Other Inhibitors
This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.
Found 37902 products of "Other Inhibitors"
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MDL-100173
CAS:<p>MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.</p>Formula:C24H26N2O4SColor and Shape:SolidMolecular weight:438.54MV061194
CAS:<p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>Formula:C28H37N5O4SColor and Shape:SolidMolecular weight:539.69NCI-006
CAS:<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Formula:C31H24F2N4O4S3Color and Shape:SolidMolecular weight:650.74MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66Pyruvate Carboxylase-IN-2
CAS:<p>Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.</p>Formula:C21H22O8Color and Shape:SolidMolecular weight:402.39Antitumor agent-47
<p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>Formula:C30H27NO11Color and Shape:SolidMolecular weight:577.54Flusoxolol
CAS:<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formula:C22H30FNO4Color and Shape:SolidMolecular weight:391.48Iroxanadine hydrobromide
CAS:<p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>Formula:C14H21BrN4OColor and Shape:SolidMolecular weight:341.25SP inhibitor 1
<p>SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.</p>Formula:C36H38N2O2Color and Shape:SolidMolecular weight:530.7DSP-6952
CAS:<p>DSP-6952 is a 5-HT4 receptor partial agonist, inhibiting visceral hypersensitivity and ameliorating gastrointestinal dysfunction.</p>Formula:C21H32BrClN4O5Color and Shape:SolidMolecular weight:535.86G12Si-1
<p>G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.</p>Formula:C29H32ClN5O3Color and Shape:SolidMolecular weight:534.05PAD-IN-2
CAS:<p>PAD-IN-2, potent PAD4 inhibitor, IC50 <1 μM; targets autoimmune/cancer disorders.</p>Formula:C27H28ClN5O2Color and Shape:SolidMolecular weight:490NA 382
CAS:<p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>Formula:C31H28N4O6Color and Shape:SolidMolecular weight:552.58AZD-3409
CAS:<p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>Formula:C34H41FN4O4S2Color and Shape:SolidMolecular weight:652.84XN methyl pyrazole
<p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>Formula:C22H24N2O4Color and Shape:SolidMolecular weight:380.44TY 11345
CAS:<p>TY 11345 is a proton pump inhibitor.</p>Formula:C18H18N3NaO2SColor and Shape:SolidMolecular weight:363.41MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formula:C34H53N15O6Color and Shape:SolidMolecular weight:767.88eIF4A3-IN-6
CAS:<p>eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)</p>Formula:C26H25N3O5Color and Shape:SolidMolecular weight:459.49PrCP-7414
CAS:<p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>Formula:C31H33Cl2N5O2Color and Shape:SolidMolecular weight:578.53AT1R antagonist 2
<p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>Formula:C29H37N5O4S2Color and Shape:SolidMolecular weight:583.77Antiproliferative agent-3
<p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>Formula:C11H12N2O5SColor and Shape:SolidMolecular weight:284.29Cicaprost
CAS:<p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>Formula:C22H30O5Color and Shape:SolidMolecular weight:374.47PNU-140457
CAS:<p>PNU-140457 is a bio-active chemical.</p>Formula:C14H14FN5O3Color and Shape:SolidMolecular weight:319.29KDOAM-25 trihydrochloride (2230731-99-2 free base)
<p>KDOAM-25 trihydrochloride, a selective KDM5 inhibitor (IC50: 19-71 nM), boosts H3K4 methylation and hinders MM1S cell growth.</p>Formula:C15H28Cl3N5O2Purity:98%Color and Shape:SolidMolecular weight:416.77NPEC-caged-(S)-3,4-DCPG
CAS:<p>mGlu8a agonist</p>Formula:C19H16N2O10Purity:98%Color and Shape:SolidMolecular weight:432.349-Hydroxyoudemansin A
CAS:<p>9-Hydroxyoudemansin A exhibits antifungal activity with a minimum inhibitory concentration (MIC) of 12.5 μg/mL against Saccharomyces cerevisiae. It shows resistance to fungi such as Candida albicans, Rhodotorula, Penicillium, and Streptomyces, with MIC values all exceeding 50 μg/mL. It does not possess antibacterial properties.</p>Formula:C16H20O4Color and Shape:SolidMolecular weight:276.328Anticancer agent 78
