Other Inhibitors
This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.
Found 37926 products of "Other Inhibitors"
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Croconic acid disodium
CAS:<p>Croconic acid (disodium) (Nacr) enhances gene expression related to lysine crotonylation (Kcr) modification, which promotes cell growth and proliferation. This compound also shows promise in boosting somatic cell nuclear transfer (SCNT) efficiency and optimizing research in cell culture conditions.</p>Formula:C5Na2O5Color and Shape:SolidMolecular weight:186.03Netobimin
CAS:<p>Netobimin is an anthelmintic effective against naturally acquired gastrointestinal nematodes in cows.</p>Formula:C14H20N4O7S2Color and Shape:SolidMolecular weight:420.46Dimesna free acid
CAS:<p>Dimesna (BNP-778), when used in conjunction with active cancer chemotherapy agents, can reduce the toxicity associated with uremia.</p>Formula:C4H10O6S4Color and Shape:SolidMolecular weight:282.38MPO-IN-8
CAS:<p>MPO-IN-8, an orally active myeloperoxidase (MPO) inhibitor, effectively inhibits the production of hypochlorous acid in neutrophils and the release of extracellular traps (NETosis). In mice exhibiting gouty arthritis, it reduces swelling, decreases peroxidase activity, and lowers IL-1β levels.</p>Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22Deacetylravidomycin N-oxide
CAS:<p>Deacetylravidomycin N-oxide is an antibiotic produced by [Streptomyces ravidus S50905] that exhibits activity against Gram-positive bacteria but is inactive against Gram-negative bacteria. Additionally, Deacetylravidomycin N-oxide demonstrates antitumor properties against P388 leukemia and methylcholanthrene A fibrosarcoma.</p>Formula:C31H33NO10Color and Shape:SolidMolecular weight:579.594TREX1-IN-2
CAS:<p>TREX1-IN-2 (Compound 15B) serves as an inhibitor of Human TREX1, displaying an IC 50 value of less than 1.00 μM. Additionally, this compound demonstrates anticancer activity in vivo.</p>Formula:C28H34Cl2N4O4Color and Shape:SolidMolecular weight:561.52-PPA
CAS:2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.Formula:C11H10N2Color and Shape:SolidMolecular weight:170.21Urease-IN-16
CAS:<p>Urease-IN-16, with an IC50 of 132 µmol/L, is a urease inhibitor that coordinates with nickel atoms through the oxygen atoms of either carbonyl or boronic acid groups. This compound holds significant potential as an additive in the development of efficient fertilizers and medical applications.</p>Formula:C14H17BN2O4SColor and Shape:SolidMolecular weight:320.17Calphostin I
CAS:<p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>Formula:C44H38O15Color and Shape:SolidMolecular weight:806.76ETH 157
CAS:<p>ETH 157 is a synthetic neutral carrier-based Na+ selective microelectrode, with sufficient selectivity against K+, Ca2+, and Mg2+ for extracellular measurement of Na+ activity.</p>Formula:C36H32N2O4Color and Shape:SolidMolecular weight:556.65Fipronil desulfinyl
CAS:<p>Fipronil desulfinyl, a photodegradation product of the insecticide Fipronil, exhibits similar in vivo toxicity to Fipronil and possesses higher environmental toxicity.</p>Formula:C12H4Cl2F6N4Color and Shape:SolidMolecular weight:389.08GK241
CAS:<p>GK241 (compound 31a-c), a 2-oxoamide-based compound, exhibits inhibitory activity against group IIA secretory phospholipase A2 (GIIA sPLA2) in humans and mice, with IC50 values of 143 nM and 68 nM, respectively. The mechanism of inhibition has been explored through molecular dynamics simulations.</p>Formula:C21H39NO4Color and Shape:SolidMolecular weight:369.54Falecalcitriol
CAS:<p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>Formula:C27H38F6O3Purity:98%Color and Shape:SolidMolecular weight:524.58Cyclo (D-Pro-L-Val)
CAS:<p>Cyclo(D-Pro-L-Val) inhibits the activity of β-glucosidase (β-glycosidase) with an IC50 of 75 μg/mL and exhibits either no inhibitory effects or only weak inhibition on other glycosidases.</p>Formula:C10H16N2O2Color and Shape:SolidMolecular weight:196.246LPM4870108
<p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>Formula:C20H19FN6O3Color and Shape:SolidMolecular weight:410.4MRS2279
CAS:<p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>Formula:C13H18ClN5O8P2Purity:98%Color and Shape:SolidMolecular weight:469.71NA 0362
CAS:<p>NA 0362 is a derivative of SF 2370 that inhibits smooth muscle contraction.</p>Formula:C28H26N4O4Color and Shape:SolidMolecular weight:482.53Veonetinib
CAS:<p>Veonetinib (example 3) is an effective inhibitor of tyrosine kinase , exhibiting IC50 values of 0.1 μM and 0.4 μM in A549 cells and LOVO cells, respectively.</p>Formula:C27H28FN3O4Color and Shape:SolidMolecular weight:477.53GSK268
<p>GSK268 is a BET inhibitor.</p>Formula:C26H27N5O3Color and Shape:SolidMolecular weight:457.53BI-1388
CAS:<p>BI-1388 is a potent HCV NS3 protease inhibitor; halts replication across genotypes, including D168V/R155K mutants.</p>Formula:C41H53N7O9SColor and Shape:SolidMolecular weight:819.97Resolvin E2
CAS:<p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45SCP1-IN-1
