LPA Receptor
Lysophosphatidic acid (LPA) receptors are a group of GPCRs that respond to LPA, a bioactive lipid involved in cell proliferation, migration, and survival. LPA signaling plays a crucial role in various physiological processes, including wound healing, vascular development, and cancer metastasis. Modulation of LPA receptor activity is being explored for therapeutic applications in cancer, fibrosis, and inflammatory diseases. At CymitQuimica, we offer a range of high-quality LPA receptor modulators to support your research in cell signaling, oncology, and inflammatory disorders.
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AM095 free acid
CAS:1228690-36-5
AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for …
Formula:
C27H24N2O5
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
456.49
Ref: TM-T10293
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 542.00 € | ||
| 200mg | 782.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
TAK-615
CAS:1664335-55-0
TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of …
Formula:
C25H22FNO4
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
419.44
Ref: TM-T9699
| 1mg | 75.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 420.00 € | ||
| 50mg | 592.00 € | ||
| 100mg | 799.00 € | ||
| 500mg | 1,591.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Edg-2 receptor inhibitor 1
CAS:1195941-38-8
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
Formula:
C27H27NO5
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T4521
| 1mg | 95.00 € | ||
| 2mg | 171.00 € | ||
| 5mg | 268.00 € | ||
| 10mg | 419.00 € | ||
| 25mg | 648.00 € | ||
| 50mg | 925.00 € | ||
| 100mg | 1,240.00 € | ||
| 1mL*10mM (DMSO) | 286.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Ki16198
CAS:355025-13-7
Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. …
Formula:
C24H25ClN2O5S
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
488.98
Ref: TM-T6347
| 5mg | 36.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 228.00 € | ||
| 200mg | 324.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
445.51
Ref: TM-T39647
| 1mg | 68.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 160.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
H2L 5765834
CAS:420841-84-5
H2L 5765834 is a lysophosphatidic acid receptors antagonist
Formula:
C21H12N2O7
Purity:
99.47% - ≥98%
Color and Shape:
Solid
Molecular weight:
404.33
Ref: TM-T22834
| 1mg | 60.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
AM095
CAS:1345614-59-6
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM …
Formula:
C27H23N2NaO5
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
478.47
Ref: TM-T2000
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 601.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
AM966
CAS:1228690-19-4
AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.
Formula:
C27H23ClN2O5
Purity:
97.32% - 99.49%
Color and Shape:
Solid
Molecular weight:
490.93
Ref: TM-T4278
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 159.00 € | ||
| 100mg | 246.00 € | ||
| 200mg | 354.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Ki16425
CAS:355025-24-0
Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 …
Formula:
C23H23ClN2O5S
Purity:
97.60% - 97.78%
Color and Shape:
Solid
Molecular weight:
474.96
Ref: TM-T6108
| 2mg | 41.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 189.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
BMS-986020
CAS:1257213-50-5
BMS-986020 (AM152) is a selective antagonist of LPA1.
Formula:
C29H26N2O5
Purity:
100% - 98.82%
Color and Shape:
Solid
Molecular weight:
482.53
Ref: TM-T4016
| 1mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
ONO-7300243
CAS:638132-34-0
ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).
Formula:
C28H31NO5
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
461.55
Ref: TM-T7393
| 1mg | 45.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 407.00 € | ||
| 100mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Tetradecyl Phosphonate
CAS:4671-75-4
Tetradecyl phosphonate is a pan-antagonist of lysophosphatidic acid 1 (LPA1), LPA2, and LPA3 receptors.
Formula:
C14H31O3P
Purity:
≥95%
Color and Shape:
White To Off-White Powder
Molecular weight:
278.37
Ref: TM-T7689
| 5mg | 55.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 409.00 € | ||
| 500mg | 662.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
1-Oleoyl lysophosphatidic acid sodium
CAS:325465-93-8
1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of …
Formula:
C21H40O7P·Na
Purity:
98.75% - 99.24%
Color and Shape:
Liquid
Molecular weight:
458.51
Ref: TM-T21654
| 1mg | 69.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 503.00 € | ||
| 100mg | 715.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
UCM-05194
CAS:2411412-36-5
UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD …
Formula:
C19H30BrO6P
Purity:
90% - 91.22%
Color and Shape:
Liquid
Molecular weight:
465.32
Ref: TM-T69647
| 1mg | 315.00 € | ||
| 5mg | 746.00 € | ||
| 10mg | 1,057.00 € | ||
| 25mg | 1,576.00 € | ||
| 50mg | 2,057.00 € | ||
| 100mg | 2,732.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
LPA2 antagonist 2
CAS:36840-10-5
LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, …
Formula:
C20H16N2O6
Purity:
96.13%
Color and Shape:
Solid
Molecular weight:
380.35
Ref: TM-T11875
| 1mg | 93.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 350.00 € | ||
| 25mg | 576.00 € | ||
| 50mg | 812.00 € | ||
| 100mg | 1,094.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
TC LPA5 4
CAS:1393814-38-4
TC LPA5 4 is a LPA5 receptor antagonist.
Formula:
C23H23ClN2O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T23438
| 1mg | 58.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 891.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
GRI977143
CAS:325850-81-5
GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.
Formula:
C22H17NO4S
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
391.44
Ref: TM-T22812
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,333.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
H2L5186303
CAS:139262-76-3
H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.
Formula:
C26H20N2O8
Purity:
97.23%
Color and Shape:
Solid
Molecular weight:
488.45
Ref: TM-T22835
| 1mg | 35.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 917.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
Radioprotectin-1
CAS:1622006-09-0
Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 …
Formula:
C23H19ClN2O6S
Purity:
98.75% - 99.43%
Color and Shape:
Solid
Molecular weight:
486.92
Ref: TM-T12684
| 1mg | 79.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 414.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 754.00 € | ||
| 1mL*10mM (DMSO) | 182.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
DBIBB
CAS:1569309-92-7
DBIBB: non-lipid LPA2 receptor agonist, treats acute radiation syndrome, aids in organic synthesis/drug research.
Formula:
C23H20N2O6S
Purity:
97.18% - 97.26%
Color and Shape:
Solid
Molecular weight:
452.48
Ref: TM-T22070
| 1mg | 41.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 543.00 € | ||
| 500mg | 1,089.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
