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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • PSB-10 hydrochloride
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    PSB-10 hydrochloride

    CAS:
    <p>PSB-10 hydrochloride is a human adenosine A3 receptor antagonist.</p>
    Formula:C16H15Cl4N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.14

    Ref: TM-T23198

  • MSX-2
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    MSX-2

    CAS:
    <p>MSX-2 is an A2A adenosine receptor antagonist.</p>
    Formula:C21H22N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.42

    Ref: TM-T25840

  • MNI-444
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    MNI-444

    CAS:
    <p>MNI-444 is a PET radiotracer for adenosine 2A receptors.</p>
    Formula:C24H26FN9O2
    Color and Shape:Solid
    Molecular weight:491.52

    Ref: TM-T33461

  • KF21213
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    KF21213

    CAS:
    <p>KF21213 shows a high affinity for the adenosine A2A receptors (Ki=3.0 nM). KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors.</p>
    Formula:C19H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:354.4

    Ref: TM-T13745

  • ATL802
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    ATL802

    CAS:
    <p>ATL802 is an adenosine A2B Receptor antagonist.</p>
    Formula:C24H22F3N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:513.47

    Ref: TM-T26681

  • MRS5698
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    MRS5698

    CAS:
    <p>MRS5698, an A3 adenosine receptor agonist with Ki ~3 nM, blocks chronic pain, highly selective (&gt;1000-fold over A1/A2A).</p>
    Formula:C28H23ClF2N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:564.97

    Ref: TM-T28106

  • ST4206
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    ST4206

    CAS:
    <p>ST4206 is an antagonist of adenosine A2A. For adenosine A2A receptor and adenosine A1 receptor, the Kis values are 12 nM and 197 nM , respectively.</p>
    Formula:C12H14N8O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:286.29

    Ref: TM-T14015

  • A1/A3 AR antagonist 3
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    A1/A3 AR antagonist 3

    CAS:
    <p>A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in</p>
    Formula:C22H19N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.42

    Ref: TM-T79027

  • PF-02575799
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    PF-02575799

    CAS:
    <p>PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).</p>
    Formula:C42H37FN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:680.77

    Ref: TM-T16158

  • PSB 0788
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    PSB 0788

    CAS:
    <p>adenosine A2B receptor antagonist</p>
    Formula:C25H27ClN6O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:543.04

    Ref: TM-T23197

  • CGS 21680
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    CGS 21680

    CAS:
    <p>CGS 21680 is a chemical compound that acts as a selective agonist for both adenosine and its A2A receptor, demonstrating a binding affinity (K i) of 27 nM.</p>
    Formula:C23H29N7O6
    Color and Shape:Solid
    Molecular weight:499.52

    Ref: TM-T6441L

  • Dansyl-NECA
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    Dansyl-NECA

    CAS:
    <p>Dansyl-NECA is a selective agonist of fluorescent adenosine A1 receptor.</p>
    Formula:C30H40N8O6S
    Color and Shape:Solid
    Molecular weight:640.75

    Ref: TM-T23964

  • PSB-1901 free base
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    PSB-1901 free base

    CAS:
    <p>PSB-1901: potent A2B Adenosine Receptor Antagonist; Ki=0.0835 nM; &gt;10,000x selective; effective in mice for preclinical studies.</p>
    Formula:C24H25BrN6O4S
    Color and Shape:Solid
    Molecular weight:573.46

    Ref: TM-T69675

  • CV1808
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    CV1808

    CAS:
    <p>CV-1808 is a coronary vasodilator, antihypertensive, and antipsychotic following systemic administration in vivo. CV-1808 is an adenosine A2 receptor agonist.</p>
    Formula:C16H18N6O4
    Color and Shape:Off-White To Pale Yellow Solid
    Molecular weight:358.35

    Ref: TM-T19696

  • GS-6201
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    GS-6201

    CAS:
    <p>GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.</p>
    Formula:C21H21F3N6O2
    Purity:99.74% - 99.78%
    Color and Shape:Solid
    Molecular weight:446.43

    Ref: TM-T15418

  • MRS 1754
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    MRS 1754

    CAS:
    <p>MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.</p>
    Formula:C26H26N6O4
    Purity:97.57% - 99.3%
    Color and Shape:Solid
    Molecular weight:486.52

    Ref: TM-T16140

  • A2B receptor antagonist 1
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    A2B receptor antagonist 1

    CAS:
    <p>A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.</p>
    Formula:C21H24N6O2
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:392.45

    Ref: TM-T10058

  • PSB-603
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    PSB-603

    CAS:
    <p>PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.</p>
    Formula:C24H25ClN6O4S
    Purity:97.13%
    Color and Shape:Solid
    Molecular weight:529.01

    Ref: TM-T23203

  • PSB 1115
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    PSB 1115

    CAS:
    <p>PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.</p>
    Formula:C14H14N4O5S
    Purity:98.69% - >99.99%
    Color and Shape:Solid
    Molecular weight:350.35

    Ref: TM-T23201

  • CymitQuimica logo
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    A1/A3 AR antagonist 1

    <p>Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.</p>
    Formula:C24H18N2O3S
    Color and Shape:Solid
    Molecular weight:414.48

    Ref: TM-T62134