Protacs and Impurities

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products per page. 259 products on this category.

Product data	Purity	Price range	Estimated delivery
PROTAC AR Degrader-4 TFA REF: TM-T73726	- - -	To inquire	Tue 03 Dec 24
PROTAC PIN1 degrader-1 REF: TM-T200020CAS: 3038591-59-9	- - -	To inquire	Tue 03 Dec 24
DZ-837 REF: TM-T200170	- - -	To inquire	Tue 03 Dec 24
PROTAC MLKL Degrader-2 REF: TM-T200218	- - -	To inquire	Tue 03 Dec 24
PROTAC CYP1B1 degrader-1 REF: TM-T74519CAS: 2411389-67-6	- - -	To inquire	Tue 03 Dec 24
ACBI2 REF: TM-T74984CAS: 2913161-19-8	- - -	To inquire	Tue 03 Dec 24
PROTAC IRAK4 degrader-3 REF: TM-T39920CAS: 2374122-43-5	- - -	To inquire	Tue 03 Dec 24
SHP2-D26 REF: TM-T40121CAS: 2458219-65-1	- - -	1,422.00 €	Tue 03 Dec 24
CMP98 REF: TM-T39750CAS: 2244684-50-0	- - -	791.00 €	Tue 03 Dec 24
MS21 REF: TM-T39929CAS: 2376137-05-0	- - -	1,422.00 €	Tue 03 Dec 24
U7D-1 REF: TM-T74682	- - -	To inquire	Tue 03 Dec 24
CRBN-6-5-5-VHL REF: TM-T35479	- - -	298.00 €	Tue 03 Dec 24
MD-222 REF: TM-T37041CAS: 2136246-72-3	- - -	738.00 €~2,675.00 €	Tue 03 Dec 24
PROTAC STING Degrader-1 REF: TM-T74896CAS: 2762552-74-7	- - -	315.00 €	Tue 03 Dec 24
INY-03-041 trihydrochloride REF: TM-T74001	- - -	To inquire	Tue 03 Dec 24
PROTAC BET Degrader-10 REF: TM-T39374CAS: 1957234-97-7	- - -	To inquire	Tue 03 Dec 24
PP-C8 REF: TM-T74359	- - -	To inquire	Tue 03 Dec 24
PROTAC RIPK degrader-6 REF: TM-T36243CAS: 2089205-64-9	- - -	To inquire	Tue 03 Dec 24
PROTAC AR-V7 degrader-1 REF: TM-T74410CAS: 2767440-24-2	- - -	To inquire	Tue 03 Dec 24
MS170 REF: TM-T39928CAS: 2376136-61-5	- - -	932.00 €	Tue 03 Dec 24

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PROTAC AR Degrader-4 TFA

PROTAC AR Degrader-4: IAP ligand, linker, AR binder; it's a SNIPER that degrades AR non-genetically.

Formula:

C₄₅H₆₈F₃N₃O₁₁

Color and Shape:

Liquid

Molecular weight:

884.03

Ref: TM-T73726

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC PIN1 degrader-1

CAS:3038591-59-9

PROTAC PIN1 degrader-1, a targeted PROTAC for PIN1, effectively degrades PIN1 protein in MDA-MB-468 triple-negative …

Formula:

C₅₁H₅₂N₁₀O₇

Color and Shape:

Liquid

Molecular weight:

917.02

Ref: TM-T200020

10mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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DZ-837

DZ-837 is a PROTAC that targets the BCL6 protein. The composition of DZ-837 includes the …

Formula:

C₄₂H₄₄FN₉O₇S

Color and Shape:

Liquid

Molecular weight:

837.92

Ref: TM-T200170

10mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC MLKL Degrader-2

PROTAC MLKL Degrader-2, a PROTAC that targets MLKL (Mixed Lineage Kinase), incorporates the PROTAC target …

Formula:

C₃₆H₃₅N₉O₉S

Color and Shape:

Liquid

Molecular weight:

769.78

Ref: TM-T200218

10mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC CYP1B1 degrader-1

CAS:2411389-67-6

Compound 6C, a PROTAC degrader, targets CYP1B1 with IC50s (95.1 nM CYP1B1, 9838.6 nM CYP1A2) …

Formula:

C₄₃H₃₉N₅O₁₀

Color and Shape:

Liquid

Molecular weight:

785.8

Ref: TM-T74519

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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ACBI2

CAS:2913161-19-8

ACBI2: potent, oral VHL PROTAC, EC50=7nM; degrades SMARCA2, DC50=1nM in RKO cells; for lung cancer …

Formula:

C₅₆H₆₈BrFN₈O₅S

Color and Shape:

Liquid

Molecular weight:

1064.16

Ref: TM-T74984

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC IRAK4 degrader-3

CAS:2374122-43-5

PROTAC IRAK4 degrader-3 is a PROTAC-induced IRAK4 degrader based on von Hippel-Lindau.

