Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Found 217 products of "Cannabinoid Receptor"
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ANEB-001
CAS:ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.Formula:C22H24ClF3N2O2Color and Shape:SolidMolecular weight:440.89CB1R Allosteric modulator 4
CAS:Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43PGN36
CAS:PGN36 (Compound 18) is a potent CB2 receptor antagonist with a high affinity (Ki=0.09 μM).Formula:C21H23N3O3Color and Shape:SolidMolecular weight:365.43CB1R Allosteric modulator 2
CAS:Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.Formula:C19H15ClFN3OColor and Shape:SolidMolecular weight:355.79GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39CB1-IN-2
CAS:CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.Formula:C17H19Cl2N5OColor and Shape:SolidMolecular weight:380.27COR167
CAS:COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.Formula:C28H38N2O2Color and Shape:SolidMolecular weight:434.61UCM 707
CAS:endocannabinoid transport inhibitorFormula:C25H37NO2Purity:98%Color and Shape:SolidMolecular weight:383.57SMM-189
CAS:SMM-189 is a potent and selective CB2 inverse agonist.Formula:C19H12Cl2O3Color and Shape:SolidMolecular weight:359.2CAY10412
CAS:Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.Formula:C25H36O2SColor and Shape:SolidMolecular weight:400.62(S)-SLV 319
CAS:Ibipinabant (SLV319), a potent CB1 antagonist, K i = 7.8 nM, >1000x selective over CB2, for obesity and diabetic research.Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Formula:C23H25FN4O4SPurity:98%Color and Shape:SolidMolecular weight:472.53Palmitoyl serinol
CAS:Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.Formula:C19H39NO3Color and Shape:SolidMolecular weight:329.52ZCZ011
CAS:ZCZ011 enhances CB1 receptor effects, crosses blood-brain barrier, and potentiates cannabimimetic behaviors in mice.Formula:C21H18N2O2SPurity:98%Color and Shape:SolidMolecular weight:362.44KLS-13019
CAS:KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).Formula:C22H29NO3Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:355.47Virodhamine trifluoroacetate
CAS:Virodhamine trifluoroacetate: full GPR55 & CB2 agonist, partial CB1 antagonist, cannabinoid receptor mixed antagonist.Formula:C24H38F3NO4Purity:98%Color and Shape:SolidMolecular weight:461.56OMDM-6
CAS:OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 μM). OMDM-6 inhibits anandamide cellular uptake with a Ki of 7.0 μM.Formula:C28H42N2O3Purity:99.66%Color and Shape:SolidMolecular weight:454.64Ref: TM-T12307
1mg85.00€5mg170.00€10mg250.00€25mg371.00€50mg522.00€100mg712.00€200mg954.00€1mL*10mM (DMSO)187.00€LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Formula:C23H29ClN6O3Color and Shape:SolidMolecular weight:472.97N-Arachidonyldopamine
CAS:N-Arachidonyldopamine (NADA) is a selective and potent endogenous CB1 receptor agonist (Ki: 250 nM).N-Arachidonyldopamine is also a potent and selective TRPV1Formula:C28H41NO3Purity:97.65%Color and Shape:SolidMolecular weight:439.632-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFormula:C23H38O4Purity:95%Color and Shape:LiquidMolecular weight:378.55GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formula:C19H16F4N4Color and Shape:SolidMolecular weight:376.35AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purity:99.6%Color and Shape:SolidMolecular weight:380.36MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Formula:C23H17Cl3N4OPurity:99.63%Color and Shape:SolidMolecular weight:471.77CB1/2 agonist 4
CAS:CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.Formula:C27H45NO3Color and Shape:SolidMolecular weight:431.65CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Formula:C24H24ClN3OColor and Shape:SolidMolecular weight:405.92UCM710
