Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 242 products of "Adenosine Receptor"
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Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Color and Shape:LiquidTC-G 1004
CAS:<p>adenosine A2A receptors antagonist</p>Formula:C22H27N7O2Purity:98%Color and Shape:SolidMolecular weight:421.5A2AR-agonist-1
CAS:<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43hA2A/hCA XII modulator 1
CAS:<p>Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.</p>Formula:C24H19N7O4SColor and Shape:SolidMolecular weight:501.52IHCH-3064
CAS:<p>IHCH-3064: dual-action cancer immunotherapy, A2AR affinity (Ki 2.2 nM), selective HDAC1 inhibitor (IC50 80.2 nM).</p>Formula:C25H21N9O2Color and Shape:SolidMolecular weight:479.49MRS 1334
CAS:<p>antagonist for the human adenosine A3 receptor</p>Formula:C31H26N2O6Purity:98%Color and Shape:SolidMolecular weight:522.55LUF6000
CAS:<p>LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).</p>Formula:C22H20Cl2N4Color and Shape:SolidMolecular weight:411.33A2A/A1 AR antagonist-1
CAS:<p>A2A/A1 AR antagonist-1 is a potent dual antagonist for ischemic stroke research with Ki values of 5.58 nM (A2A) and 24.2 nM (A1).</p>Formula:C15H12N6O2Color and Shape:SolidMolecular weight:308.29LUF 5834
CAS:<p>A2A and A2B adenosine receptor partial agonist</p>Formula:C17H12N6OSPurity:98%Color and Shape:SolidMolecular weight:348.385'-(N-Cyclopropyl)carboxamidoadenosine
CAS:<p>adenosine A2 receptor agonist</p>Formula:C13H16N6O4Purity:98%Color and Shape:SolidMolecular weight:320.3A1AR antagonist 5
CAS:<p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>Formula:C17H15ClN4OColor and Shape:SolidMolecular weight:326.78A1AR antagonist 3
CAS:<p>Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.</p>Formula:C25H20N2O3SColor and Shape:SolidMolecular weight:428.5XCC
CAS:<p>XCC is an Adenosine receptor antagonist.</p>Formula:C19H22N4O5Purity:98%Color and Shape:SolidMolecular weight:386.4A1AR antagonist 4
CAS:<p>Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.</p>Formula:C23H25N3O2Color and Shape:SolidMolecular weight:375.46MRS1097
CAS:<p>MRS1097 is a selective antagonist A3 adenosine receptor.</p>Formula:C26H27NO4Purity:98%Color and Shape:SolidMolecular weight:417.5MRS-1191
CAS:<p>MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).</p>Formula:C31H27NO4Color and Shape:SolidMolecular weight:477.55Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52Lu AA 47070
CAS:<p>adenosine A2A receptor antagonist</p>Formula:C17H20F2N3O6PSPurity:98%Color and Shape:SolidMolecular weight:463.39A1AR antagonist 2
CAS:<p>Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.</p>Formula:C17H12N4OColor and Shape:SolidMolecular weight:288.3Adenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Formula:C17H19ClFN5O3Color and Shape:SolidMolecular weight:395.82A1/A3 AR antagonist 2
CAS:<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Formula:C22H16N2O3SColor and Shape:SolidMolecular weight:388.44AB-MECA
CAS:<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Formula:C18H21N7O4Purity:98%Color and Shape:SolidMolecular weight:399.4A2AAR/HDAC-IN-1
CAS:<p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>Formula:C24H21N7O2Color and Shape:SolidMolecular weight:439.47LASSBio-1359
CAS:<p>LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.</p>Formula:C17H18N2O3Purity:98%Color and Shape:SolidMolecular weight:298.34PSB 11 hydrochloride
CAS:<p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>Formula:C16H18ClN5OPurity:98%Color and Shape:SolidMolecular weight:331.8Adenosine receptor antagonist 3
CAS:<p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>Formula:C16H14N6SColor and Shape:SolidMolecular weight:322.39Adentri
CAS:<p>Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.</p>Formula:C18H24N4O3Purity:98%Color and Shape:SolidMolecular weight:344.41A2A receptor antagonist 3
CAS:<p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>Formula:C26H26N6O2Color and Shape:SolidMolecular weight:454.52MRS1186
CAS:<p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>Formula:C16H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:341.75Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Formula:C17H20N4O2Purity:99.97%Color and Shape:SolidMolecular weight:312.37MRS1177
CAS:<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Formula:C20H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:389.79XU1
CAS:<p>XU1（Benzo[c][1,8]naphthyridin-6(5h)-One） is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Formula:C12H8N2OPurity:98.58% - 99.59%Color and Shape:SolidMolecular weight:196.2HEMADO
CAS:<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Formula:C17H23N5O4Purity:98%Color and Shape:SolidMolecular weight:361.4A1AR antagonist 6
CAS:<p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>Formula:C17H15N3O2Color and Shape:SolidMolecular weight:293.32Lu AA41063
CAS:<p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>Formula:C16H17F2N3O2SColor and Shape:SolidMolecular weight:353.39Neladenoson dalanate HCl
CAS:<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Formula:C35H35Cl2N7O4S2Purity:98%Color and Shape:SolidMolecular weight:752.73A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formula:C32H24N4O4SColor and Shape:SolidMolecular weight:560.62Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Formula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31Sipagladenant
CAS:<p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>Formula:C20H19N3O4SColor and Shape:SolidMolecular weight:397.45SCH-202676 HBr
CAS:<p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>Formula:C15H13N3SPurity:98%Color and Shape:SolidMolecular weight:267.35A3AR antagonist 2
CAS:<p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>Formula:C22H16N6O3Color and Shape:SolidMolecular weight:412.4TH-162
CAS:<p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42PQ-69
CAS:<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Formula:C20H19FN4OColor and Shape:SolidMolecular weight:350.39MRS 1523
CAS:<p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.</p>Formula:C23H29NO3SPurity:98%Color and Shape:SolidMolecular weight:399.55Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65CAY10680
CAS:<p>CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.</p>Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4
