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HIV Protease

HIV Protease

HIV Protease inhibitors are a class of antiretroviral drugs that specifically target the protease enzyme of the Human Immunodeficiency Virus (HIV). By inhibiting this enzyme, these compounds prevent the virus from processing its polyproteins into mature, functional proteins, thereby blocking the production of new infectious virions. HIV Protease inhibitors are a cornerstone of highly active antiretroviral therapy (HAART) used to manage HIV/AIDS. At CymitQuimica, we provide a variety of HIV Protease inhibitors to support your research in HIV treatment, drug resistance, and virology.

Found 474 products of "HIV Protease"

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  • CymitQuimica logo
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    HIV-1 protease-IN-7

    CAS:
    HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].
    Formula:C68H104N10O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1285.68

    Ref: TM-T74942

  • HIV-1 protease-IN-12
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    HIV-1 protease-IN-12

    CAS:
    <p>HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-</p>
    Formula:C25H35N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.63

    Ref: TM-T79537

  • HIV-1 inhibitor-3
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    HIV-1 inhibitor-3

    CAS:
    HIV-1 inhibitor-3 is an HIV infection inhibitor.
    Formula:C9H10F2N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.18

    Ref: TM-T11564

  • HIV-1 protease-IN-9
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    HIV-1 protease-IN-9

    CAS:
    HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a
    Formula:C37H41N7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:679.83

    Ref: TM-T79295

  • NNRTIs-IN-1
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    NNRTIs-IN-1

    CAS:
    <p>NNRTIs-IN-1 is a potent non-nucleoside reverse transcriptase inhibitor (NNRTI) with notable anti-resistance efficacy, effectively inhibiting both the wild-type</p>
    Formula:C28H22N6O3
    Color and Shape:Solid
    Molecular weight:490.51

    Ref: TM-T78948

  • L 687908
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    L 687908

    CAS:
    L 687908 is a potent inhibitor of hydroxyethylene-containing HIV protease.
    Formula:C40H51N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:681.86

    Ref: TM-T24336

  • HIV-IN-8
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    HIV-IN-8

    CAS:
    HIV-IN-8 (Compound 9) acts as an HIV inhibitor, suppressing HIV replication with an effective concentration (EC50) of 13 μg/mL [1].
    Formula:C36H30O16
    Color and Shape:Solid
    Molecular weight:718.61

    Ref: TM-T79974

  • PNU-103017
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    PNU-103017

    CAS:
    PNU-103017 is an inhibitor of HIV protease.
    Formula:C28H28N2O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:504.6

    Ref: TM-T16555

  • DGKα-IN-8
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    DGKα-IN-8

    CAS:
    DGKα-IN-8 (Example 51) is a potent diacylglycerol kinase alpha (DGKα) inhibitor, exhibiting an IC50 of 22.491 nM and an EC50 of 0.256 nM.
    Formula:C23H19ClF3N5O
    Color and Shape:Solid
    Molecular weight:473.88

    Ref: TM-T79828

  • Azt-pmap
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    Azt-pmap

    CAS:
    <p>AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].</p>
    Formula:C20H25N6O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.42

    Ref: TM-T14488

  • R 87366
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    R 87366

    CAS:
    R 87366 is used as a water-soluble HIV protease inhibitor.
    Formula:C32H39N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.7

    Ref: TM-T26024

  • Berlopentin
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    Berlopentin

    CAS:
    <p>Berlopentin is splenopentin analog used to treat HIV-positive patients. It also has immunostimulatory properties.</p>
    Formula:C35H55N9O11
    Color and Shape:Solid
    Molecular weight:777.86

    Ref: TM-T23785

  • Capravirine
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    Capravirine

    CAS:
    Capravirine, a non-nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
    Formula:C20H20Cl2N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451.37

    Ref: TM-T26946

  • L 694746
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    L 694746

    CAS:
    L 694746 is an inhibitor of HIV-1 protease.
    Formula:C35H42N2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:618.72