CAS:<p>SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.</p>Formula:C20H19F3N2O7S2Purity:99.53%Color and Shape:SoildMolecular weight:520.5ART615
<p>ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).</p>Formula:C21H21F3N4O2Color and Shape:SolidMolecular weight:418.41CPX-351
CAS:<p>CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.</p>Formula:C36H42N4O15Purity:98.95% - 99.763%Color and Shape:SolidMolecular weight:770.74Tandutinib (MLN518) HCl
<p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>Formula:C31H43ClN6O4Purity:98%Color and Shape:SolidMolecular weight:599.16HYL001
CAS:<p>HYL001 (compound 338) is a potent inhibitor of the TGFβ receptor 1 (ALK5), exhibiting approximately nine times the efficacy of its structurally related counterpart, galunisertib, in eliminating liver metastasis tumors generated in mice.</p>Formula:C21H18N4OColor and Shape:SolidMolecular weight:342.39ONL-1204
CAS:<p>ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.</p>Formula:C71H100N18O16Color and Shape:SolidMolecular weight:1461.66ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Color and Shape:SolidRORγt inhibitor 2
CAS:<p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>Formula:C31H33F5N2O7SColor and Shape:SolidMolecular weight:672.66K-Ras-IN-4
CAS:<p>K-Ras-IN-4 (compound CP163) is an inhibitor of K-Ras.</p>Formula:C31H28F4N6O3SColor and Shape:SolidMolecular weight:640.65NSC-217913
CAS:<p>NSC-217913 acts as an inhibitor of WWP1, exhibiting an IC50 value of 158.3 μM.</p>Formula:C9H8Cl2N4O2SColor and Shape:SolidMolecular weight:307.16Hydroxyethyl disulfide
CAS:<p>Hydroxyethyl disulfide can counteract the inhibitory effects of showdomycin on methotrexate-resistant thymidylate synthase and is protected from deactivation by its substrate, deoxyuridine monophosphate, thus preserving the antibiotic's activity.</p>Formula:C4H10O2S2Color and Shape:SolidMolecular weight:154.25UNC7467
CAS:<p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>Formula:C20H13NO3Purity:98.28% - 98.64%Color and Shape:SoildMolecular weight:315.32Anti-TSWV agent 1
<p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>Formula:C22H27ClN4OS3Color and Shape:SolidMolecular weight:495.12Fosfocytocin
CAS:<p>Fosfocytocin can be found in the Pseudomonas fluorescens strain PK-52 and exhibits very weak antibacterial activity.</p>Formula:C12H20N4O13P2Color and Shape:SolidMolecular weight:490.254Domitroban
CAS:<p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>Formula:C20H27NO4SColor and Shape:SolidMolecular weight:377.5Nemotinic acid
CAS:<p>Nemotinic acid exhibits activity against Gram-positive bacteria, mycobacteria, and fungi, while also displaying weaker activity against Gram-negative bacteria.</p>Formula:C11H10O3Color and Shape:SolidMolecular weight:190.195Cryptosporiopsin
CAS:<p>Cryptosporiopsin can be isolated from strains of Cryptosporiopsis sp. and Sporormia affinis. It exhibits antimicrobial activity against various basidiomycetes, alga fungi, ascomycetes, and glaucomycetes responsible for wood decay. Additionally, it inhibits the germination of Phytophthora potatoes spores. Cryptosporiopsin also shows some activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C10H10Cl2O4Color and Shape:SolidMolecular weight:265.09Neomycin F
CAS:<p>Paromomycin II is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria, mycobacteria, and protozoa. It is particularly effective in treating amoebic dysentery and certain bacterial dysentery cases.</p>Formula:C23H45N5O14Color and Shape:SolidMolecular weight:615.628Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formula:C24H26N2O13Color and Shape:SolidMolecular weight:550.47Mevidalen HBA
CAS:<p>Mevidalen (LY3154207), a potent D1 positive allosteric modulator, is in clinical trials for Lewy body dementia.</p>Formula:C31H35Cl2NO6Color and Shape:SolidMolecular weight:588.52Iroxanadine hydrobromide
CAS:<p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>Formula:C14H21BrN4OColor and Shape:SolidMolecular weight:341.25ATM-3507 trihydrochloride (1861449-70-8 free base)
<p>ATM-3507 trihydrochloride is a potent tropomyosin inhibitor (IC50s: 3.83-6.84 μM in human melanoma cell lines).</p>Formula:C37H49Cl3FN5O2Purity:98%Color and Shape:SolidMolecular weight:721.17SLC7A11-IN-2
CAS:<p>SLC7A11-IN-2 (Compound 1) is an inhibitor of SLC7A11/xCT. It disrupts the oxidative balance in HeLa cells by decreasing intracellular glutathione levels and increasing oxidative stress, thereby inducing cell death with an IC50 of 10.23 μM. Molecular dynamics simulations have demonstrated that SLC7A11-IN-2 exhibits a stronger binding affinity to SLC7A11 compared to Erastin. This compound is useful for research in the field of cervical cancer.</p>Formula:C19H24N4O3Color and Shape:SolidMolecular weight:356.42PZ-3022
CAS:<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Formula:C20H21N5OColor and Shape:SolidMolecular weight:347.41Pyriftalid
