Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
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AM-1235
CAS:335161-27-8
AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.
Formula:
C24H21FN2O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
404.43
Ref: TM-T29930
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
CB2R PAM
CAS:2244579-87-9
CB2R PAM, an oral drug, boosts CB2 receptor response to specific agonists, showing potential in …
Formula:
C21H24BrFN2O2
Purity:
98.17%
Color and Shape:
Liquid
Molecular weight:
435.33
Ref: TM-T37075
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 280.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 627.00 € | ||
| 500mg | 1,311.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Olorinab
CAS:1268881-20-4
Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor …
Formula:
C18H23N5O3
Purity:
97.13% - 97.67%
Color and Shape:
Solid
Molecular weight:
357.41
Ref: TM-T14302
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
OMDM-6
CAS:616884-67-4
OMDM-6 is a dual agonist of TRPV1(EC50 = 75 nM) and CB1 (Ki = 3.2 …
Formula:
C28H42N2O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
454.64
Ref: TM-T12307
| 1mg | 115.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 200mg | 1,444.00 € | ||
| 1mL*10mM (DMSO) | 283.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
(R)-Monlunabant
CAS:2765579-76-6
(R)-Monlunabant ((R)-MRI-1891) serves as a CB1 receptor antagonist utilized in obesity and metabolic disease research …
Formula:
C26H22ClF3N6O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
591
Ref: TM-T83533
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Jun 2025
Tedalinab
CAS:916591-01-0
Tedalinab is an effective and selective cannabinoid receptor 2 agonist.
Formula:
C19H21F2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T17027
| 25mg | 1,084.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 2,242.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
PSNCBAM-1
CAS:877202-74-9
PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with …
Formula:
C22H21ClN4O
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
392.88
Ref: TM-T28468
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 625.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
COR659
CAS:544450-68-2
COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
Formula:
C16H16ClNO3S
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T36520
| 1mg | 52.00 € | ||
| 2mg | 75.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 178.00 € | ||
| 25mg | 324.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 620.00 € | ||
| 200mg | 843.00 € | ||
| 1mL*10mM (DMSO) | 128.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
Amauromine
CAS:88360-87-6
Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a …
Formula:
C32H36N4O2
Color and Shape:
Solid
Molecular weight:
508.65
Ref: TM-T36566
| 1mg | 520.00 € | ||
| 250µg | 188.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
CB 65
CAS:913534-05-1
CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of …
Formula:
C22H28ClN3O3
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
417.93
Ref: TM-T41230
| 1mg | 64.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 335.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 710.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
GW 833972A
CAS:1092502-33-4
GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.
Formula:
C18H14Cl2F3N5O
Purity:
99.93%
Color and Shape:
Soild
Molecular weight:
444.24
Ref: TM-T64394
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € | ||
| 1mL*10mM (DMSO) | 944.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
AM841
CAS:871978-21-1
AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus …
Formula:
C26H39NO3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
445.66
Ref: TM-T78949
| 5mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 16 Jun 2025
CB-25
CAS:869376-63-6
CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in …
Formula:
C25H41NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
403.6
Ref: TM-T78083
| 2mg | 96.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
AEF0117
CAS:1610878-71-1
AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used …
Formula:
C29H40O3
Purity:
99.58%
Color and Shape:
Liquid
Molecular weight:
436.63
Ref: TM-T79909
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,093.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
OMDM-5
CAS:616884-66-3
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing …
Formula:
C26H44N2O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
432.64
Ref: TM-T12306
| 1mg | 87.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 284.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 867.00 € | ||
| 200mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 221.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
GP 1a
CAS:511532-96-0
GP 1a: potent CB2 receptor agonist (EC50=7.1), 30x CB2 over CB1 preference, boosts P-ERK1/2, aids …
Formula:
C23H22Cl2N4O
Purity:
99.44%
Color and Shape:
Liquid
Molecular weight:
441.35
Ref: TM-T41231
| 1mg | 56.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 341.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 722.00 € | ||
| 500mg | 1,454.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
CB1 antagonist 1
CAS:890037-68-0
CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and …
Formula:
C26H22Cl2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.39
Ref: TM-T10510
| 25mg | 2,015.00 € | ||
| 50mg | 2,642.00 € | ||
| 100mg | 3,515.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
CB1 inverse agonist 1
CAS:852315-00-5
MRL-650 is an oral, selective CB1 agonist; IC50: CB1=7.5 nM, CB2=4100 nM; anorexigenic effects noted.
Formula:
C25H18Cl3N3O3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
514.79
Ref: TM-T10694
| 1mg | 77.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 645.00 € | ||
| 200mg | 869.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Monday 16 Jun 2025
MDA77
CAS:1103774-21-5
MDA77 is a CB2 agonist with an EC50 value of 5.82 nM and exhibits no …
Formula:
C21H23N3O3
Color and Shape:
Liquid
Molecular weight:
365.43
Ref: TM-T201417
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 14 Jul 2025
Taranabant
CAS:701977-09-5
Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.
Formula:
C27H25ClF3N3O2
Purity:
99.06% - 99.06%
Color and Shape:
Solid
Molecular weight:
515.96
Ref: TM-T13080L
| 1mg | 98.00 € |
Estimated delivery in United States, on Monday 14 Jul 2025