CAS:UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).Formula:C19H34O3Purity:98%Color and Shape:SolidMolecular weight:310.47MM-22
CAS:biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamideFormula:C36H60N4O5SPurity:98%Color and Shape:SolidMolecular weight:660.95CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Formula:C22H32N2OColor and Shape:SolidMolecular weight:340.5S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Formula:C23H27FN2O4Color and Shape:SolidMolecular weight:414.47PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49AZD-2207
CAS:AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.Formula:C25H25Cl2F3N4O4SColor and Shape:SolidMolecular weight:605.46Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Formula:C21H30O2Color and Shape:SolidMolecular weight:314.46CB1 inverse agonist 2
CAS:CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.Formula:C24H20ClFN2OSColor and Shape:SolidMolecular weight:438.94GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39AM-6538
CAS:AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.Formula:C26H25Cl2N5O4Color and Shape:SolidMolecular weight:542.41COR 170
CAS:inverse agonist of CB2 receptorsFormula:C31H36N2O2Purity:98%Color and Shape:SolidMolecular weight:468.63NIDA 41020
CAS:NIDA 41020 is a CB1 receptor antagonist.Formula:C23H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:459.37LH 21
CAS:LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.Formula:C20H20Cl3N3Color and Shape:SolidMolecular weight:408.75CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purity:98%Color and Shape:SolidMolecular weight:481.59O-2093
CAS:anandamide uptake inhibitorFormula:C34H43Cl2NO3Purity:98%Color and Shape:SolidMolecular weight:584.62CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Formula:C23H18FN5O2S2Color and Shape:SolidMolecular weight:479.55CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Formula:C24H23Cl2N3OColor and Shape:SolidMolecular weight:440.36TC-C 14G
CAS:CB1 receptor inverse agonistFormula:C24H17Cl2F2NO4Purity:98%Color and Shape:SolidMolecular weight:492.3(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4Olorinab
CAS:Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Formula:C18H23N5O3Purity:97.67% - 98.47%Color and Shape:SolidMolecular weight:357.41CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Formula:C24H24N2O5SPurity:98.56%Color and Shape:SolidMolecular weight:452.52SR144528
CAS:SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).Formula:C29H34ClN3OPurity:99.63%Color and Shape:SolidMolecular weight:476.05Nonabine
CAS:Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Formula:C25H33NO2Purity:99.82% - 99.94%Color and Shape:SolidMolecular weight:379.54CB1R antagonist 1
CAS:CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Formula:C18H23F3N2O3SPurity:99.65%Color and Shape:SolidMolecular weight:404.45CB2R PAM
CAS:CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in neuropathic pain relief.Formula:C21H24BrFN2O2Purity:99.09%Color and Shape:SolidMolecular weight:435.33SCH-336
CAS:SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.
Formula:C23H25NO8S3Purity:95.01%Color and Shape:SolidMolecular weight:539.64PSB-CB5
CAS:PSB-CB5 (GPR18-IN-32)2 is a GRP18 antagonist with anti-inflammatory activity and can be used to study obesity and metabolic disorders.Formula:C20H17ClN2O2SPurity:99.26%Color and Shape:SolidMolecular weight:384.88AZD1940
CAS:AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.Formula:C20H29F2N3O2SPurity:98.68%Color and Shape:SolidMolecular weight:413.52Ref: TM-T30252