    Ref: TM-T24343

  • L-697661
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    L-697661

    CAS:
    L-697661, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.
    Formula:C16H15Cl2N3O2
    Color and Shape:Solid
    Molecular weight:352.22

    Ref: TM-T27770

  • I-XW-053
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    I-XW-053

    CAS:
    <p>I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-</p>
    Formula:C22H16N2O2
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:340.37

    Ref: TM-T20000

  • KNI-272
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    KNI-272

    CAS:
    <p>Kynostatin-272 is a HIV protease inhibitor. KNI-272 blocked the maturation of viral particles.</p>
    Formula:C33H41N5O6S2
    Color and Shape:Solid
    Molecular weight:667.84

    Ref: TM-T27737

  • Indinavir, threo-
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    Indinavir, threo-

    CAS:
    Indinavir, threo- is a protease inhibitor utilized as a component of highly active antiretroviral treatment to HIV/AIDS.
    Formula:C36H47N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:613.79

    Ref: TM-T25535

  • DMP 323
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    DMP 323

    CAS:
    DMP 323 is a potent inhibitor of HIV-1 protease.
    Formula:C35H38N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:566.69

    Ref: TM-T24008

  • A 74704
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    A 74704

    CAS:
    A 74704 is a pseudo C2-symmetric inhibitor of HIV-1 protease and its diester analog.
    Formula:C43H52N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:736.9

    Ref: TM-T26440

  • Ulonivirine
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    Ulonivirine

    CAS:
    Ulonivirine is an orally active non-nucleoside reverse transcriptase inhibitor that exhibits high antiviral activity and can be used to study HIV-1 infection.
    Formula:C18H8ClF6N5O3
    Color and Shape:Solid
    Molecular weight:491.73

    Ref: TM-T63308

  • Droxinavir HCl
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    Droxinavir HCl

    CAS:
    Droxinavir HCl is an antiviral agent and HIV protease inhibitor.
    Formula:C29H52ClN5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:570.22

    Ref: TM-T25352

  • PDDC inhibitor
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    PDDC inhibitor

    CAS:
    PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.
    Formula:C27H29N5O4
    Purity:96.09% - 99.39%
    Color and Shape:Solid
    Molecular weight:487.55

    Ref: TM-T69757

  • HIV-1 inhibitor-54
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    HIV-1 inhibitor-54

    CAS:
    HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.
    Formula:C27H30N6O4S
    Purity:98.05% - 99.39%
    Color and Shape:Soild
    Molecular weight:534.63

    Ref: TM-T67833

  • Saphenamycin
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    Saphenamycin

    CAS:
    <p>Saphenamycin is an antibiotic from a strain of Streptomyces.</p>
    Formula:C23H18N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.40

    Ref: TM-T26176

  • Emtricitabine triphosphate
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    Emtricitabine triphosphate

    CAS:
    Emtricitabine triphosphate is an active metabolite of Emtricitabine, a drug for HIV/HBV that inhibits reverse transcriptase.
    Formula:C8H13FN3O12P3S
    Color and Shape:Solid
    Molecular weight:487.19

    Ref: TM-T70596

  • BI-2540
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    BI-2540

    CAS:
    <p>BI-2540 is a HIV non-nucleoside reverse transcriptase ( NNRT ) inhibitor .</p>
    Formula:C24H15ClF5NO5
    Color and Shape:Solid
    Molecular weight:527.83

    Ref: TM-T73435

  • Lamivudine, (+/-)-trans-
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    Lamivudine, (+/-)-trans-

    CAS:
    <p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>
    Formula:C8H11N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:229.26

    Ref: TM-T25609

  • Lentiginosine
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    Lentiginosine

    CAS:
    Lentiginosine is a selective amyloglucosidase inhibitor.
    Formula:C8H15NO2
    Color and Shape:Solid
    Molecular weight:157.21

    Ref: TM-T25662

  • HIV-1 inhibitor-52
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    HIV-1 inhibitor-52

    CAS:
    HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.
    Formula:C46H72FNO5S
    Color and Shape:Solid
    Molecular weight:770.13

