Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
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Istradefylline
CAS:155270-99-8
Istradefylline (KW-6002)(Ki of 2.2 nM) is a selective adenosine A2A receptor (A2AR) antagonist, which is …
Formula:
C20H24N4O4
Purity:
98.18% - 98.57%
Color and Shape:
Solid
Molecular weight:
384.43
Ref: TM-T6552
| 5mg | 41.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 152.00 € | ||
| 200mg | 222.00 € | ||
| 500mg | 370.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AZD4635
CAS:1321514-06-0
AZD4635 (HTL1071) is a new-type adenosine 2A receptor (A2AR) inhibitor(Ki=1.7 nM).
Formula:
C15H11ClFN5
Purity:
99.15% - 99.61%
Color and Shape:
Solid
Molecular weight:
315.73
Ref: TM-T4265
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 451.00 € | ||
| 500mg | 985.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
5-Iodotubercidin
CAS:24386-93-4
5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.
Formula:
C11H13IN4O4
Purity:
99.98%
Color and Shape:
Tan Solid
Molecular weight:
392.15
Ref: TM-T6745
| 1mg | 45.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 718.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PD 117519
CAS:96392-15-3
PD 117519 (CI947) is an agonist of adenosine receptor
Formula:
C19H21N5O4
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
383.4
Ref: TM-T7509
| 2mg | 35.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Piclidenoson
CAS:152918-18-8
Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust …
Formula:
C18H19IN6O4
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
510.29
Ref: TM-T7188
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 308.00 € | ||
| 50mg | 496.00 € | ||
| 100mg | 771.00 € | ||
| 200mg | 1,023.00 € | ||
| 500mg | 1,538.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Swertisin
CAS:6991-10-2
Swertisin: an herbal molecule with antihyperglycemic, antidiabetic, anti-inflammatory, and antioxidant properties; blocks adenosine A1 receptor.
Formula:
C22H22O10
Purity:
99.74% - 99.79%
Color and Shape:
Solid
Molecular weight:
446.4
Ref: TM-TN2247
| 1mg | 69.00 € | ||
| 5mg | 245.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 602.00 € | ||
| 50mg | 829.00 € | ||
| 1mL*10mM (DMSO) | 277.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
VPC171
CAS:1018830-99-3
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
Formula:
C18H12F3NOS
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
347.35
Ref: TM-T29112
| 1mg | 71.00 € | ||
| 2mg | 93.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 175.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 638.00 € | ||
| 200mg | 859.00 € | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BAY-545
CAS:1699717-32-2
BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).
Formula:
C18H22F3N3O4S
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
433.45
Ref: TM-T8512
| 1mg | 86.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 238.00 € | ||
| 25mg | 428.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 857.00 € | ||
| 200mg | 1,153.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
1-Ethyl-6-aminouracil
CAS:41862-09-3
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines …
Formula:
C6H9N3O2
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
155.15
Ref: TM-T8613
| 2mg | 55.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 388.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Regadenoson
CAS:313348-27-5
Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a …
Formula:
C15H18N8O5
Purity:
100% - 99.78%
Color and Shape:
Off-White Solid
Molecular weight:
390.35
Ref: TM-T2671
| 2mg | 46.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 407.00 € | ||
| 500mg | 914.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
5'-N-Ethylcarboxamidoadenosine
CAS:35920-39-9
NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the …
Formula:
C12H16N6O4
Purity:
≥95%
Color and Shape:
Powder
Molecular weight:
308.29
Ref: TM-T7340
| 5mg | 53.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 146.00 € | ||
| 100mg | 207.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Namodenoson
CAS:163042-96-4
Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
Formula:
C18H18ClIN6O4
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
544.73
Ref: TM-T6884
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Taminadenant
CAS:1337962-47-6
Taminadenant is an adenosine receptor antagonist.
Formula:
C10H8BrN7
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
306.12
Ref: TM-T16980
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Proxyphylline
CAS:603-00-9
Proxyphylline (7-(2-Hydroxypropyl)theophylline) is a dual of adenosine A1/A2a receptor inhibitor and phosphodiesterase (PDE) inhibitor.
Formula:
C10H14N4O3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
238.24
Ref: TM-T5940
| 500mg | 53.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DPCPX
CAS:102146-07-6
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
Formula:
C16H24N4O2
Purity:
99.93%
Color and Shape:
White Solid
Molecular weight:
304.39
Ref: TM-T22744
| 10mg | 48.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 139.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CPI-444
CAS:1202402-40-1
CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse …
Formula:
C20H21N7O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
407.43
Ref: TM-T7183
| 1mg | 40.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 528.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
A2B receptor antagonist 2
CAS:784-90-7
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM …
Formula:
C12H15N5
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
229.28
Ref: TM-T37793
| 10mg | 45.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Capadenoson
CAS:544417-40-5
Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
Formula:
C25H18ClN5O2S2
Purity:
98.85% - 99.62%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-TQ0125
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Enprofylline
CAS:41078-02-8
Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.
Formula:
C8H10N4O2
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
194.19
Ref: TM-T21389
| 2mg | 43.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 146.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 326.00 € | ||
| 200mg | 453.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
SCH 58261
CAS:160098-96-4
SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for …
Formula:
C18H15N7O
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
345.36
Ref: TM-T6979
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 361.00 € | ||
| 100mg | 577.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