CAS:<p>Pyriftalid is a novel insecticide known for its potent inhibitory activity against a variety of pests. It is widely utilized in agriculture to effectively manage crop pests, thereby enhancing both the yield and quality of crops. Additionally, research is exploring the use of Pyriftalid in boosting plant resistance to pests and diseases.</p>Formula:C15H14N2O4SColor and Shape:SolidMolecular weight:318.35Rivasterat
CAS:<p>Rivasterat is a cholesterol-derived steroid known for its anti-inflammatory properties.</p>Formula:C37H54O8Color and Shape:SolidMolecular weight:626.82XD23
CAS:<p>XD23 is a potent osteosarcoma inhibitor that functions by downregulating DKK1 and activating the WNT/β-catenin signaling pathway.</p>Formula:C22H26ClN7O3Color and Shape:SolidMolecular weight:471.94Allosucrose
CAS:<p>Allosucrose is a biochemical.</p>Formula:C12H22O11Color and Shape:SolidMolecular weight:342.30SHR902275
CAS:<p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>Formula:C26H23F3N4O4Color and Shape:SolidMolecular weight:512.48Cofpropamine
CAS:<p>Cofpropamine, a caffeine derivative that inhibits polyadenylation, enhances the suppressive effects of Cyclophosphamide in animal models of rat adjuvant arthritis and mouse collagen-induced arthritis.</p>Formula:C13H21N5O3Color and Shape:SolidMolecular weight:295.34LK-732
CAS:<p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>Formula:C25H29N5O3SColor and Shape:SolidMolecular weight:479.59Erizepine
CAS:<p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>Formula:C20H22N2Color and Shape:SolidMolecular weight:290.4Reumycin
CAS:<p>Reumycin is a 7-azaindole antibiotic that exhibits cytotoxicity against tumor cells such as Ellrich carcinoma, Sarcoma-180, Sarcoma-37, and lymphosarcoma.</p>Formula:C6H5N5O2Color and Shape:SolidMolecular weight:179.136DXR-IN-3
CAS:<p>DXR-IN-3 is an anti-Toxoplasma DXR inhibitor. It exhibits in vitro activity against the TgDXR enzyme, with an IC50 value of 0.62 μM and a Ki value of 0.19 μM. Furthermore, DXR-IN-3 can inhibit the proliferation of Toxoplasma, displaying an IC50 value of 5.46 μM.</p>Formula:C10H12Cl2NO5PSColor and Shape:SolidMolecular weight:360.15XN methyl pyrazole
<p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>Formula:C22H24N2O4Color and Shape:SolidMolecular weight:380.44PSMA-1007
CAS:<p>PSMA-1007 is a novel Glu-Ureido-type prostate-specific membrane antigen (PSMA) inhibitor.</p>Formula:C49H55FN8O16Color and Shape:SolidMolecular weight:1030.015-Hydroxy-4-oxo-L-norvaline
CAS:<p>5-Hydroxy-4-oxo-L-norvaline is an antifungal antibiotic that inhibits protein biosynthesis.</p>Formula:C5H9NO4Color and Shape:SolidMolecular weight:147.129Demethylblasticidin S
CAS:<p>Demethylblasticidin S is an antifungal antibiotic produced by Streptomyces griseochromogenes.</p>Formula:C16H24N8O5Color and Shape:SolidMolecular weight:408.412Flusoxolol
CAS:<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formula:C22H30FNO4Color and Shape:SolidMolecular weight:391.481-Deamino-1-hydroxygentamicin C2
CAS:<p>1-Deamino-1-hydroxygentamicin C2 (AntibioticSU-1) is an aminoglycoside antibiotic effective against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H40N4O8Color and Shape:SolidMolecular weight:464.554Citreamicin ξ
CAS:<p>Citreamicin ξ exhibits activity against both Gram-positive aerobic and anaerobic bacteria.</p>Formula:C30H25NO11Color and Shape:SolidMolecular weight:575.52JBIR-22
CAS:<p>JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.</p>Formula:C23H33NO6Color and Shape:SolidMolecular weight:419.51SOS1-IN-6
CAS:<p>SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).</p>Formula:C26H28F3N3O2Color and Shape:SolidMolecular weight:471.51Isohematinic acid
CAS:<p>Isohematinic acid exhibits mild activity against anaerobic bacteria.</p>Formula:C8H9NO4Color and Shape:SolidMolecular weight:183.161TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Color and Shape:SolidMolecular weight:548.52AMG-315
CAS:<p>AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.</p>Formula:C24H41NO2Color and Shape:SolidMolecular weight:375.59Antitumor agent-47
<p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>Formula:C30H27NO11Color and Shape:SolidMolecular weight:577.54Milbemycin β1
CAS:<p>Milbemycin β1 is a macrolide antibiotic with insecticidal properties effective against agricultural pests, aphids, larvae, and others.</p>Formula:C32H48O7Color and Shape:SolidMolecular weight:544.719Gentamicin A
CAS:<p>Gentamicin A is an antibiotic exhibiting effective antibacterial activity against both Gram-positive and Gram-negative bacteria, and it also demonstrates activity against most methicillin-sensitive staphylococci.</p>Formula:C18H36N4O10Color and Shape:SolidMolecular weight:468.499PD-149163
CAS:<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formula:C42H71N9O6Color and Shape:SolidMolecular weight:798.07Olanzapine/Samidorphan
CAS:<p>Olanzapine/Samidorphan, a tablet blending olanzapine and samidorphan, targets schizophrenia and bipolar I, curbing weight gain.</p>Formula:C38H46N6O4SColor and Shape:SolidMolecular weight:682.88Sapintoxin D
CAS:<p>Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.</p>Formula:C30H37NO8Color and Shape:SolidMolecular weight:539.62SSM3 TFA
