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GPCR19

GPCR19

GPCR19, also known as GPR19, is a member of the G protein-coupled receptor family with roles that are still being elucidated in various physiological processes. Although less characterized than other GPCRs, GPCR19 is of interest in research focused on discovering new therapeutic targets for metabolic diseases, cancer, and neurological disorders. At CymitQuimica, we offer a selection of research tools and reagents to support your investigations into the functions and potential therapeutic applications of GPCR19.

Found 31 products of "GPCR19"

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  • SB756050
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    SB756050

    CAS:
    <p>SB756050 is a specific TGR5 agonist.</p>
    Formula:C21H28N2O8S2
    Purity:98.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:500.59

    Ref: TM-T4352

  • Ursodeoxycholic acid sodium
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    Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Formula:C24H40NaO4
    Purity:99.66% - 99.96%
    Color and Shape:Solid
    Molecular weight:415.56

    Ref: TM-T29078

  • CAY10789
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    CAY10789

    CAS:
    <p>CAY10789: potent CysLT1R antagonist (IC50 2.8 µM), GPBAR1 agonist (EC50 3 µM), reduces U937 cell adhesion, TNF-α, stable with promising pharmacokinetics.</p>
    Formula:C17H15NO2
    Color and Shape:Solid
    Molecular weight:265.31

    Ref: TM-T60439

  • WB403
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    WB403

    CAS:
    <p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>
    Formula:C19H19BrN2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.34

    Ref: TM-T29154

  • TGR5 agonist 3
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    TGR5 agonist 3

    CAS:
    <p>Compound 8, a cholic acid derivative, functions as a selective TGR5 agonist and exhibits an EC50 value of 5 μM [1].</p>
    Formula:C28H48O5
    Color and Shape:Solid
    Molecular weight:464.68

    Ref: TM-T79424

  • INT-777 R-enantiomer
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    INT-777 R-enantiomer

    CAS:
    <p>INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5.</p>
    Formula:C27H46O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:450.65

    Ref: TM-T11662

  • RO5527239
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    RO5527239

    CAS:
    <p>RO5527239 is a potent, orally available GPBAR1 agonist agent.</p>
    Formula:C28H31N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.56

    Ref: TM-T26108

  • INT-777
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    INT-777

    CAS:
    <p>INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.</p>
    Formula:C27H46O5
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:450.65

    Ref: TM-T11662L

  • CymitQuimica logo
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    5-HT7R antagonist 1

    <p>5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.</p>
    Formula:C14H18Cl2N4
    Color and Shape:Solid
    Molecular weight:313.23

    Ref: TM-T60790

  • TGR5 Receptor Agonist 3
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    TGR5 Receptor Agonist 3

    CAS:
    <p>TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) &amp; 209 nM (mTGR5), ensures gallbladder safety and reduces filling.</p>
    Formula:C29H27N3O6
    Color and Shape:Solid
    Molecular weight:513.54

    Ref: TM-T63554

  • GPBAR1-IN-3
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    GPBAR1-IN-3

    CAS:
    <p>GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].</p>
    Formula:C21H23NO2
    Color and Shape:Solid
    Molecular weight:321.41

    Ref: TM-T60863