Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 249 products of "Adenosine Receptor"
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Theophylline-d6
CAS:Theophylline-d6, an internal standard for theophylline quantification in GC/LC-MS, relaxes bronchial muscles and treats asthma/COPD.Formula:C7H2D6N4O2Color and Shape:SolidMolecular weight:186.2Norisoboldine
CAS:Norisoboldine, potential rheumatoid arthritis therapy, protects joints and modulates immunity by inhibiting MAPKs, not NF-κB.Formula:C18H19NO4Purity:98.12% - 99.7%Color and Shape:SolidMolecular weight:313.35SCH442416
CAS:SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).Formula:C20H19N7O2Purity:99.58%Color and Shape:SolidMolecular weight:389.41Ref: TM-T23336
1mg46.00€5mg88.00€10mg132.00€25mg266.00€50mg409.00€100mg573.00€200mg807.00€1mL*10mM (DMSO)92.00€Derenofylline
CAS:Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formula:C18H20N4OPurity:98.09%Color and Shape:SolidMolecular weight:308.38ZM241385
CAS:ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Formula:C16H15N7O2Purity:97.02% - 99.69%Color and Shape:SolidMolecular weight:337.34ABT-702 dihydrochloride
CAS:ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.Formula:C22H21BrCl2N6OPurity:98.42% - 98.98%Color and Shape:SolidMolecular weight:536.25Ref: TM-T4668
1mg58.00€2mg82.00€5mg113.00€10mg177.00€25mg333.00€50mg502.00€100mg710.00€500mg1,494.00€1mL*10mM (DMSO)133.00€Regadenoson hydrate
CAS:Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.Formula:C15H20N8O6Purity:98%Color and Shape:SolidMolecular weight:408.372-Chloroadenosine
CAS:2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, and A3 receptors( Ki:300, 80, and 1,900 nM, respectivelyFormula:C10H12ClN5O4Purity:99.23%Color and Shape:White PowderMolecular weight:301.69Preladenant
CAS:Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has >1000-fold selectivity over all other adenosineFormula:C25H29N9O3Purity:98.02% - 99.68%Color and Shape:SolidMolecular weight:503.56Xanthine amine congener hydrochloride
CAS:Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.Formula:C21H29ClN6O4Color and Shape:SolidMolecular weight:464.95Inosine
CAS:Inosine (NSC-20262), an endogenous purine nucleoside produced by the catabolism of adenosine, is an agonist of adenosine receptors A1R and A2AR. Low-Cost!Formula:C10H12N4O5Purity:99.51% - 99.89%Color and Shape:SolidMolecular weight:268.238-Cyclopentyl-1,3-dimethylxanthine
CAS:8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formula:C12H16N4O2Purity:98.58% - 99.9%Color and Shape:SolidMolecular weight:248.28Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Tecadenoson
CAS:Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formula:C14H19N5O5Purity:98.83%Color and Shape:SolidMolecular weight:337.33Binodenoson
CAS:Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formula:C17H25N7O4Purity:99.74%Color and Shape:SolidMolecular weight:391.42Ref: TM-T9516
1mg94.00€5mg222.00€10mg334.00€25mg557.00€50mg745.00€100mg1,044.00€1mL*10mM (DMSO)245.00€CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28CGS 21680 Hydrochloride
CAS:CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formula:C23H29N7O6·HClPurity:96.74% - 99.53%Color and Shape:SolidMolecular weight:535.98Ref: TM-T6441
1mg38.00€2mg50.00€5mg81.00€10mg109.00€25mg215.00€50mg389.00€100mg575.00€1mL*10mM (DMSO)95.00€Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg42.00€5mg62.00€10mg88.00€25mg141.00€50mg215.00€100mg318.00€200mg442.00€1mL*10mM (DMSO)59.00€Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formula:C25H18ClN5O2S2Purity:98.85% - 99.57%Color and Shape:SolidMolecular weight:520.03SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Ref: TM-T6979
1mg38.00€2mg49.00€5mg80.00€10mg118.00€25mg213.00€50mg344.00€100mg550.00€1mL*10mM (DMSO)81.00€A2B receptor antagonist 2
CAS:A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).Formula:C12H15N5Purity:100%Color and Shape:SolidMolecular weight:229.28Fostamatinib
CAS:Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn.