    Ref: TM-T72565

  • GS-9822
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    GS-9822

    CAS:
    <p>GS-9822 is a new LEDGIN inhibitor targeting LEDGF/p75 to alter HIV integration, showing a block-and-lock effect in cells.</p>
    Formula:C36H39ClN4O4S
    Color and Shape:Solid
    Molecular weight:659.24

    Ref: TM-T69782

  • Methyl piperazine-2-carboxylate
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    Methyl piperazine-2-carboxylate

    CAS:
    Methyl piperazine-2-carboxylate (compound 4) is a potent activator of METTL3/METTL14/WTAP. It enhances the production of HIV-1p24 viral particles and increases the level of N6-methyladenosine in the viral RNA genome.
    Formula:C6H12N2O2
    Color and Shape:Solid
    Molecular weight:144.172

    Ref: TM-T204361

  • A 76889
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    A 76889

    CAS:
    A 76889 is an inhibitor of HIV-1 protease.
    Formula:C44H58N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:794.98

    Ref: TM-T26445

  • ATPase-IN-6
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    ATPase-IN-6

    CAS:
    ATPase-IN-6 is an inhibitor of H+/K+-ATPase (ATPase) and a derivative of imidazopyridine. It exhibits significant antiviral activity against various viruses, such as HIV-1 and SARS-CoV-2. ATPase-IN-6 is applicable in antiviral infection research.
    Formula:C29H25N3O4S
    Color and Shape:Solid
    Molecular weight:511.59

    Ref: TM-T211132

  • NBD-14189
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    NBD-14189

    CAS:
    NBD-14189: Potent HIV-1 entry blocker, binds gp120, IC50: 89 nM, strong antiviral (EC50 <200 nM).
    Formula:C18H16F4N4O2S
    Color and Shape:Solid
    Molecular weight:428.40

    Ref: TM-T62340

  • BRN3OMe
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    BRN3OMe

    CAS:
    <p>BRN3OMe is an effective inhibitor of HIV-1 reverse transcriptase (HIV-1 reverse transcriptase), showing potential for antiviral drug research.</p>
    Formula:C7H13N3O4
    Color and Shape:Solid
    Molecular weight:203.196

    Ref: TM-T204926

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    HIV-1 inhibitor-44

    HIV-1 inhibitor-44 (compound 11l) is an HIV-1 reverse transcriptase inhibitor that exhibits activity against wild-type HIV-1 strains (EC50: 0.209 μM).
    Formula:C23H26N2O4S
    Color and Shape:Solid
    Molecular weight:426.53

    Ref: TM-T62319

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    HIV-1 inhibitor-17

    HIV-1 inhibitor-18 blocks HIV-1 capsid, acts on NL4-3 strain (EC50: 2.57 μM), has low cytotoxicity (MT-4 CC50: >8.55).
    Formula:C32H32N4O5S
    Color and Shape:Solid
    Molecular weight:584.69

    Ref: TM-T64131

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    HIV-1 inhibitor-40

    HIV-1 inhibitor-40 (4ab) is a potent NNRTI (EC50: 1.9 nM), non-toxic in vivo, and a sensitive CYP inhibitor.
    Formula:C25H18N6O2
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T62452

  • HIV-1-IN-86
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    HIV-1-IN-86

    CAS:
    HIV-1-IN-86 (compound 6m) is an HIV-1 inhibitor with an EC50 of 0.77 μM, exhibiting antiviral activity.
    Formula:C20H17N3O7S
    Color and Shape:Solid
    Molecular weight:443.43

    Ref: TM-T212486

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    HIV-1 protease-IN-6

    HIV-1 protease-IN-6 (17d) strongly inhibits HIV-1 protease (IC50: 21 pM, Ki: 4.7 pM) and effectively targets DRV-resistant mutants.
    Formula:C27H31FN2O6S
    Color and Shape:Solid
    Molecular weight:530.61

    Ref: TM-T63733

  • Fipravirimat
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    Fipravirimat