1mg130.00€5mg311.00€10mg535.00€25mg847.00€50mg1,169.00€100mg1,586.00€1mL*10mM (DMSO)344.00€JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purity:99.93%Color and Shape:SolidMolecular weight:438.47Ref: TM-T19705
1mg52.00€5mg119.00€10mg177.00€25mg313.00€50mg465.00€100mg662.00€1mL*10mM (DMSO)142.00€AM-1235
CAS:AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.Formula:C24H21FN2O3Purity:99.92%Color and Shape:SolidMolecular weight:404.43O-2050
CAS:O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.Formula:C23H31NO4SPurity:98%Color and Shape:SolidMolecular weight:417.56Heptadecanoyl ethanolamide
CAS:Heptadecanoyl ethanolamide, an endogenous cannabinoid, serves as a synthetic analog of PEA, featuring an odd-numbered (17-carbon) fatty acid chain [1].Formula:C19H39NO2Color and Shape:SolidMolecular weight:313.52COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg38.00€5mg86.00€10mg123.00€25mg215.00€50mg299.00€100mg411.00€200mg560.00€1mL*10mM (DMSO)94.00€PF-03550096
CAS:PF-03550096, an orally active synthetic cannabinoid (CB), selectively binds to peripheral CB2 receptors with a Ki value of 7.9 nM, demonstrating analgesic activity [1].Formula:C19H28N4O4Color and Shape:SolidMolecular weight:376.45URB447
CAS:URB447, a peripherally restricted CB1 cannabinoid antagonist with IC50 values of 313 nM for rat CB1 receptor and 41 nM for human CB2 receptor, effectively reduces food intake and body weight gain in mice. It achieves these effects without penetrating the brain or antagonizing central CB1-dependent responses, making it a potential research tool for obesity studies [1].Formula:C25H21ClN2OColor and Shape:SolidMolecular weight:400.9Tedalinab
CAS:Tedalinab is an effective and selective cannabinoid receptor 2 agonist.Formula:C19H21F2N3OPurity:98%Color and Shape:SolidMolecular weight:345.39GW405833 hydrochloride
CAS:GW405833 hydrochloride, a potent and selective agonist of the cannabinoid-2 (CB2) receptor (EC 50 = 0.65 nM; maximum inhibition = 44.6%), exhibits significant antihyperalgesic effects in various rodent pain models [1] [2] [3].Formula:C23H25Cl3N2O3Color and Shape:SolidMolecular weight:483.822-Linoleoyl Glycerol
CAS:2-Arachidonoyl glycerol (2-AG), a natural endocannabinoid ligand for the CB1 receptor, was isolated from porcine brain and characterized. Its congener, 2-linoleoyl glycerol (2-LG), which has a linoleoyl group instead of an arachidonoyl group, also exists alongside 2-AG in vivo. While 2-LG exhibits low intrinsic activity, it enhances the activity of 2-AG and other endocannabinoids through an "entourage" effect, attributed to the inhibition of breakdown and reuptake pathways that typically decrease endocannabinoid levels post-release.Formula:C21H38O4Color and Shape:SolidMolecular weight:354.531GSK494581A
CAS:GSK494581A is a GPR55 agonist and glycine transporter subtype 1 inhibitor.Formula:C27H28F2N2O4SPurity:98%Color and Shape:SolidMolecular weight:514.58PF 514273
CAS:PF 514273 is a CB1 receptor antagonist.Formula:C21H17Cl2F2N3O2Purity:98%Color and Shape:SolidMolecular weight:452.28PSNCBAM-1
CAS:PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with hypophagic effects in vivo.Formula:C22H21ClN4OPurity:99.86%Color and Shape:SolidMolecular weight:392.88Hemopressin(rat) TFA
CAS:Hemopressin(rat) TFA, a nonapeptide from hemoglobin α1-chain, selectively inhibits CB1 receptors and reduces inflammatory pain.Formula:C55H78F3N13O14Color and Shape:SolidMolecular weight:1202.2811(Z),14(Z)-Eicosadienoic Acid Ethanolamide
CAS:11(Z),14(Z)-Eicosadienoic acid ethanolamide is an ethanolamide derivative of 11(Z),14(Z)-eicosadienoic acid.Formula:C22H41NO2Color and Shape:SolidMolecular weight:351.57SAD-448