CAS:<p>SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..</p>Formula:C22H32N12O2Color and Shape:SolidMolecular weight:496.57AM-3189
CAS:<p>AM-3189: potent, selective GPR40 agonist with low CNS penetration, good pharmacokinetics, and efficacy mirroring AMG 837.</p>Formula:C27H25ClN2O3Color and Shape:SolidMolecular weight:460.95LA-810
CAS:<p>LA-810 is a nitrous oxide donor.</p>Formula:C15H25N5O7SColor and Shape:SolidMolecular weight:419.45Heparastatin
CAS:<p>Heparastatin is an inhibitor of heparanase.</p>Formula:C8H11F3N2O5Purity:98%Color and Shape:SolidMolecular weight:272.18AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:460.01EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Color and Shape:SolidMolecular weight:475.54Cyclophellitol
CAS:<p>Cyclophellitol is an inhibitor of β-glycosidase, with an IC50 of 0.8 μg/mL.</p>Formula:C7H12O5Color and Shape:SolidMolecular weight:176.167BMS-748730
CAS:<p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>Formula:C22H26ClN7O3SColor and Shape:SolidMolecular weight:504.01Exicorilant
CAS:<p>Exicorilant is a selective oral GR antagonist (Ki: 7 nM) that may reduce obesity, glucose intolerance, & dyslipidemia.</p>Formula:C26H23F4N7O3SPurity:98%Color and Shape:SolidMolecular weight:589.56Cinatrin A
CAS:<p>Cinatrin A exhibits inhibitory activity against phospholipase A2 (phospholipaseA2).</p>Formula:C18H26O8Color and Shape:SolidMolecular weight:370.394Dioxolamycin
CAS:<p>Dioxolamycin is an antitumor antibiotic that inhibits the activity of L-1210 cells.</p>Formula:C11H15NO6Color and Shape:SolidMolecular weight:257.24Oxamicetin
CAS:<p>Oxamicetin is a nucleoside antibiotic with antibacterial and antimycobacterial properties.</p>Formula:C29H42N6O10Color and Shape:SolidMolecular weight:634.678NS2B/NS3-IN-4
CAS:<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Formula:C15H11NO4Color and Shape:SolidMolecular weight:269.25GG-43
<p>GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].</p>Formula:C21H21NO3Color and Shape:SolidMolecular weight:335.4Furaprevir
CAS:<p>Furaprevir is an HCV NS3/4A Inhibitor</p>Formula:C47H56N6O10SColor and Shape:SolidMolecular weight:897.05AEP-IN-1
<p>APE-IN-1, a potent AEP inhibitor (IC50: 89 nM), aids Alzheimer's diagnosis and drug research.</p>Formula:C18H27N3O3Color and Shape:SolidMolecular weight:333.43Glucoallosamidin B
CAS:<p>Glucoallosamidin B is a glycoside antibiotic identifiable in the Streptomyces species strain (Streptomycessp. SA-684). It functions as an inhibitor of chitinase activity. Experiments demonstrate that Glucoallosamidin B significantly inhibits the chitinase of Candida albicans (ATCC 10231), with an IC50 value of 0.8 μg/mL.</p>Formula:C25H42N4O14Color and Shape:SolidMolecular weight:622.619CU-2010
CAS:<p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>Formula:C37H42N6O6SColor and Shape:SolidMolecular weight:698.83CYP1B1-IN-2
<p>CYP1B1-IN-2 (compound 9j) is a highly potent and selective inhibitor of CYP1B1, a cytochrome P450 enzyme. It exhibits an IC50 value of 0.52 nM [1].</p>Formula:C20H11F3O2Color and Shape:SolidMolecular weight:340.3PD-1/PD-L1-IN-16
<p>PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.</p>Formula:C34H30N4O4Color and Shape:SolidMolecular weight:558.63KCa2 channel modulator 2
<p>Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.</p>Formula:C16H15ClFN5Color and Shape:SolidMolecular weight:331.78LPA5 antagonist 1
<p>LPA5 antagonist 1: selective, potent (IC50=32 nM), high brain permeability, studies inflammatory/neuropathic pain.</p>Formula:C28H26N2O4SColor and Shape:SolidMolecular weight:486.58DS69910557
<p>DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism & osteoporosis research.</p>Formula:C32H33Cl2FN4O3Color and Shape:SolidMolecular weight:611.53Lasonolide A
CAS:<p>Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.</p>Formula:C41H60O9Color and Shape:SolidMolecular weight:696.91Cbl-b-IN-1
CAS:<p>Cbl-b-IN-1 is a potent Cbl-b inhibitor (IC50 <100 nM) with potential anticancer activity for the study of intestinal inflammation.</p>Formula:C29H34N6O2Purity:99.68%Color and Shape:SolidMolecular weight:498.631Balanol
CAS:<p>Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.</p>Formula:C28H26N2O10Color and Shape:SolidMolecular weight:550.516"'-Deamino-6"'-hydroxyparomomycin I
CAS:<p>6"'-Deamino-6"'-hydroxyparomomycin I is an aminoglycoside antibiotic produced by Streptomyces rimosus forma paromomycinus A67 15, exhibiting activity against both Gram-positive and Gram-negative bacteria. It serves as an intermediate in the biosynthesis of paromomycin.</p>Formula:C23H44N4O15Color and Shape:SolidMolecular weight:616.613Chrymutasin B
CAS:<p>Chrymutasin B is a glycoside antitumor antibiotic known for its cytotoxic properties.</p>Formula:C32H31NO13Color and Shape:SolidMolecular weight:637.587Epoxyquinomicin B
CAS:<p>Epoxyquinomicin B is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus, with a minimum inhibitory concentration (MIC) of 6.25-12.5 µg/mL. It also shows cytotoxicity in cancer cells L1210, with an IC50 of 16.3 µg/mL. Additionally, Epoxyquinomicin B demonstrates anti-inflammatory effects on collagen-induced arthritis.</p>Formula:C14H11NO6Color and Shape:SolidMolecular weight:289.24Resorcinomycin A