<p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>Formula:C19H14BrNO4Color and Shape:SolidMolecular weight:400.22GRPR antagonist-1
<p>GRPR antagonist-1 targets GRPR, kills specific cancer cells (e.g., PC3, Pan02, HGC-27), and promotes apoptosis by modulating Bcl-2 and Bax.</p>Formula:C29H33F3N4O4Color and Shape:SolidMolecular weight:558.59SCP1-IN-2
<p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>Formula:C19H17F3N2O6S2Color and Shape:SolidMolecular weight:490.478,9-Epoxyeicosatrienoic acid
CAS:<p>8,9-Epoxyeicosatrienoic acid offers unique protective effects on the glomerulus. It inhibits the increase in glomerular albumin permeability caused by circulating permeability factors (FSPF). Additionally, 8,9-Epoxyeicosatrienoic acid is used in research related to glomerular dysfunction.</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47(±)-HIP-B
CAS:<p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>Formula:C6H8N2O4Purity:98%Color and Shape:SolidMolecular weight:172.14Erizepine
CAS:<p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>Formula:C20H22N2Color and Shape:SolidMolecular weight:290.4LK-732
CAS:<p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>Formula:C25H29N5O3SColor and Shape:SolidMolecular weight:479.594-Chloropyridine
CAS:<p>4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.</p>Formula:C5H4ClNColor and Shape:SolidMolecular weight:113.55VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Formula:C21H14ClN3O2Color and Shape:SolidMolecular weight:375.81SORT1-IN-3
CAS:<p>SORT1-IN-3 (compound 5) is a SORT1 inhibitor characterized by its ability to permeate the blood-brain barrier.</p>Formula:C16H26ClNO3Color and Shape:SolidMolecular weight:315.84Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formula:C24H26N2O13Color and Shape:SolidMolecular weight:550.47UNC7467
CAS:<p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>Formula:C20H13NO3Purity:98.28% - 98.64%Color and Shape:SoildMolecular weight:315.32Tandutinib (MLN518) HCl
Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.Formula:C31H43ClN6O4Purity:98%Color and Shape:SolidMolecular weight:599.16MRS2279
CAS:<p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>Formula:C13H18ClN5O8P2Purity:98%Color and Shape:SolidMolecular weight:469.71Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formula:C32H33N5O4Purity:98%Color and Shape:SolidMolecular weight:551.64U 80215
CAS:<p>U 80215 is an enzyme-competitive inhibitor.</p>Formula:C42H60N8O6SColor and Shape:SolidMolecular weight:805.04Antitumor agent-65
CAS:<p>Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.</p>Formula:C18H17NO10Color and Shape:SolidMolecular weight:407.33MU1656
CAS:<p>MU1656 is a selective inhibitor of histone methyltransferase DOT1L, which significantly inhibits cancer cell proliferation in hematological malignancies.</p>Formula:C32H45N7O2Purity:96.92%Color and Shape:SolidMolecular weight:559.75Glucosylceramide synthase-IN-3
<p>Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.</p>Formula:C21H20FN3O3Color and Shape:SolidMolecular weight:381.4GNE-616
CAS:<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formula:C24H23F4N5O3SPurity:98%Color and Shape:SolidMolecular weight:537.53Fostriecin (free base)
CAS:<p>Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.</p>Formula:C19H27O9PColor and Shape:SolidMolecular weight:430.39FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formula:C21H26FN5O2Purity:98%Color and Shape:SolidMolecular weight:399.46BMS-986120
CAS:BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.Formula:C23H23N5O5S2Color and Shape:SolidMolecular weight:513.59Glyphosate-trimesium
CAS:<p>Glyphosate-trimesium is a herbicide.</p>Formula:C6H16NO5PSColor and Shape:SolidMolecular weight:245.23