    CAS:
    Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.
    Formula:C43H67FN2O4S
    Color and Shape:Solid
    Molecular weight:727.07

    Ref: TM-T70147

  • BMIM-TFSI
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    BMIM-TFSI

    CAS:
    <p>BMIM-TFSI (compound8) is an HIV-1 integrase inhibitor that effectively suppresses both the 3'-processing (3'-P) and strand transfer (ST) steps of the integration process. It is applicable in HIV-1 research.</p>
    Formula:C10H15F6N3O4S2
    Color and Shape:Solid
    Molecular weight:419.364

    Ref: TM-T204101

  • BI 224436
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    BI 224436

    CAS:
    <p>BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.</p>
    Formula:C27H26N2O4
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T14559

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    HIV-IN-3

    <p>HIV-IN-3 (Compound 22a) is a potent inhibitor of HIV (IC50: 1.5 μM). HIV-IN-3 has potential for the study of HIV-related diseases.</p>
    Formula:C21H32ClN7O3
    Color and Shape:Solid
    Molecular weight:465.98

    Ref: TM-T62978

  • Integrase-LEDGF/p75 allosteric inhibitor 1
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    Integrase-LEDGF/p75 allosteric inhibitor 1

    CAS:
    <p>Oral HIV-1 allosteric integrase inhibitor, blocks DNA integration, antiviral, potent against NL432 (EC50: 3.9 nM).</p>
    Formula:C33H41NO6S
    Color and Shape:Solid
    Molecular weight:579.75

    Ref: TM-T64096

  • L 702007
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    L 702007

    CAS:
    <p>L 702007 is an inhibitor of HIV-1 reverse transcriptase.</p>
    Formula:C18H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.41

    Ref: TM-T24346

  • HIV-1 inhibitor-61
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    HIV-1 inhibitor-61

    CAS:
    HIV-1 Inhibitor-61 (2c) serves as a potent inhibitor of HIV-1 reverse transcriptase, exhibiting an EC50 value of 0.07 nM in NL4-3 wt MT-4 cells [1].
    Formula:C24H24F2N2O2S
    Color and Shape:Solid
    Molecular weight:442.52

    Ref: TM-T86580

  • Desthiazolylmethyl ritonavir
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    Desthiazolylmethyl ritonavir

    CAS:
    <p>Desthiazolylmethyl ritonavir is an alkaline-catalyzed degradation product of the HIV protease inhibitor Ritonavir.</p>
    Formula:C33H43N5O4S
    Color and Shape:Solid
    Molecular weight:605.791

    Ref: TM-T204277

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    HIV-1 inhibitor-8

    HIV-1 inhibitor-8: potent oral NNRTI, low toxicity, IC50: 0.081 μM, effective on multiple strains, EC50: 4.44-54.5 nM.
    Formula:C25H21N5OS
    Color and Shape:Solid
    Molecular weight:439.53

    Ref: TM-T62526

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    HIV-1 inhibitor-14

    <p>HIV-1 inhibitor-14: potent, broad HIV-1 RT inhibitor. IC50=0.14μM. Effective against wild-type and resistant strains, EC50=5.79-28.3nM.</p>
    Formula:C29H32N6O4S
    Color and Shape:Solid
    Molecular weight:560.67

    Ref: TM-T63963

  • ZK-316
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    ZK-316

    CAS:
    ZK-316 is a potent and broad-spectrum NNRTI inhibitor with an EC50 range of 0.99 to 75.1 nM. It is applicable for HIV research.
    Formula:C27H22D6N6O3S2
    Color and Shape:Solid
    Molecular weight:554.72

    Ref: TM-T207116

  • (S)-Batylalcohol
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    (S)-Batylalcohol

    CAS:
    <p>(S)-Batylalcohol (1-O-Octadecyl-sn-glycerol) is an analogue of phosphonoformic acid (PFA) and demonstrates higher in vitro antiviral activity against human immunodeficiency virus type 1 (HIV-1) compared to PFA. This compound is applicable in antiretroviral research.</p>
    Formula:C21H44O3
    Color and Shape:Solid
    Molecular weight:344.572