CAS:<p>Resorcinomycin A is an antibiotic with potent antimycobacterial activity and relatively weaker activity against mycoplasma.</p>Formula:C14H20N4O5Color and Shape:SolidMolecular weight:324.332BAY-091
CAS:<p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>Formula:C26H21FN4O2Purity:97.66% - 99.23%Color and Shape:SoildMolecular weight:440.47D6808
<p>D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.</p>Formula:C30H25F3N6O2Color and Shape:SolidMolecular weight:558.55NPEC-caged-(S)-3,4-DCPG
CAS:<p>mGlu8a agonist</p>Formula:C19H16N2O10Purity:98%Color and Shape:SolidMolecular weight:432.34SGK1-IN-3
<p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>Formula:C23H20Cl2N6O3SColor and Shape:SolidMolecular weight:531.413'-O-Decarbamoylirumamycin
CAS:<p>3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.</p>Formula:C40H64O11Color and Shape:SolidMolecular weight:720.93Enacyloxin IIa
CAS:<p>Enacyloxin IIa (ENX IIa) is a polyene antibiotic with activity against both Gram-positive and Gram-negative bacteria, while exhibiting weak antifungal properties and no effect on yeast.</p>Formula:C33H45Cl2NO11Color and Shape:SolidMolecular weight:702.617Nocardicin B
CAS:<p>Nocardicin B was originally isolated from Nocardia uniformis subsp. tsugamanensis [ATCC 21806], showing weak antibacterial activity against Proteus and Corynebacterium species.</p>Formula:C23H24N4O9Color and Shape:SolidMolecular weight:500.46Baumycin C1
CAS:<p>Baumycin C1 is an antitumor antibiotic (antibiotic).</p>Formula:C28H29NO11Color and Shape:SolidMolecular weight:555.53Endophenazine C
CAS:<p>Endophenazine C is a type of phenazine antibiotic.</p>Formula:C19H20N2O2Color and Shape:SolidMolecular weight:308.37Phoslactomycin A
CAS:<p>Phoslactomycin A exhibits weaker activity against Gram-positive bacteria, yet it shows stronger efficacy against fungi.</p>Formula:C29H46NO10PColor and Shape:SolidMolecular weight:599.65Polyoxin F
CAS:<p>Polyoxin F is a nucleoside-type antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight disease.</p>Formula:C23H30N6O15Color and Shape:SolidMolecular weight:630.52Clavamycin C
CAS:<p>Clavamycin C exhibits significant antifungal activity against Candida species, which can be antagonized by dipeptides or tripeptides, though not by amino acids. It lacks antibacterial properties and does not inhibit β-lactamase activity.</p>Formula:C13H22N4O8Color and Shape:SolidMolecular weight:362.336Kinamycin A
CAS:<p>Kinamycin A possesses antibacterial and antimycobacterial properties, yet it exhibits reduced efficacy against Gram-negative bacteria.</p>Formula:C24H20N2O10Color and Shape:SolidMolecular weight:496.4233-O-Demethylmonensin B
CAS:<p>3-O-Demethylmonensin B is a polyether antibiotic produced by the bacterium *Streptomyces cinnamoneus* LO-63.</p>Formula:C34H58O11Color and Shape:SolidMolecular weight:642.82Fluoropolyoxin M
CAS:<p>Fluoropolyoxin M exhibits inhibitory activity against Escherichia coli and Enterococcus faecium.</p>Formula:C16H22FN5O11Color and Shape:SolidMolecular weight:479.371Trichodermin
CAS:<p>Trichodermin is a naturally occurring sesquiterpene antibiotic (antibiotic) and a powerful inhibitor of protein synthesis (protein synthesis). It binds to eukaryotic ribosomes, inhibiting protein translation by interacting with peptidyl transferase. Trichodermin suppresses oral cancer growth by inducing apoptosis (apoptosis)-related mitochondrial dysfunction and HDAC-2-mediated signaling. It exhibits potent antimicrobial activity against filamentous fungi, yeasts, and bacteria.</p>Formula:C17H24O4Color and Shape:SolidMolecular weight:292.37Elacestrant S enantiomer
<p>Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.</p>Formula:C30H38N2O2Purity:98%Color and Shape:SolidMolecular weight:458.63Carpetimycin A
CAS:<p>Carpetimycin A exhibits potent activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. It also acts as a strong inhibitor of β-lactamase.</p>Formula:C14H18N2O6SColor and Shape:SolidMolecular weight:342.368Resorthiomycin
CAS:<p>Resorthiomycin is an antitumor antibiotic that can inhibit L5178Y leukemia cells in vitro.</p>Formula:C14H20O4SColor and Shape:SolidMolecular weight:284.3713-Methoxy-2,5-toluquinone
CAS:<p>3-Methoxy-2,5-toluquinone is an antimicrobial agent that exhibits moderate antibacterial and antifungal properties.</p>Formula:C8H8O3Color and Shape:SolidMolecular weight:152.147Ezomycin D2
CAS:<p>Ezomycin D2 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia sclerotiorum and Botrytis cinerea. It helps control diseases like sclerotinia blight and gray mold in crops, as well as candidiasis.</p>Formula:C19H27N5O14Color and Shape:SolidMolecular weight:549.443Juglomycin A
CAS:<p>Juglomycin A exhibits broad-spectrum antibacterial and anti-mycobacterial activity and can inhibit Ehrlich ascites carcinoma in mice.</p>Formula:C14H10O6Color and Shape:SolidMolecular weight:274.226MV061194
