G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5800 products of "G-protein Coupled Receptors and 7-TM Receptors"

Purity (%)

100

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Fluphenazine decanoate
CAS:
- 5002-47-1
Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.
Formula:C₃₂H₄₄F₃N₃O₂S
Purity:98.14%
Color and Shape:Solid
Molecular weight:591.77
Ref: TM-T7943
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Aripiprazole monohydrate
CAS:
- 851220-85-4
Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.
Formula:C₂₃H₂₉Cl₂N₃O₃
Color and Shape:Solid
Molecular weight:466.4
Ref: TM-T62982
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Ziprasidone mesylate
CAS:
- 185021-64-1
Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.
Formula:C₂₂H₂₅ClN₄O₄S₂
Color and Shape:Solid
Molecular weight:509.04
Ref: TM-T63504
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Metergoline
CAS:
- 17692-51-2
Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.
Formula:C₂₅H₂₉N₃O₂
Purity:99.83% - 99.97%
Color and Shape:Solid
Molecular weight:403.52
Ref: TM-T4008
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SDZ WAG 994
CAS:
- 130714-47-5
SDZ WAG 994 is an A1 adenosine receptor agonist.
Formula:C₁₇H₂₅N₅O₄
Purity:99.82%
Color and Shape:Solid
Molecular weight:363.41
Ref: TM-T23347
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Ciproxifan maleate
CAS:
- 184025-19-2
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity
Formula:C₂₀H₂₂N₂O₆
Purity:99.39%
Color and Shape:Solid
Molecular weight:386.4
Ref: TM-T2004
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Desvenlafaxine succinate hydrate
CAS:
- 386750-22-7
Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
Formula:C₂₀H₃₃NO₇
Purity:99.26%
Color and Shape:White Crystalline Powde
Molecular weight:399.48
Ref: TM-T6188
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Epinastine hydrochloride
CAS:
- 108929-04-0
Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
Formula:C₁₆H₁₅N₃·HCl
Purity:99.26% - 99.62%
Color and Shape:White Solid
Molecular weight:285.77
Ref: TM-T6488
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1-Oleoyl lysophosphatidic acid sodium
CAS:
- 325465-93-8
1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2
Formula:C₂₁H₄₀O₇P·Na
Purity:98.75% - 99.24%
Color and Shape:Solid
Molecular weight:458.51
Ref: TM-T21654
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Flibanserin
CAS:
- 167933-07-5
Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:C₂₀H₂₁F₃N₄O
Purity:99.37% - 99.93%
Color and Shape:White Powder
Molecular weight:390.4
Ref: TM-T4297
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BAY 41-2272
CAS:
- 256376-24-6
BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.
Formula:C₂₀H₁₇FN₆
Purity:99.54%
Color and Shape:Solid
Molecular weight:360.39
Ref: TM-T6775
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2-Methoxyidazoxan monohydrochloride
CAS:
- 109544-45-8
L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.
Formula:C₁₂H₁₄N₂O₃·HCl
Purity:98.99%
Color and Shape:Solid
Molecular weight:270.72
Ref: TM-T23283
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SB-200646
CAS:
- 143797-63-1
SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
Formula:C₁₅H₁₄N₄O
Purity:99.61%
Color and Shape:Solid
Molecular weight:266.3
Ref: TM-T8357
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BMS 182874 hydrochloride
CAS:
- 1215703-04-0
BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.
Formula:C₁₇H₂₀ClN₃O₃S
Purity:97.01%
Color and Shape:Solid
Molecular weight:381.88
Ref: TM-T21790
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nifenalol.HCl
CAS:
- 5704-60-9
Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.
Formula:C₁₁H₁₇ClN₂O₃
Purity:99.96%
Color and Shape:Solid
Molecular weight:260.72
Ref: TM-T8663
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ICI 118,551 hydrochloride
CAS:
- 72795-01-8
ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3
Formula:C₁₇H₂₈ClNO₂
Purity:99.296% - 99.76%
Color and Shape:Solid
Molecular weight:313.86
Ref: TM-T11607
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Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.
Formula:C₁₂₈H₂₁₉N₄₅O₃₆S
Purity:94.61%
Color and Shape:Solid
Molecular weight:2996.45
Ref: TM-TP1045L
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AZD1283
CAS:
- 919351-41-0
AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).
Formula:C₂₃H₂₆N₄O₅S
Purity:98.37% - 99.63%
Color and Shape:Solid
Molecular weight:470.54
Ref: TM-T3536
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GW627368
CAS:
- 439288-66-1
GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.
Formula:C₃₀H₂₈N₂O₆S
Purity:99.75% - 99.92%
Color and Shape:Solid
Molecular weight:544.62
Ref: TM-T1978
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Alimemazine hemitartrate
CAS:
- 4330-99-8
Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.
Formula:C₁₈H₂₂N₂SC₄H₆O₆
Purity:98.16% - 99.69%
Color and Shape:Solid
Molecular weight:448.53
Ref: TM-T3282