CAS:SAD-448 is a cannabinoid receptor type 1 (CB1) agonist. SAD-448 controls spasticity via action on the peripheral nerve CB1 receptor.Formula:C24H28N4O8SColor and Shape:SolidMolecular weight:532.57O-2545 hydrochloride
CAS:O-2545 is a potent water-soluble central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptor agonist with Ki values of 1.5 and 0.32 nM, respectively. Typically, cannabinoid agonists are highly lipophilic and require solubilization through surfactant agents or binding to water miscible substances like albumin, Tween 80, or Emulphor for use. When dissolved in saline, O-2545 has shown high efficacy in mouse behavioral models, administered either intravenously or intracerebroventricularly.Formula:C26H36N2O2HClColor and Shape:SolidMolecular weight:445Tricosanoyl Ethanolamide
CAS:Tricosanoyl ethanolamide, a fatty N-acyl ethanolamine within the endocannabinoid family, has an ethanolamine metabolite whose significance remains to be established.Formula:C25H51NO2Color and Shape:SolidMolecular weight:397.688Isopropyl dodec-11-enylfluorophosphonate
CAS:Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibitsFormula:C15H30FO2PPurity:98%Color and Shape:SolidMolecular weight:292.37MCHB-1
CAS:MCHB-1, a potent agonist of the human cannabinoid 2 (CB2) receptor (EC50= 0.52 nM), demonstrates high selectivity for CB2 over CB1 (Kis = 3.7 and 110 nM, respectively), distinguishing itself from similar benzimidazole compounds that significantly alleviate peripheral pain while minimizing central nervous system side effects in mice.Formula:C28H37N3O2Color and Shape:SolidMolecular weight:447.623CB1 antagonist 1
CAS:CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, andFormula:C26H22Cl2N4Purity:98%Color and Shape:SolidMolecular weight:461.39Amauromine
CAS:Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.Formula:C32H36N4O2Color and Shape:SolidMolecular weight:508.65γ-Linolenoyl monoethanolamide
CAS:γ-Linolenoyl monoethanolamide, a fatty N-acyl ethanolamine, acts as an endocannabinoid [1] [2].Formula:C20H35NO2Color and Shape:SolidMolecular weight:321.505CB 65
CAS:CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of 3.3 and > 1000 nM for CB2 and CB1 receptors respectively.Formula:C22H28ClN3O3Purity:99.53%Color and Shape:SolidMolecular weight:417.93(R)-Monlunabant
CAS:(R)-Monlunabant ((R)-MRI-1891) serves as a CB1 receptor antagonist utilized in obesity and metabolic disease research [1].Formula:C26H22ClF3N6O3SPurity:98%Color and Shape:SolidMolecular weight:591CB1 inverse agonist 1
CAS:MRL-650 is an oral, selective CB1 agonist; IC50: CB1=7.5 nM, CB2=4100 nM; anorexigenic effects noted.Formula:C25H18Cl3N3O3Purity:99.92%Color and Shape:SolidMolecular weight:514.79Ref: TM-T10694
1mg50.00€5mg105.00€10mg155.00€25mg224.00€50mg314.00€100mg427.00€200mg577.00€1mL*10mM (DMSO)129.00€AM841
CAS:AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor.Formula:C26H39NO3SPurity:98%Color and Shape:SolidMolecular weight:445.66Prostaglandin E2-1-glyceryl ester
CAS:Prostaglandin E2-1-glyceryl ester, a member of the Prostaglandin Glycerol Ester family, serves as an endocannabinoid ligand targeting the CB1 receptor. This compound triggers a swift and transient surge in intracellular free calcium levels [1] [2].Formula:C23H38O7Color and Shape:SolidMolecular weight:426.55PSB-SB1202
CAS:PSB-SB1202 (Compound 21a), a phenyl coumarin compound, acts as a CB1/CB2 agonist. It demonstrates EC50 values of 56 and 14 nM and K i values of 32 and 49 nM for CB1 and CB2 receptors, respectively [1].Formula:C23H26O4Color and Shape:SolidMolecular weight:366.45CB2R-IN-1