CAS:<p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>Formula:C28H37N5O4SColor and Shape:SolidMolecular weight:539.692-Hydroxybutirosin
CAS:<p>2-Hydroxybutirosin is an antibiotic that can be found in Bacillus circulans.</p>Formula:C21H41N5O13Color and Shape:SolidMolecular weight:571.576Roselipin 1A
CAS:<p>Roselipin 1A inhibits diacylglycerol acyltransferase (DGAT) in rats.</p>Formula:C40H72O14Color and Shape:SolidMolecular weight:776.991Dihydrocompactin
CAS:<p>Dihydrocompactin is an antifungal metabolite derived from Penicillium citrinum and acts as an inhibitor of 3-hydroxy-3-methylglutaryl coenzyme-A reductase (HMG-CoA reductase).</p>Formula:C23H36O5Color and Shape:SolidMolecular weight:392.529Pilatin
CAS:<p>Pilatin exhibits inhibitory effects on both bacteria and fungi, and it strongly suppresses the incorporation of thymidine and uridine into DNA and RNA in Ehrlich ascites tumor cells.</p>Formula:C21H26O7Color and Shape:SolidMolecular weight:390.427Pacidamycin 5T
CAS:<p>Pacidamycin 5T is found in the bacterium Streptomyces coeruleorubidus [NRRL 18370].</p>Formula:C36H44N8O12Color and Shape:SolidMolecular weight:780.78YKL-04-085
CAS:<p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>Formula:C30H29N5O2Color and Shape:SolidMolecular weight:491.6Parimycin
CAS:<p>Parimycin exhibits activity against Gram-positive and Gram-negative bacteria, as well as tumors, but shows no efficacy against fungi. It inhibits tumor cells such as GXF 251L, H640, LXFA 629L, MCF-7, and MEXF 514L, with an IC70 range of 0.9-6.7 μg/mL.</p>Formula:C22H20O7Color and Shape:SolidMolecular weight:396.39Nebramycin Ⅳ
CAS:<p>Nebramycin IV is an aminoglycoside antibiotic with a broad antimicrobial spectrum, demonstrating significant efficacy against Gram-positive bacteria, Gram-negative bacteria, and mycobacteria.</p>Formula:C19H38N6O11Color and Shape:SolidMolecular weight:526.53916-Hydroxyroridin L-2
CAS:<p>16-Hydroxyroridin L-2 is a member of the verrucarin subclass of antibiotics with antitumor properties.</p>Formula:C29H38O10Color and Shape:SolidMolecular weight:546.606Bagremycin A
CAS:<p>Bagremycin A is identified in the actinobacterium strain Streptomyces (Streptomyces) Tu 4128. It exhibits weak antimicrobial activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.26910-Deoxymethymycin
CAS:<p>10-Deoxymethymycin (AntibioticYC 17) exhibits antibiotic activity against Gram-positive bacteria.</p>Formula:C25H43NO6Color and Shape:SolidMolecular weight:453.612Acremonol
CAS:<p>Acremonol exhibits activity against Gram-positive bacteria and fungi.</p>Formula:C14H18O6Color and Shape:SolidMolecular weight:282.29Micacocidin B
CAS:<p>Micacocidin B is an antibiotic that exhibits exceptional activity against Mycoplasma species.</p>Formula:C27H37CuN3O4S3Color and Shape:SolidMolecular weight:627.34Cytochalasin M
CAS:<p>Cytochalasin M exhibits various biological activities, including reversible inhibition of cytoplasmic division and the suppression of both endocytosis and exocytosis in macrophages.</p>Formula:C30H37NO6Color and Shape:SolidMolecular weight:507.618Fluvirucin A1
CAS:<p>Fluvirucin A1 is a novel antibiotic effective against the Influenza A virus.</p>Formula:C23H44N2O5Color and Shape:SolidMolecular weight:428.61Eulicin
CAS:<p>Eulicin is an antifungal agent that inhibits human immunodeficiency virus (HIV) infection and replication. It demonstrates broad-spectrum activity against both Gram-positive and Gram-negative bacteria and can be found in Streptomyces.</p>Formula:C24H52N8O2Color and Shape:SolidMolecular weight:484.7221-Hydroxyoxaunomycin
CAS:<p>1-Hydroxyoxaunomycin is an antibiotic that inhibits the growth of U210 cells as well as the synthesis of DNA and RNA, with IC50 values of 0.0005 μg/mL, 1.00 μg/mL, and 0.76 μg/mL, respectively.</p>Formula:C26H29NO11Color and Shape:SolidMolecular weight:531.509Gentamicin C2
CAS:<p>Gentamicin C2 is an aminoglycoside antibiotic.</p>Formula:C20H41N5O7Color and Shape:SolidMolecular weight:463.569Erabulenol A
CAS:<p>Erabulenol A is a cholesterol ester transfer protein (CETP) inhibitor, extracted from Penicillumsp.</p>Formula:C20H20O6Color and Shape:SolidMolecular weight:356.369Cycloleucomelone
CAS:<p>Cycloleucomelone is a secondary metabolite and a fungal pigment.</p>Formula:C18H10O7Color and Shape:SolidMolecular weight:338.268Herbimycin B
CAS:<p>Herbimycin B, an ansamycin antibiotic, functions as an inhibitor of Src family kinases. It exhibits herbicidal effects on most monocotyledonous and dicotyledonous plants and can inhibit the activity of tobacco mosaic virus (TMV), HeLa cells, and Ehrlich cells.</p>Formula:C29H40N2O7Color and Shape:SolidMolecular weight:528.637Exophilin A
CAS:<p>Exophilin A is an antibiotic that exhibits activity against Gram-positive bacteria.</p>Formula:C30H56O10Color and Shape:SolidMolecular weight:576.76Dykellic acid
CAS:<p>Dykellic acid is a RhoA inhibitor. It can suppress the migration and motility of B16 cells and inhibit the tubular formation of HUVECs. Dykellic acid shows potential for use in cancer research.</p>Formula:C14H16O4Color and Shape:SolidMolecular weight:248.274Diolmycin A1
