LPA Receptor
Lysophosphatidic acid (LPA) receptors are a group of GPCRs that respond to LPA, a bioactive lipid involved in cell proliferation, migration, and survival. LPA signaling plays a crucial role in various physiological processes, including wound healing, vascular development, and cancer metastasis. Modulation of LPA receptor activity is being explored for therapeutic applications in cancer, fibrosis, and inflammatory diseases. At CymitQuimica, we offer a range of high-quality LPA receptor modulators to support your research in cell signaling, oncology, and inflammatory disorders.
Found 21 products for "LPA Receptor".
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AM095 free acid
CAS:AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for recombinant human or mouse LPA1).Formula:C27H24N2O5Purity:99.88%Color and Shape:SolidMolecular weight:456.4899Edg-2 receptor inhibitor 1
CAS:Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).Formula:C27H27NO5Purity:99.47%Color and Shape:SolidMolecular weight:445.507TAK-615
CAS:TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.Formula:C25H22FNO4Purity:99.73%Color and Shape:SolidMolecular weight:419.4449ACT-1016-0707
CAS:ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis modelsFormula:C19H23ClN4O4SPurity:99.90%Color and Shape:White SolidMolecular weight:438.93Ki16198
CAS:Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).Formula:C24H25ClN2O5SPurity:98.09%Color and Shape:SolidMolecular weight:488.984BMS-986020 sodium
CAS:BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formula:C29H25N2NaO5Purity:99.83%Color and Shape:White SolidMolecular weight:504.51Tetradecyl Phosphonate
CAS:Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formula:C14H31O3PPurity:99.95%Color and Shape:SolidMolecular weight:278.3679AM966
CAS:AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.Formula:C27H23ClN2O5Purity:98.06% - 99.79%Color and Shape:White SolidMolecular weight:490.935ONO-7300243
CAS:ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).Formula:C28H31NO5Purity:99.66%Color and Shape:SolidMolecular weight:461.5494BMS-986020
CAS:BMS-986020 (AM152) is a selective antagonist of LPA1.Formula:C29H26N2O5Purity:98.82% - >99.99%Color and Shape:SolidMolecular weight:482.5271AM095
CAS:AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.Formula:C27H23N2NaO5Purity:97.05% - 99.71%Color and Shape:SolidMolecular weight:478.4717H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:98.25% - 99.47%Color and Shape:SolidMolecular weight:404.3292Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formula:C23H23ClN2O5SPurity:97.6% - 97.78%Color and Shape:White SolidMolecular weight:474.96BMS-986278
CAS:BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,Formula:C22H31N5O5Purity:99.83% - 99.88%Color and Shape:White SolidMolecular weight:445.512Radioprotectin-1
CAS:Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.Formula:C23H19ClN2O6SPurity:98.63% - 99.27%Color and Shape:White SolidMolecular weight:486.925LPA2 antagonist 1
CAS:LPA2 antagonist 1 is a potent LPA2 antagonist.Formula:C20H23Cl2N5O2S2Purity:99.85%Color and Shape:SolidMolecular weight:500.465LPA2 antagonist 2
CAS:LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.Formula:C20H16N2O6Purity:99.29%Color and Shape:SolidMolecular weight:380.3508TC LPA5 4
CAS:TC LPA5 4 is a LPA5 receptor antagonist.Formula:C23H23ClN2O3Purity:99.93%Color and Shape:SolidMolecular weight:410.89ASP6432
CAS:ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.Formula:C26H32KN4O6S2Color and Shape:SolidMolecular weight:599.78LPA1 receptor antagonist 1
CAS:LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a lysophosphatidic acid receptor antagonist for the study of idiopathic pulmonary fibrosis.Formula:C28H26N4O4Purity:99.56% - 99.87%Color and Shape:SolidMolecular weight:482.53