CAS:CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).Formula:C23H27F3N4O6S3Purity:98%Color and Shape:SolidMolecular weight:608.67CB-25
CAS:CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in cancer cells, though not affecting hCB1-CHO cellsFormula:C25H41NO3Purity:98%Color and Shape:SolidMolecular weight:403.6CB-52
CAS:CB-52 acts as a neutral antagonist and ligand for the CB2 cannabinoid receptor [1].Formula:C26H43NO3Color and Shape:SolidMolecular weight:417.62OMDM-5
CAS:OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM).Formula:C26H44N2O3Purity:99.73%Color and Shape:SolidMolecular weight:432.64Ref: TM-T12306
1mg93.00€5mg177.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,071.00€1mL*10mM (DMSO)210.00€O-Arachidonoyl glycidol
CAS:O-Arachidonoyl glycidol (compound 1), a 2-arachidonoylglycerol (2-AG) analog, effectively inhibits the hydrolysis of cytosolic 2-oleoylglycerol (2-OG) with an IC50 value of 4.5 µM, and also blocks 2-OG and anandamide hydrolysis in membrane fractions with IC50 values of 19 µM and 12 µM, respectively [1].Formula:C23H36O3Color and Shape:SolidMolecular weight:360.53GSK-554418A
CAS:GSK-554418A, a novel azaindole CB(2) agonists, is used for the treatment of chronic pain. It is efficacious in the acute model and the chronic joint pain model.Formula:C19H19ClN4O2Color and Shape:SolidMolecular weight:370.83CAY10508
CAS:CAY10508 is a potent and selective inverse agonist for the central cannabinoid (CB1) receptor with therapeutic potential for treating obesity and drug dependence, lacking psychotropic effects. It exhibits a Ki value of 243 nM and an EC50 of 195 nM. At a concentration of 10 µM, CAY10508 displaces [3H]-CP-55,940 with 100% efficacy at the CB1 receptor and 35% at the peripheral cannabinoid (CB2) receptor. Its inverse agonist activity at the CB1 receptor was confirmed through a [35S]-GTPγS binding assay.Formula:C21H14Br2N2O2Color and Shape:SolidMolecular weight:486.2GP 1a
CAS:GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids skin healing, anti-inflammatory.
Formula:C23H22Cl2N4OPurity:99.79%Color and Shape:SolidMolecular weight:441.35GW 833972A
CAS:GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.
Formula:C18H14Cl2F3N5OPurity:99.93%Color and Shape:SoildMolecular weight:444.24Bzo-poxizid
CAS:Bzo-poxizid is a synthetic cannabinoid and a psychoactive substance.Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.40BAY 38-7271
CAS:BAY 38-7271: potent neuroprotective, selective CB1/CB2 agonist, Ki of 1.85 nM (CB1) & 5.96 nM (CB2).Formula:C20H21F3O5SPurity:98%Color and Shape:SolidMolecular weight:430.44AM8936
AM8936: potent CB1 agonist, EC50 rCB1=8.6nM/hCB1=1.4nM, Ki rat CB1=0.55nM; potential for CNS, metabolic, pain, glaucoma research.Formula:C25H33NO3Color and Shape:SolidMolecular weight:395.53CBR Agonist-2
CBR Agonist-2: CB1 receptor agonist, EC50 - 960 nM, Ki - 970 nM, useful for hCB1R-related disease research.Formula:C27H27FN4OColor and Shape:SolidMolecular weight:442.53PSB-KK1415
CAS:PSB-KK1415 is a selective agonist for the human orphan G protein-coupled receptor GPR18, with an EC50 of 19.1 nM.Formula:C24H23ClN6O2Molecular weight:462.93Cannabigerovarin
CAS:Cannabigerovarin (CBGV) is a compound categorized as a phytocannabinoid.Formula:C19H28O2Molecular weight:288.42Ac-Atovaquone
CAS:Ac-Atovaquone, an ester-acetylated derivative of atovaquone, acts as a potent inhibitor of cytochrome bc1 (cytochrome bc1). This compound shows potential for use in malaria research.Formula:C24H21ClO4Color and Shape:SolidMolecular weight:408.87CBR Agonist-1
CBR Agonist-1 targets CB1R and CB2R with Ki of 0.18 μM and 1.22 μM, useful for studying cannabinoid-related diseases.Formula:C27H27FN4OColor and Shape:SolidMolecular weight:442.53
