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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • Norisoboldine hydrochloride

    CAS:
    <p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>
    Formula:C18H20ClNO4
    Color and Shape:Solid
    Molecular weight:349.81
  • FSCPX

    CAS:
    <p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>
    Formula:C23H27FN4O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.55
  • LUF7690

    CAS:
    <p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>
    Formula:C25H24FN5O6S
    Color and Shape:Solid
    Molecular weight:541.55
  • Adenosine receptor antagonist 1

    CAS:
    <p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>
    Formula:C22H15ClFN7O
    Color and Shape:Solid
    Molecular weight:447.86
  • N6-Benzyl-5'-ethylcarboxamido adenosine

    CAS:
    <p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>
    Formula:C19H22N6O4
    Color and Shape:Solid
    Molecular weight:398.42
  • A3AR modulator 1


    <p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>
    Formula:C23H25IN4
    Color and Shape:Solid
    Molecular weight:484.38
  • Adenosine receptor agonist 1


    <p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>
    Formula:C12H14ClN5O2Se
    Color and Shape:Solid
    Molecular weight:374.68
  • PSB 0777 ammonium salt

    CAS:
    <p>adenosine A2A receptor full agonist</p>
    Formula:C18H24N6O7S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55
  • Apadenoson TFA


    <p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>
    Formula:C25H31F3N6O8
    Purity:98.08%
    Color and Shape:Soild
    Molecular weight:600.55
  • Heterobivalent ligand-1


    <p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>
    Formula:C86H115FN16O21
    Color and Shape:Solid
    Molecular weight:1727.93
  • GW-328267

    CAS:
    <p>GW-328267 is an agonist of the adenosine A2 receptor.</p>
    Formula:C21H26N10O4
    Color and Shape:Solid
    Molecular weight:482.5
  • MRS-1706

    CAS:
    <p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>
    Formula:C27H29N5O5
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:503.55
  • Xanthine amine congener trihydrochloride

    CAS:
    <p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>
    Formula:C21H29ClN6O4
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:464.95
  • ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:463.33
  • Xanthine amine congener dihydrochloride

    CAS:
    <p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>
    Formula:C21H30Cl2N6O4
    Color and Shape:Solid
    Molecular weight:501.41
  • A-286501

    CAS:
    <p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>
    Formula:C11H14BrN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.17
  • Danshenol B


    <p>Danshenol B is a natural product that can be used as a reference standard.</p>
    Formula:C22H26O4
    Color and Shape:Solid
    Molecular weight:354.446
  • AR ligand 40


    <p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>
    Formula:C21H25N5
    Color and Shape:Solid
    Molecular weight:347.211
  • Theophyllol

    CAS:
    <p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>
    Formula:C9H10N4Na2O4
    Color and Shape:Solid
    Molecular weight:284.18
  • LUF6096

    CAS:
    <p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>
    Formula:C22H21Cl2N3O
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:414.33