Formula:

C₅₇H₆₈FN₁₁O₈S

Color and Shape:

Solid

Molecular weight:

1086.3

Ref: TM-T39920

100mg		To inquire
500mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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SHP2-D26

CAS:2458219-65-1

SHP2-D26: potent SHP2 degrader binding VHL-1/SHP2, neddylation & proteasome-dependent.

Formula:

C₅₆H₇₉ClN₁₂O₆S₂

Color and Shape:

Liquid

Molecular weight:

1115.9

Ref: TM-T40121

25mg 1,422.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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CMP98

CAS:2244684-50-0

CMP98, a PROTAC, fails to degrade VHL; useful as CM11 negative control; contains two active …

Formula:

C₅₈H₈₂N₈O₁₄S₂

Color and Shape:

Liquid

Molecular weight:

1179.45

Ref: TM-T39750

10mg 791.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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MS21

CAS:2376137-05-0

MS21 is a unique AKT degrader that selectively hampers the proliferation of cancers with mutations …

Formula:

C₅₈H₇₉ClN₁₂O₆S

Color and Shape:

Liquid

Molecular weight:

1107.86

Ref: TM-T39929

25mg 1,422.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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U7D-1

U7D-1: First-class USP7 PROTAC degrader, DC50 33 nM, anticancer, induces apoptosis in Jeko-1.

Formula:

C₅₃H₆₅N₉O₇

Color and Shape:

Liquid

Molecular weight:

940.14

Ref: TM-T74682

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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CRBN-6-5-5-VHL

Potent cereblon degrader with a DC50 of 1.5 nM, fully degrades cereblon in MM1S cells; …

Ref: TM-T35479

5mg 298.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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MD-222

CAS:2136246-72-3

MD-222: a first-in-class, highly potent PROTAC that degrades MDM2, activates p53, and exhibits anticancer properties.

Formula:

C₄₈H₄₇Cl₂FN₆O₆

Color and Shape:

Solid

Molecular weight:

893.84

Ref: TM-T37041

5mg		738.00 €
10mg		1,272.00 €
25mg		2,675.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC STING Degrader-1

CAS:2762552-74-7

PROTAC STING Degrader-1 (Compound SP23) is a STING-targeted PROTAC degrader exhibiting a DC50 of 3.2 …

Formula:

C₃₄H₃₃N₇O₁₀

Color and Shape:

Liquid

Molecular weight:

699.67

Ref: TM-T74896

1mg 315.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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INY-03-041 trihydrochloride

INY-03-041 trihydrochloride: potent, selective PROTAC AKT degrader; combines Ipatasertib and Lenalidomide; IC50s: AKT1 (2.0 nM), …

Formula:

C₄₄H₅₉Cl₄N₇O₅

Color and Shape:

Liquid

Molecular weight:

907.8

Ref: TM-T74001

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC BET Degrader-10

CAS:1957234-97-7

PROTAC BET Degrader-10 targets and degrades BRD4 with a DC50 of 49 nM, using Cereblon …

Formula:

C₃₉H₃₉ClN₈O₆S

Color and Shape:

Liquid

Molecular weight:

783.3

Ref: TM-T39374

5mg		233.00 €
10mg		373.00 €
25mg		699.00 €
50mg		1,039.00 €
100mg		1,544.00 €
200mg		To inquire
500mg		To inquire
1mL*10mM (DMSO)		322.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PP-C8

PP-C8: PROTAC CDK12-Cyclin K degrader with DC50s 416/412 nM; synergizes with PARP inhibitor against TNBC.

Formula:

C₄₃H₅₁FN₁₂O₇

Color and Shape:

Liquid

Molecular weight:

866.94

Ref: TM-T74359

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC RIPK degrader-6

CAS:2089205-64-9

PROTAC RIPK degrader-6 (example 1) is a PROTAC designed for the targeted degradation of RIP …

Formula:

C₄₃H₄₈N₆O₁₁S₂

Color and Shape:

Liquid

Molecular weight:

889.01

Ref: TM-T36243

5mg		450.00 €
10mg		653.00 €
25mg		1,198.00 €
1mL*10mM (DMSO)		721.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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PROTAC AR-V7 degrader-1

CAS:2767440-24-2

Potent, oral AR-V7 degrader (Compound 6); DC50: 0.32µM; targets AR-DBD via VHL E3; EC50: 0.88µM …

Formula:

C₄₁H₅₂N₆O₆S₂

Color and Shape:

Liquid

Molecular weight:

789.02

Ref: TM-T74410

5mg		To inquire
50mg		To inquire

Estimated delivery in United States, on Tuesday 3 Dec 2024

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MS170

CAS:2376136-61-5

MS170, specific PROTAC AKT degrader, potent with DC 50 of 32 nM, binds AKT1/2/3 with …

Formula:

C₄₅H₅₆ClN₉O₇

Color and Shape:

Solid

Molecular weight:

870.45

Ref: TM-T39928

5mg 932.00 €

Estimated delivery in United States, on Tuesday 3 Dec 2024

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