Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 242 products of "Adenosine Receptor"
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5'-Amino-5'-deoxyadenosine
CAS:<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Formula:C10H14N6O3Purity:95.55%Color and Shape:SolidMolecular weight:266.26Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Color and Shape:LiquidAdenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Formula:C17H19ClFN5O3Color and Shape:SolidMolecular weight:395.82A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Formula:C17H12N4OColor and Shape:SolidMolecular weight:288.3TC-G 1004
CAS:<p>adenosine A2A receptors antagonist</p>Formula:C22H27N7O2Purity:98%Color and Shape:SolidMolecular weight:421.5SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Formula:C15H13N3SPurity:98%Color and Shape:SolidMolecular weight:267.35A2AR-agonist-1
CAS:<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43Lu AA 47070
CAS:<p>adenosine A2A receptor antagonist</p>Formula:C17H20F2N3O6PSPurity:98%Color and Shape:SolidMolecular weight:463.39VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36Acefylline piperazine
CAS:<p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>Formula:C9H10N4O4·xC4H10N2Color and Shape:SolidMolecular weight:562.54CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52CVT-2759
CAS:<p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>Formula:C17H24N6O6Color and Shape:SolidMolecular weight:408.41MRS-1191
CAS:<p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>Formula:C31H27NO4Color and Shape:SolidMolecular weight:477.55Adenosine receptor inhibitor 2
CAS:<p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>Formula:C17H20BrN5O2Color and Shape:SolidMolecular weight:406.28Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Formula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Formula:C20H19N3O4SColor and Shape:SolidMolecular weight:397.45Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31
