Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 249 products of "Adenosine Receptor"
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Adenosine receptor antagonist 2
CAS:Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFormula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31Sipagladenant
CAS:Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.Formula:C20H19N3O4SColor and Shape:SolidMolecular weight:397.45SCH-202676 HBr
CAS:SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.Formula:C15H13N3SPurity:98%Color and Shape:SolidMolecular weight:267.35A3AR antagonist 2
CAS:A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.Formula:C22H16N6O3Color and Shape:SolidMolecular weight:412.4TH-162
CAS:TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42PQ-69
CAS:PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.Formula:C20H19FN4OColor and Shape:SolidMolecular weight:350.39MRS 1523
CAS:MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.Formula:C23H29NO3SPurity:98%Color and Shape:SolidMolecular weight:399.55Inupadenant
CAS:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65CAY10680
CAS:CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4FR-194921
CAS:FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Formula:C23H23N5OColor and Shape:SolidMolecular weight:385.46CVT-2759
CAS:CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.Formula:C17H24N6O6Color and Shape:SolidMolecular weight:408.41Adenosine receptor inhibitor 2
CAS:Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.Formula:C17H20BrN5O2Color and Shape:SolidMolecular weight:406.28Acefylline piperazine
CAS:Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.Formula:C9H10N4O4·xC4H10N2Color and Shape:SolidMolecular weight:562.54JNJ-40255293
CAS:JNJ-40255293 is an antagonist of adenosine A2A/A1.Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42ATL-801
CAS:ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.Formula:C24H25N7O3Color and Shape:SolidMolecular weight:459.5Kira8 Hydrochloride
CAS:Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formula:C31H30Cl2N6O3SPurity:98%Color and Shape:SolidMolecular weight:637.58