    Ref: TM-T204561

  • PD 134922
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    PD 134922

    CAS:
    PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.
    Formula:C37H61N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:719.97

    Ref: TM-T28329

  • MIV-150
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    MIV-150

    CAS:
    MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).
    Formula:C19H17FN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.36

    Ref: TM-T16081

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    HIV-1 inhibitor-41

    <p>HIV-1 inhibitor-41 (B23): Oral non-nucleoside reverse transcriptase blocker, EC50 of 50 nM (E138K), 20.8 nM (WT), low hERG/CYP impact, non-toxic.</p>
    Formula:C16H15F2N3OS
    Color and Shape:Solid
    Molecular weight:335.37

    Ref: TM-T61031

  • 4'-Ethynyl-2'-deoxyadenosine
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    4'-Ethynyl-2'-deoxyadenosine

    CAS:
    4'-E-dA is a potent nucleoside RT inhibitor for drug-resistant HIV (EC50: 98 nM in MT-4 cells).
    Formula:C12H13N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:275.26

    Ref: TM-T10141

  • DPC 684
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    DPC 684

    CAS:
    DPC 684 is a potent and selective HIV-1 protease inhibitor with an IC90 of 5.7-40 nM and a Ki of 0.021 nM. It competitively inhibits HIV-1 protease, preventing viral polyprotein cleavage. Compared to cellular proteases, DPC 684 shows high selectivity for retroviral proteases. The compound exhibits low protein binding and offers broad-spectrum inhibition against various wild-type and mutant HIV-1 proteases, with an IC90 of 1.9-6.3 nM. DPC 684 is significant for HIV research.
    Formula:C35H48FN5O5S
    Color and Shape:Solid
    Molecular weight:669.85

    Ref: TM-T211711

  • BRD-K98645985
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    BRD-K98645985

    CAS:
    BRD-K98645985: BAF inhibitor, binds ARID1A, reverses HIV-1 latency, EC50 ~2.37μM, alters nucleosome placement.
    Formula:C33H43N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.73

    Ref: TM-T10605

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    ZLM-66

    <p>ZLM-66: Doravirine analog, HIV-1 NNRTI inhibitor, IC50: 41nM, EC50: HIV-1 13nM, cIAP1 0.32nM; useful in AIDS research.</p>
    Color and Shape:Solid

    Ref: TM-T64303

  • GSK3739936
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    GSK3739936

    CAS:
    <p>GSK3739936 inhibits HIV-1 integrase (IC50: 11.1 nM, EC50: 1.7 nM), weak on CYP (IC50 &gt;24.3 μM), rapid absorption, moderate clearance, high oral availability.</p>
    Formula:C34H43FN2O4
    Color and Shape:Solid
    Molecular weight:562.71

    Ref: TM-T63977

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    HIV-1 inhibitor-18

    <p>HIV-1 inhibitor-18 blocks HIV-1 capsid, effective on NL4-3 strain (EC50: 5.14 μM), slightly toxic (MT-4CC50&gt;9.51).</p>
    Formula:C27H31N3O6S
    Color and Shape:Solid
    Molecular weight:525.62

    Ref: TM-T63687

  • Telinavir
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    Telinavir

    CAS:
    Telinavir (SC-52151) is a potent and selective inhibitor of HIV protease. It effectively inhibits both HIV-1 and HIV-2, as well as lymphotropic, monocytotropic strains, and wild isolates of simian immunodeficiency viruses, with an EC50 of 26 ng/mL (43 nM). Telinavir shows high protein binding in human plasma and a low distribution rate in red blood cells.
    Formula:C33H44N6O5
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T207029

  • BMS-818251
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    BMS-818251

    CAS:
    BMS-818251 is a potent small-molecule inhibitor that targets HIV-1 entry, with an EC50 value of 0.019 nM. It exhibits over 10 times greater efficacy on the cross-subtype panels of the 208-HIV-1 strain compared to BMS-626529. BMS-818251 enhances potency through interactions with gp120 residues in the conserved β20-β21 hairpin.
    Formula:C29H26N6O5S
    Color and Shape:Solid
    Molecular weight:570.619