Formula:C23H26FN6O9PPurity:93.08% - 99.38%Color and Shape:SolidMolecular weight:580.46Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5Alloxazine
CAS:Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.Formula:C10H6N4O2Purity:99.75%Color and Shape:SolidMolecular weight:214.18Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43Ref: TM-T7183
2mg34.00€5mg52.00€10mg73.00€25mg128.00€50mg197.00€100mg295.00€200mg442.00€1mL*10mM (DMSO)52.00€MIPS521
CAS:MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.Formula:C19H10ClF6NOSPurity:99.76%Color and Shape:SolidMolecular weight:449.8Ref: TM-T9330
1mg35.00€2mg50.00€5mg74.00€10mg105.00€25mg178.00€50mg313.00€100mg485.00€1mL*10mM (DMSO)82.00€DPCPX
CAS:DPCPX (PD 116948) is an A1 adenosine receptor antagonistFormula:C16H24N4O2Purity:99.23% - 99.93%Color and Shape:White SolidMolecular weight:304.39CCPA
CAS:CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptorFormula:C15H20ClN5O4Purity:99.1%Color and Shape:Off-White To Light Yellow SolidMolecular weight:369.8Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34Ref: TM-T2373
2mg35.00€5mg51.00€10mg80.00€25mg131.00€50mg210.00€100mg313.00€200mg445.00€1mL*10mM (DMSO)215.00€PD 117519
CAS:PD 117519 (CI947) is an agonist of adenosine receptorFormula:C19H21N5O4Purity:99.98%Color and Shape:SolidMolecular weight:383.4SDZ WAG 994
CAS:SDZ WAG 994 is an A1 adenosine receptor agonist.Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41Ref: TM-T23347
1mg63.00€5mg114.00€10mg172.00€25mg299.00€50mg432.00€100mg587.00€200mg792.00€1mL*10mM (DMSO)120.00€Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.735-Iodotubercidin
CAS:5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.
Formula:C11H13IN4O4Purity:99.98%Color and Shape:Tan SolidMolecular weight:392.15Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
2mg34.00€5mg49.00€10mg84.00€25mg114.00€50mg166.00€100mg236.00€200mg353.00€1mL*10mM (DMSO)54.00€N6,N6-Dimethyladenosine
CAS:N6,N6-Dimethyladenosine is find in mycobacterium bovis Bacille Calmette-Guérin tRNA.
Formula:C12H17N5O4Purity:98.79%Color and Shape:White PowderMolecular weight:295.29AZD4635
CAS:AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).Formula:C15H11ClFN5Purity:99.15% - 99.90%Color and Shape:SolidMolecular weight:315.73Ref: TM-T4265
1mg37.00€2mg52.00€5mg79.00€10mg116.00€25mg188.00€50mg296.00€100mg457.00€500mg1,008.00€1mL*10mM (DMSO)87.00€1-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg84.00€5mg161.00€10mg235.00€25mg420.00€50mg605.00€100mg842.00€200mg1,134.00€1mL*10mM (DMSO)172.00€Regadenoson
CAS:Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.Formula:C15H18N8O5Purity:99.57% - 99.81%Color and Shape:Off-White SolidMolecular weight:390.35Ref: TM-T2671
2mg47.00€5mg65.00€10mg92.00€25mg173.00€50mg273.00€100mg416.00€500mg935.00€1mL*10mM (DMSO)72.00€Reversine
CAS:Reversine, a small synthetic purine analogue (2, 6-disubstituted purine), is a potent inhibitior of Aurora A/B/C(IC50s=150-500 nM).Formula:C21H27N7OPurity:98% - 99.45%Color and Shape:SolidMolecular weight:393.49Ref: TM-T1825
1mg35.00€2mg50.00€5mg66.00€10mg84.00€25mg156.00€50mg212.00€100mg371.00€1mL*10mM (DMSO)66.00€Swertisin
CAS:Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.Formula:C22H22O10Purity:99.74% - 99.89%Color and Shape:SolidMolecular weight:446.40Adenosine receptor antagonist 4
CAS:Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formula:C10H13N3Purity:99.63% - 99.65%Color and Shape:Off-White PowderMolecular weight:175.23Istradefylline
CAS:Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is under development in Phase 3 trails.Formula:C20H24N4O4Purity:98.18% - 99.95%Color and Shape:SolidMolecular weight:384.43VPC171
CAS:VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).Formula:C18H12F3NOSPurity:99.78%Color and Shape:SolidMolecular weight:347.35Ref: TM-T29112
1mg49.00€5mg96.00€10mg124.00€25mg222.00€50mg309.00€100mg439.00€200mg592.00€1mL*10mM (DMSO)88.00€Piclidenoson
CAS:Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.Formula:C18H19IN6O4Purity:99.83% - ≥95%Color and Shape:SolidMolecular weight:510.29Ref: TM-T7188
2mg42.00€5mg62.00€10mg89.00€25mg183.00€50mg298.00€100mg464.00€200mg663.00€1mL*10mM (DMSO)70.00€5'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formula:C12H16N6O4Purity:98.95% - ≥95%Color and Shape:PowderMolecular weight:308.29Proxyphylline
CAS:Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.Formula:C10H14N4O3Purity:99.48%Color and Shape:SolidMolecular weight:238.24Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.46
