Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 242 products of "Adenosine Receptor"
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Xanthine amine congener hydrochloride
CAS:<p>Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.</p>Formula:C21H29ClN6O4Color and Shape:SolidMolecular weight:464.95Norisoboldine
CAS:<p>Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.</p>Formula:C18H19NO4Purity:98.12% - 99.7%Color and Shape:SolidMolecular weight:313.35SCH442416
CAS:<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Derenofylline
CAS:<p>Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)</p>Formula:C18H20N4OPurity:98.09%Color and Shape:SolidMolecular weight:308.38CGS 21680 Hydrochloride
CAS:<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Formula:C23H29N7O6·HClPurity:96.74% - 99.53%Color and Shape:SolidMolecular weight:535.98Regadenoson hydrate
CAS:<p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>Formula:C15H20N8O6Purity:98%Color and Shape:SolidMolecular weight:408.37Preladenant
CAS:<p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosine</p>Formula:C25H29N9O3Purity:98.02% - 99.68%Color and Shape:SolidMolecular weight:503.56ZM241385
CAS:<p>ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.</p>Formula:C16H15N7O2Purity:97.02% - 99.69%Color and Shape:SolidMolecular weight:337.348-Cyclopentyl-1,3-dimethylxanthine
CAS:<p>8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.</p>Formula:C12H16N4O2Purity:98.58% - >99.99%Color and Shape:SolidMolecular weight:248.28CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28Inosine
CAS:<p>Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!</p>Formula:C10H12N4O5Purity:99.51% - 99.89%Color and Shape:SolidMolecular weight:268.23Tecadenoson
CAS:<p>Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.</p>Formula:C14H19N5O5Purity:98.83%Color and Shape:SolidMolecular weight:337.332-Chloroadenosine
CAS:<p>2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectively</p>Formula:C10H12ClN5O4Purity:99.23%Color and Shape:White PowderMolecular weight:301.69ABT-702 dihydrochloride
CAS:<p>ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.</p>Formula:C22H21BrCl2N6OPurity:98.42% - 98.98%Color and Shape:SolidMolecular weight:536.25Tozadenant
CAS:<p>Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)</p>Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5SCH 58261
CAS:<p>SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.</p>Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Alloxazine
CAS:<p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18Reversine
CAS:<p>Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).</p>Formula:C21H27N7OPurity:98% - 98.42%Color and Shape:SolidMolecular weight:393.49Fostamatinib
CAS:<p>Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.</p>Formula:C23H26FN6O9PPurity:93.08% - 99.38%Color and Shape:SolidMolecular weight:580.46Capadenoson
CAS:<p>Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.</p>Formula:C25H18ClN5O2S2Purity:98.85% - 99.57%Color and Shape:SolidMolecular weight:520.03Adenosine amine congener
CAS:<p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43A2B receptor antagonist 2
CAS:<p>A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).</p>Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28Proxyphylline
CAS:<p>Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.</p>Formula:C10H14N4O3Purity:99.48%Color and Shape:SolidMolecular weight:238.24CCPA
CAS:<p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>Formula:C15H20ClN5O4Purity:99.1%Color and Shape:Off-White To Light Yellow SolidMolecular weight:369.8DPCPX
CAS:<p>DPCPX (PD 116948) is an A1 adenosine receptor antagonist</p>Formula:C16H24N4O2Purity:99.23% - 99.93%Color and Shape:White SolidMolecular weight:304.39Nitrobenzylthioinosine
CAS:<p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Vipadenant
CAS:<p>Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).</p>Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34PD 117519
CAS:<p>PD 117519 (CI947) is an agonist of adenosine receptor</p>Formula:C19H21N5O4Purity:99.98%Color and Shape:SolidMolecular weight:383.4SDZ WAG 994
CAS:<p>SDZ WAG 994 is an A1 adenosine receptor agonist.</p>Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41MIPS521
CAS:<p>MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.</p>Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73Regadenoson
CAS:<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.355'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purity:98.95% - ≥95%Color and Shape:PowderMolecular weight:308.295-Iodotubercidin
CAS:<p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15Taminadenant
CAS:<p>Taminadenant is an adenosine receptor antagonist.</p>Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12AZD4635
CAS:<p>AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).</p>Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.73VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Piclidenoson
CAS:<p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>Formula:C18H19IN6O4Purity:99.83% - ≥95%Color and Shape:SolidMolecular weight:510.29Istradefylline
CAS:<p>Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.</p>Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43Enprofylline
CAS:<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Swertisin
CAS:<p>Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.</p>Formula:C22H22O10Purity:99.74% - 99.89%Color and Shape:SolidMolecular weight:446.4Adenosine receptor antagonist 4
CAS:<p>Adenosine receptor antagonist 4 is an adenosine receptor antagonist.</p>Formula:C10H13N3Purity:99.63% - 99.65%Color and Shape:Off-White PowderMolecular weight:175.231-Ethyl-6-aminouracil
CAS:<p>1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high</p>Formula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15N6,N6-Dimethyladenosine
CAS:<p>N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.</p>Formula:C12H17N5O4Purity:98.79%Color and Shape:White PowderMolecular weight:295.29Binodenoson
CAS:<p>Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.</p>Formula:C17H25N7O4Purity:99.74%Color and Shape:SolidMolecular weight:391.42Rolofylline
CAS:<p>Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.</p>Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.365'-Amino-5'-deoxyadenosine
CAS:<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Formula:C10H14N6O3Purity:95.55%Color and Shape:SolidMolecular weight:266.26