    Ref: TM-T204307

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    HIV-1 inhibitor-13

    <p>HIV-1 inhibitor-13: oral NNRTI, IC50=0.14μM for HIV-1 RT, effective on resistant strains (EC50=2.85-18nM).</p>
    Formula:C30H32N6O3
    Color and Shape:Solid
    Molecular weight:524.61

    Ref: TM-T63677

  • L-697639
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    L-697639

    CAS:
    L-697639 inhibits of HIV-1 reverse transcriptase and HIV-1 replication.
    Formula:C18H21N3O2
    Color and Shape:Solid
    Molecular weight:311.38

    Ref: TM-T27769

  • Gardiquimod hydrochloride
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    Gardiquimod hydrochloride

    CAS:
    Gardiquimod (hydrochloride) is an imidazoquinoline class TLR7/8 agonist. It can inhibit HIV-1 infection in macrophages and activated peripheral blood mononuclear cells (PBMCs). At concentrations below 10 μM, Gardiquimod (hydrochloride) specifically activates TLR7.
    Formula:C17H24ClN5O
    Color and Shape:Solid
    Molecular weight:349.858

    Ref: TM-T204751

  • NBD-10007
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    NBD-10007

    CAS:
    NBD-10007 is an inhibitor of HIV-1 entry.
    Formula:C20H25ClN4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.96

    Ref: TM-T24522

  • Cyclotriazadisulfonamide
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    Cyclotriazadisulfonamide

    CAS:
    <p>Cyclotriazadisulfonamide (CADA) is a specific inhibitor of HIV entry that targets CD4 by preventing the co-translational translocation of human CD4 (huCD4) into the endoplasmic reticulum (ER) lumen through a signal peptide (SP)-dependent mechanism.</p>
    Formula:C31H39N3O4S2
    Color and Shape:Solid
    Molecular weight:581.79

    Ref: TM-T39264

    ne
    Discontinued
    Discontinued product
  • Aurothioglucose
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    Aurothioglucose

    CAS:
    <p>Aurothioglucose is a active-site TrxR1 inhibitor.</p>
    Formula:C6H11AuO5S
    Purity:98%
    Color and Shape:Yellow Crystals Solid
    Molecular weight:392.18

    Ref: TM-T14351

    100mg
    Discontinued
    Discontinued product
  • 3-Deazaadenosine
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    3-Deazaadenosine

    CAS:
    3-Deazaadenosine, an inhibitor of S-adenosylhomocysteine hydrolase with a Ki of 3.9 μM, exhibits anti-inflammatory, anti-proliferative, and anti-HIV activity.
    Formula:C11H14N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:266.25

    Ref: TM-T10111L

    5mg
    Discontinued
    Discontinued product
  • BMS-378806
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    BMS-378806

    <p>BMS-378806 is an HIV inhibitor with EC50: 0.85-26.5nM for various strains.</p>
    Formula:C22H22N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.43

    Ref: TM-T22609

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product
  • Oxindole
    Targetmol
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    Oxindole

    CAS:
    <p>Oxindole (Indolin-2-one) is an aromatic heterocyclic building block. 2-indolinone derivatives have become lead compounds in the research of kinase inhibitors.Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic target for anti-cancer drug development.</p>
    Formula:C8H7NO
    Purity:99.34%
    Color and Shape:Off-White Crystalline Powder
    Molecular weight:133.15

    Ref: TM-FR16741

    1g
    Discontinued
    5g
    Discontinued
    10g
    Discontinued
    Discontinued product
  • HIV-1 integrase inhibitor
    Targetmol
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    HIV-1 integrase inhibitor

    CAS:
    Hiv-1 integrase inhibitor is an effective anti-HIV drug.
    Formula:C11H9N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.21

    Ref: TM-T11566

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product