CAS:<p>Diolmycin A1 is an antibiotic known for its anticoccidial activity.</p>Formula:C18H19NO3Color and Shape:SolidMolecular weight:297.348Queenslandon
CAS:<p>Queenslandon exhibits moderate antifungal activity against fungi such as Streptomyces, Penicillium, Aspergillus fumigatus, and Aspergillus flavus, and has no effect on bacteria.</p>Formula:C20H26O8Color and Shape:SolidMolecular weight:394.42Feigrisolide D
CAS:<p>Feigrisolide D is a lactone produced by Streptomyces griseus. It exhibits moderate inhibitory activity against 3α-hydroxysteroid dehydrogenase.</p>Formula:C22H38O7Color and Shape:SolidMolecular weight:414.5333-O-Demethylmonensin A
CAS:<p>3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).</p>Formula:C35H60O11Color and Shape:SolidMolecular weight:656.84Neoenactin A
CAS:<p>Neoenactin A exhibits potent activity against yeasts and filamentous fungi.</p>Formula:C19H36N2O5Color and Shape:SolidMolecular weight:372.5Monamycin H1
CAS:<p>Monamycin H1 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.</p>Formula:C34H56ClN7O8Color and Shape:SolidMolecular weight:726.30Enteromycin
CAS:<p>Enteromycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C6H8N2O5Color and Shape:SolidMolecular weight:188.138Bacithrocin B
CAS:<p>Bacithrocin B is a thrombin inhibitor that suppresses the activity of thrombin, Factor Xa, trypsin, and papain, with IC50 values of 84 μM, 17 μM, 1.7 μM, and 0.02 μM, respectively.</p>Formula:C19H29N5O3Color and Shape:SolidMolecular weight:375.46511-Deacetoxywortmannin
CAS:<p>11-Deacetoxywortmannin is an antibiotic with potent antibacterial and anti-inflammatory properties, and it also exhibits anti-edema effects.</p>Formula:C21H22O6Color and Shape:SolidMolecular weight:370.396PKCiota-IN-1
CAS:<p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>Formula:C25H22FN5OColor and Shape:SolidMolecular weight:427.47Dehatrine
CAS:<p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>Formula:C37H38N2O6Color and Shape:SolidMolecular weight:606.71Ezomycin A2
CAS:<p>Ezomycin A2 is an antifungal antibiotic. It is primarily effective against plant pathogens such as Sclerotinia and Botrytis, showing efficacy in controlling crop diseases like sclerotinia rot, botrytis blight, and candidiasis.</p>Formula:C19H26N6O12Color and Shape:SolidMolecular weight:530.443Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Formula:C24H26O8Color and Shape:SolidMolecular weight:442.46Cephemimycin
CAS:<p>Cephemimycin exhibits mild antibacterial and antifungal activity.</p>Formula:C16H22N4O9SColor and Shape:SolidMolecular weight:446.432Antimalarial agent 3
<p>Antimalarial agent 3 has a potent IC50 of 0.035 μM against Plasmodium and high selectivity for mammalian cells.</p>Formula:C15H16BrN3O2Color and Shape:SolidMolecular weight:350.21Chuangxinmycin
CAS:<p>Chuangxinmycin is an antibiotic that can be isolated from Actinoplanes tsinanensis CPCC 200056. It exhibits antibacterial activity both in vitro and in vivo, making it useful for research related to infections.</p>Formula:C12H11NO2SColor and Shape:SolidMolecular weight:233.2862-Hydroxygentamicin B
CAS:<p>2-Hydroxygentamicin B is an aminoglycoside antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C19H38N4O11Color and Shape:SolidMolecular weight:498.525Nafarelin acetate hydrate
CAS:<p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>Formula:C66H83N17O13·xC2H4O2·xH2OColor and Shape:SolidMolecular weight:1400.563NCI-006
CAS:<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Formula:C31H24F2N4O4S3Color and Shape:SolidMolecular weight:650.74Glidobactin G
CAS:<p>Glidobactin G is an antitumor antibiotic with activity against pathogenic fungi and yeasts. Additionally, Glidobactin G prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Formula:C27H44N4O7Color and Shape:SolidMolecular weight:536.6619-cis-13,14-Dihydroretinoic acid
CAS:<p>9-cis-13,14-Dihydroretinoic acid (9CDHRA) is a selective retinoid X receptor (RXR) agonist with a Kd of 90 nM. It can ameliorate memory deficits caused by impaired RXR signaling in vivo. This compound shows potential for research in the fields of neuroscience and metabolic diseases.</p>Formula:C20H30O2Color and Shape:SolidMolecular weight:302.451Bis(N-methylthioformohydroxamate)nickel (II)
CAS:<p>Bis(N-methylthioformohydroxamate)nickel (II) is a nickel-containing antibiotic that exhibits significant activity against both Gram-positive and Gram-negative bacteria, as well as antitumor properties.</p>Formula:C4H8N2NiO2S2Color and Shape:SolidMolecular weight:238.942Enamidonin
CAS:<p>Enamidonin is a lipopeptide antibiotic. It inhibits EGF-dependent [3H] thymidine incorporation in Balb/MK cells with an IC50 of 10 μg/mL and can restore the transformed SRCTS-NRK cells to their normal flat shape with an ED50 of 10 μg/mL. It exhibits no antibacterial activity.</p>Formula:C37H51N7O7Color and Shape:SolidMolecular weight:705.844Deflectin 1a
