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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • SCH 58261

    CAS:
    <p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>
    Formula:C18H15N7O
    Purity:99.07% - 99.75%
    Color and Shape:Solid
    Molecular weight:345.36
  • Tozadenant

    CAS:
    <p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>
    Formula:C19H26N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.5
  • CPI-444

    CAS:
    <p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>
    Formula:C20H21N7O3
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:407.43
  • Preladenant

    CAS:
    <p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has &gt;1000-fold selectivity over all other adenosine</p>
    Formula:C25H29N9O3
    Purity:98.02% - 99.68%
    Color and Shape:Solid
    Molecular weight:503.56
  • Binodenoson

    CAS:
    <p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>
    Formula:C17H25N7O4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:391.42
  • Proxyphylline

    CAS:
    <p>Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.</p>
    Formula:C10H14N4O3
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:238.24
  • DPCPX

    CAS:
    <p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>
    Formula:C16H24N4O2
    Purity:99.23% - 99.93%
    Color and Shape:White Solid
    Molecular weight:304.39
  • Tecadenoson

    CAS:
    <p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>
    Formula:C14H19N5O5
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:337.33
  • A2B receptor antagonist 2

    CAS:
    <p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>
    Formula:C12H15N5
    Purity:100%
    Color and Shape:Solid
    Molecular weight:229.28
  • Inosine

    CAS:
    <p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>
    Formula:C10H12N4O5
    Purity:99.51% - 99.89%
    Color and Shape:Solid
    Molecular weight:268.23
  • CHEMBL241987

    CAS:
    <p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>
    Formula:C16H11N3O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:261.28
  • Adenosine receptor antagonist 4

    CAS:
    <p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>
    Formula:C10H13N3
    Purity:99.63% - 99.65%
    Color and Shape:Off-White Powder
    Molecular weight:175.23
  • 5-Iodotubercidin

    CAS:
    <p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>
    Formula:C11H13IN4O4
    Purity:99.98%
    Color and Shape:Tan Solid
    Molecular weight:392.15
  • MIPS521

    CAS:
    <p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>
    Formula:C19H10ClF6NOS
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:449.8
  • CCPA

    CAS:
    <p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>
    Formula:C15H20ClN5O4
    Purity:99.1%
    Color and Shape:Off-White To Light Yellow Solid
    Molecular weight:369.8
  • 5'-N-Ethylcarboxamidoadenosine

    CAS:
    <p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>
    Formula:C12H16N6O4
    Purity:98.95% - ≥95%
    Color and Shape:Powder
    Molecular weight:308.29
  • Regadenoson

    CAS:
    <p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>
    Formula:C15H18N8O5
    Purity:99.57% - 99.81%
    Color and Shape:Off-White Solid
    Molecular weight:390.35
  • Namodenoson

    CAS:
    <p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>
    Formula:C18H18ClIN6O4
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:544.73
  • BAY-545

    CAS:
    <p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>
    Formula:C18H22F3N3O4S
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:433.45
  • Vipadenant

    CAS:
    <p>Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).</p>
    Formula:C16H15N7O
    Purity:97.25% - 97.36%
    Color and Shape:Solid
    Molecular weight:321.34