solid
Molecular weight:
326.18
Ref: TM-T6735
| 1mg | 52.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 694.00 € | ||
| 200mg | 917.00 € | ||
| 500mg | 1,417.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
GV150013
CAS:167355-22-8
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
534.65
Ref: TM-T27503
| 1mg | 182.00 € | ||
| 5mg | 443.00 € | ||
| 10mg | 604.00 € | ||
| 25mg | 915.00 € | ||
| 50mg | 1,229.00 € | ||
| 100mg | 1,617.00 € | ||
| 200mg | 2,189.00 € | ||
| 1mL*10mM (DMSO) | 627.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
GI 181771
CAS:305366-98-7
GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used …
Formula:
C34H31N5O6
Purity:
95.63%
Color and Shape:
Solid
Molecular weight:
605.64
Ref: TM-T15382
| 1mg | 182.00 € | ||
| 5mg | 416.00 € | ||
| 50mg | 1,290.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