CAS:<p>Deflectin 1a is an antibiotic with activities such as lysing bacteria, lysing red blood cells, and inhibiting Ehrlich ascites cancer cells. However, its effectiveness can be neutralized by the addition of serum or serum albumin.</p>Formula:C21H24O5Color and Shape:SolidMolecular weight:356.412Pyloricidin A
CAS:<p>Pyloricidin A is an antibiotic effective against Helicobacter pylori, produced by Bacillus sp. HC-70. It exhibits strong anti-Helicobacter pylori activity and shows no efficacy against other bacteria or yeasts.</p>Formula:C31H51N5O10Color and Shape:SolidMolecular weight:653.76Acrylamidine
CAS:<p>Acrylamidine exhibits weak antifungal and yeast activity.</p>Formula:C3H6N2Color and Shape:SolidMolecular weight:70.09SX 3202
CAS:<p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>Formula:C17H11BrFN3O4Color and Shape:SolidMolecular weight:420.19Leu-AMS R enantiomer
CAS:<p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>Formula:C16H25N7O7SPurity:98%Color and Shape:SolidMolecular weight:459.48BSc5367
CAS:<p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>Formula:C20H15N3O2Color and Shape:SoildMolecular weight:329.35Antiproliferative agent-3
<p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>Formula:C11H12N2O5SColor and Shape:SolidMolecular weight:284.29PD-1-IN-17 TFA
<p>PD-1-IN-17 TFA is a potent PD-1 inhibitor, blocking 92% of splenocyte growth at 100 nM.</p>Formula:C15H23F3N6O9Color and Shape:SolidMolecular weight:488.37Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formula:C27H25FN6O2Color and Shape:SolidMolecular weight:484.52MC4355
<p>MC4355 is a dual inhibitor of EZH2 and histone deacetylase (HDAC).</p>Formula:C30H36N4O5Color and Shape:SolidMolecular weight:532.63AT1R antagonist 2
<p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>Formula:C29H37N5O4S2Color and Shape:SolidMolecular weight:583.77P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Formula:C21H16F3N9Color and Shape:SolidMolecular weight:451.42PrCP-7414
CAS:<p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>Formula:C31H33Cl2N5O2Color and Shape:SolidMolecular weight:578.53DD04107
CAS:<p>DD04107 inhibits α-CGRP release, targets Synaptotagmin 1 in sensory neurons.</p>Formula:C48H88N14O12SColor and Shape:SolidMolecular weight:1085.36MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formula:C34H53N15O6Color and Shape:SolidMolecular weight:767.88Hynapene C
CAS:<p>Hynapene C exhibits an inhibitory minimum inhibitory concentration (MIC) of 34.7 μM against Eimeria acervulina.</p>Formula:C18H24O3Color and Shape:SolidMolecular weight:288.381Curvulic acid
CAS:<p>Curvulic acid exhibits relatively weak activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C11H12O6Color and Shape:SolidMolecular weight:240.209Carzinophillin A
CAS:<p>Carzinophillin A exhibits inhibitory effects on both ascites carcinoma and Yoshida sarcoma.</p>Formula:C31H33N3O11Color and Shape:SolidMolecular weight:623.607rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Color and Shape:SolidMolecular weight:504.38Carpetimycin D
CAS:<p>Carpetimycin D exhibits potent activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. Additionally, Carpetimycin D strongly inhibits β-lactamase.</p>Formula:C14H20N2O9S2Color and Shape:SolidMolecular weight:424.447Darlucin A
CAS:<p>Darlucin A exhibits both antibacterial and antifungal properties, accompanied by mild cytotoxicity.</p>Formula:C19H16N2O3Color and Shape:SolidMolecular weight:320.342Oximidine Ⅲ
CAS:<p>Oximidine III is an antitumor antibiotic that selectively inhibits the growth of rat fibroblast 3Y1 cells and induces mutations in various tumor genes. The inhibitory effects of Oximidine III on vH-ras-3Y1, v-src-3Y1 cells, and normal 3Y1 cells have IC50 values of 14 nM, 4.5 nM, and 140 nM, respectively. Additionally, Oximidine III arrests cells with RAS or SRC mutations in the G1 phase of the cell cycle and increases the expression of p21WAF1.</p>Formula:C23H24N2O6Color and Shape:SolidMolecular weight:424.45Exfoliamycin
CAS:<p>Exfoliamycin is a naphthoquinone antibiotic found in the Streptomyces strain Exfoliamycin Tu 1424, and it exhibits activity against Gram-positive bacteria.</p>Formula:C22H26O9Color and Shape:SolidMolecular weight:434.436Fusarin C
CAS:<p>Fusarin C is a mutagenic compound found in strains of the Fusarium genus.</p>Formula:C23H29NO7Color and Shape:SolidMolecular weight:431.479Dienomycin B
CAS:<p>Dienomycin B exhibits mild antibacterial activity.</p>Formula:C18H23NO2Color and Shape:SolidMolecular weight:285.38Phoslactomycin B
CAS:<p>Phoslactomycin B exhibits relatively weak activity against Gram-positive bacteria but demonstrates stronger activity against fungi.</p>Formula:C25H40NO8PColor and Shape:SolidMolecular weight:513.5614-Hydroxyphlebiarubrone
CAS:<p>4-Hydroxyphlebiarubrone is a quinone antibiotic. It exhibits weaker resistance against Gram-negative bacteria and possesses cytotoxic properties.</p>Formula:C19H12O5Color and Shape:SolidMolecular weight:320.30Myxovirescin A
CAS:<p>Myxovirescin A is an antibiotic with activity against Gram-negative bacteria.</p>Formula:C35H61NO8Color and Shape:SolidMolecular weight:623.861
